Automated design of multi-target ligands by generative deep learning
Isigkeit, Laura, Hörmann, Tim, Schallmayer, Espen, Scholz, Katharina, Lillich, Felix F., Ehrler, Johanna H. M., Hufnagel, Benedikt, Büchner, Jasmin, Marschner, Julian A., Pabel, Jörg, Proschak, Ewgenij, Merk, Daniel
Published in Nature communications (11.09.2024)
Published in Nature communications (11.09.2024)
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Photosensitization enables Pauson-Khand-type reactions with nitrenes
Li, Fang, Zhu, W. Felix, Empel, Claire, Datsenko, Oleksandr, Kumar, Adarsh, Xu, Yameng, Ehrler, Johanna H. M., Atodiresei, Iuliana, Knapp, Stefan, Mykhailiuk, Pavel K., Proschak, Ewgenij, Koenigs, Rene M.
Published in Science (American Association for the Advancement of Science) (02.02.2024)
Published in Science (American Association for the Advancement of Science) (02.02.2024)
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Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator
Dötsch, Lara, Davies, Caitlin, Hennes, Elisabeth, Schönfeld, Julia, Kumar, Adarsh, Guita, Celine Da Cruz Lopes, Ehrler, Johanna H.M., Hiesinger, Kerstin, Thavam, Sasikala, Janning, Petra, Sievers, Sonja, Knapp, Stefan, Proschak, Ewgenij, Ziegler, Slava, Waldmann, Herbert
Published in Journal of medicinal chemistry (28.03.2024)
Published in Journal of medicinal chemistry (28.03.2024)
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Compilation and evaluation of a fatty acid mimetics screening library
Ehrler, Johanna H.M., Brunst, Steffen, Tjaden, Amelie, Kilu, Whitney, Heering, Jan, Hernandez-Olmos, Victor, Krommes, Andre, Kramer, Jan S., Steinhilber, Dieter, Schubert-Zsilavecz, Manfred, Müller, Susanne, Merk, Daniel, Proschak, Ewgenij
Published in Biochemical pharmacology (01.10.2022)
Published in Biochemical pharmacology (01.10.2022)
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Development of a Potent and Selective G2A (GPR132) Agonist
Hernandez-Olmos, Victor, Heering, Jan, Marinescu, Beatrice, Schermeng, Tina, Ivanov, Vladimir V., Moroz, Yurii S., Nevermann, Sheila, Mathes, Marius, Ehrler, Johanna H. M., Alnouri, Mohamad Wessam, Wolf, Markus, Haydo, Alicia S., Schmachtel, Tessa, Zaliani, Andrea, Höfner, Georg, Kaiser, Astrid, Schubert-Zsilavecz, Manfred, Beck-Sickinger, Annette G., Offermanns, Stefan, Gribbon, Philipp, Rieger, Michael A., Merk, Daniel, Sisignano, Marco, Steinhilber, Dieter, Proschak, Ewgenij
Published in Journal of medicinal chemistry (11.07.2024)
Published in Journal of medicinal chemistry (11.07.2024)
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Designing a Small Fluorescent Inhibitor to Investigate Soluble Epoxide Hydrolase Engagement in Living Cells
Brunst, Steffen, Schönfeld, Julia, Breunig, Peter, Burgers, Luisa D., DeMeglio, Murphy, Ehrler, Johanna H. M., Lillich, Felix F., Weizel, Lilia, Hefendehl, Jasmin K., Fürst, Robert, Proschak, Ewgenij, Hiesinger, Kerstin
Published in ACS medicinal chemistry letters (14.07.2022)
Published in ACS medicinal chemistry letters (14.07.2022)
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