A phase Ib study of the highly selective MET-TKI savolitinib plus gefitinib in patients with EGFR-mutated, MET-amplified advanced non-small-cell lung cancer
Yang, Jin-Ji, Fang, Jian, Shu, Yong-Qian, Chang, Jian-Hua, Chen, Gong-Yan, He, Jian Xing, Li, Wei, Liu, Xiao-Qing, Yang, Nong, Zhou, Caicun, Huang, Jian An, Frigault, Melanie M., Hartmaier, Ryan, Ahmed, Ghada F., Egile, Coumaran, Morgan, Shethah, Verheijen, Remy B., Mellemgaard, Anders, Yang, Liu, Wu, Yi-Long
Published in Investigational new drugs (01.04.2021)
Published in Investigational new drugs (01.04.2021)
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Journal Article
The Structural Basis of Actin Filament Branching by the Arp2/3 Complex
Rouiller, Isabelle, Xu, Xiao-Ping, Amann, Kurt J., Egile, Coumaran, Nickell, Stephan, Nicastro, Daniela, Li, Rong, Pollard, Thomas D., Volkmann, Niels, Hanein, Dorit
Published in The Journal of cell biology (10.03.2008)
Published in The Journal of cell biology (10.03.2008)
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Journal Article
The RickA protein of Rickettsia conorii activates the Arp2/3 complex
Cossart, Pascale, Gouin, Edith, Egile, Coumaran, Dehoux, Pierre, Villiers, Véronique, Adams, Josephine, Gertler, Frank, Li, Rong
Published in Nature (29.01.2004)
Published in Nature (29.01.2004)
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Journal Article
Discovery and Pharmacokinetic and Pharmacological Properties of the Potent and Selective MET Kinase Inhibitor 1‑{6-[6-(4-Fluorophenyl)-[1,2,4]triazolo[4,3‑b]pyridazin-3-ylsulfanyl]benzothiazol-2-yl}-3-(2-morpholin-4-ylethyl)urea (SAR125844)
Ugolini, Antonio, Kenigsberg, Mireille, Rak, Alexey, Vallée, Francois, Houtmann, Jacques, Lowinski, Maryse, Capdevila, Cécile, Khider, Jean, Albert, Eva, Martinet, Nathalie, Nemecek, Conception, Grapinet, Sandrine, Bacqué, Eric, Roesner, Manfred, Delaisi, Christine, Calvet, Loreley, Bonche, Fabrice, Semiond, Dorothée, Egile, Coumaran, Goulaouic, Hélène, Schio, Laurent
Published in Journal of medicinal chemistry (11.08.2016)
Published in Journal of medicinal chemistry (11.08.2016)
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Journal Article
IQGAP1 Stimulates Actin Assembly through the N-Wasp-Arp2/3 Pathway
Le Clainche, Christophe, Schlaepfer, Dominik, Ferrari, Aldo, Klingauf, Mirko, Grohmanova, Katarina, Veligodskiy, Alexey, Didry, Dominique, Le, Diep, Egile, Coumaran, Carlier, Marie-France, Kroschewski, Ruth
Published in The Journal of biological chemistry (05.01.2007)
Published in The Journal of biological chemistry (05.01.2007)
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Journal Article
Activation of Arp2/3 complex-mediated actin polymerization by cortactin
Zhan, Xi, Uruno, Takehito, Liu, Jiali, Zhang, Peijun, Fan, Ying-xin, Egile, Coumaran, Li, Rong, Mueller, Susette C
Published in Nature cell biology (01.03.2001)
Published in Nature cell biology (01.03.2001)
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Journal Article
MET genetic abnormalities unreliable for patient selection for therapeutic intervention in oropharyngeal squamous cell carcinoma
Lacroix, Ludovic, Post, Sophie F, Valent, Alexander, Melkane, Antoine E, Vielh, Philippe, Egile, Coumaran, Castell, Christelle, Larois, Christelle, Micallef, Sandrine, Saulnier, Patrick, Goulaouic, Hélène, Lefebvre, Anne-Marie, Temam, Stéphane
Published in PloS one (17.01.2014)
Published in PloS one (17.01.2014)
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Journal Article
Activation of the CDC42 Effector N-WASP by the Shigella flexneri IcsA Protein Promotes Actin Nucleation by Arp2/3 Complex and Bacterial Actin-Based Motility
Egile, Coumaran, Loisel, Thomas P., Laurent, Valérie, Li, Rong, Pantaloni, Dominique, Sansonetti, Philippe J., Carlier, Marie-France
