Synthesis and evaluation of chemical linchpins for highly selective CK2α targeting
Greco, Francesco A., Krämer, Andreas, Wahl, Laurenz, Elson, Lewis, Ehret, Theresa A.L., Gerninghaus, Joshua, Möckel, Janina, Müller, Susanne, Hanke, Thomas, Knapp, Stefan
Published in European journal of medicinal chemistry (05.10.2024)
Published in European journal of medicinal chemistry (05.10.2024)
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Back-Pocket Optimization of 2‑Aminopyrimidine-Based Macrocycles Leads to Potent EPHA2/GAK Kinase Inhibitors
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Published in Journal of medicinal chemistry (08.08.2024)
Published in Journal of medicinal chemistry (08.08.2024)
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Journal Article
Structural Basis for Highly Selective Class II Alpha Phosphoinositide-3-Kinase Inhibition
Kücükdisli, Murat, Bel-Abed, Hassen, Cirillo, Davide, Lo, Wen-Ting, Efrém, Nina-Louisa, Horatscheck, André, Perepelittchenko, Liudmila, Prokofeva, Polina, Ehret, Theresa A. L., Radetzki, Silke, Neuenschwander, Martin, Specker, Edgar, Médard, Guillaume, Müller, Susanne, Wilhelm, Stephanie, Kuster, Bernhard, von Kries, Jens Peter, Haucke, Volker, Nazaré, Marc
Published in Journal of medicinal chemistry (26.10.2023)
Published in Journal of medicinal chemistry (26.10.2023)
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