Published in The Journal of cell biology (20.09.1999)
Published in The Journal of cell biology (20.09.1999)
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Journal Article
Cortactin regulates cell migration through activation of N-WASP
Kowalski, Jennifer R, Egile, Coumaran, Gil, Susana, Snapper, Scott B, Li, Rong, Thomas, Sheila M
Published in Journal of cell science (01.01.2005)
Published in Journal of cell science (01.01.2005)
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Journal Article
Structure of Arp2/3 Complex in Its Activated State and in Actin Filament Branch Junctions
Volkmann, Niels, Amann, Kurt J., Stoilova-McPhie, Svetla, Egile, Coumaran, Winter, Dirk C., Hazelwood, Larnele, Heuser, John E., Li, Rong, Pollard, Thomas D., Hanein, Dorit
Published in Science (American Association for the Advancement of Science) (28.09.2001)
Published in Science (American Association for the Advancement of Science) (28.09.2001)
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Journal Article
GRB2 Links Signaling to Actin Assembly by Enhancing Interaction of Neural Wiskott-Aldrich Syndrome Protein (N-WASp) with Actin-related Protein (ARP2/3) Complex
Carlier, Marie-France, Nioche, Pierre, Broutin-L'Hermite, Isabelle, Boujemaa, Rajaa, Le Clainche, Christophe, Egile, Coumaran, Garbay, Christiane, Ducruix, Arnaud, Sansonetti, Philippe, Pantaloni, Dominique
Published in The Journal of biological chemistry (21.07.2000)
Published in The Journal of biological chemistry (21.07.2000)
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Journal Article
Interaction of N-WASP with hnRNPK and Its Role in Filopodia Formation and Cell Spreading
Yoo, Youngdong, Wu, Xiaoyang, Egile, Coumaran, Li, Rong, Guan, Jun-Lin
Published in The Journal of biological chemistry (02.06.2006)
Published in The Journal of biological chemistry (02.06.2006)
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Journal Article
Activation of Arp2/3 Complex-Dependent Actin Polymerization by Plant Proteins Distantly Related to Scar/WAVE
Frank, Mary, Egile, Coumaran, Dyachok, Julia, Djakovic, Stevan, Nolasco, Michelle, Li, Rong, Smith, Laurie G., Chrispeels, Maarten J.
Published in Proceedings of the National Academy of Sciences - PNAS (16.11.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (16.11.2004)
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Journal Article
Control of Actin Filament Length and Turnover by Actin Depolymerizing Factor (ADF/Cofilin) in the Presence of Capping Proteins and ARP2/3 Complex
Ressad, Fariza, Didry, Dominique, Egile, Coumaran, Pantaloni, Dominique, Carlier, Marie-France
Published in The Journal of biological chemistry (23.07.1999)
Published in The Journal of biological chemistry (23.07.1999)
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Journal Article
Phase II study of the PI3K inhibitor pilaralisib (SAR245408; XL147) in patients with advanced or recurrent endometrial carcinoma
Matulonis, Ursula, Vergote, Ignace, Backes, Floor, Martin, Lainie P, McMeekin, Scott, Birrer, Michael, Campana, Frank, Xu, Yi, Egile, Coumaran, Ghamande, Sharad
Published in Gynecologic oncology (01.02.2015)
Published in Gynecologic oncology (01.02.2015)
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Journal Article
Phase I Safety, Pharmacokinetic, and Pharmacodynamic Study of SAR245408 (XL147), an Oral Pan-Class I PI3K Inhibitor, in Patients with Advanced Solid Tumors
SHAPIRO, Geoffrey I, RODON, Jordi, YI XU, EGILE, Coumaran, EDELMAN, Gerald, BEDELL, Cynthia, KWAK, Eunice L, BASELGA, Jose, BRANA, Irene, PANDYA, Shuchi S, SCHEFFOLD, Christian, LAIRD, A. Douglas, NGUYEN, Linh T
Published in Clinical cancer research (2014)
Published in Clinical cancer research (2014)
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