Novel coumarins active against Trypanosoma cruzi and toxicity assessment using the animal model Caenorhabditis elegans
Soares, Fabiana Gomes Nascimento, Göethel, Gabriela, Kagami, Luciano Porto, das Neves, Gustavo Machado, Sauer, Elisa, Birriel, Estefania, Varela, Javier, Gonçalves, Itamar Luís, Von Poser, Gilsane, González, Mercedes, Kawano, Daniel Fábio, Paula, Fávero Reisdorfer, de Melo, Eduardo Borges, Garcia, Solange Cristina, Cerecetto, Hugo, Eifler-Lima, Vera Lucia
Published in BMC pharmacology & toxicology (19.12.2019)
Published in BMC pharmacology & toxicology (19.12.2019)
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Journal Article
α- and β-Glucosidase inhibitors: chemical structure and biological activity
Borges de Melo, Eduardo, da Silveira Gomes, Adriane, Carvalho, Ivone
Published in Tetrahedron (29.10.2006)
Published in Tetrahedron (29.10.2006)
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Synthesis and anti-Mycobacterium tuberculosis activity of imide-β-carboline and carbomethoxy-β-carboline derivatives
Lopes-Ortiz, Mariana Aparecida, Panice, Manuela Ribeiro, Borges de Melo, Eduardo, Ataide Martins, João Paulo, Baldin, Vanessa Pietrowski, Agostinho Pires, Cláudia Terêncio, Caleffi-Ferracioli, Katiany Rizzieri, Dias Siqueira, Vera Lúcia, Bertin de Lima Scodro, Regiane, Sarragiotto, Maria Helena, Cardoso, Rosilene Fressatti
Published in European journal of medicinal chemistry (01.02.2020)
Published in European journal of medicinal chemistry (01.02.2020)
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Multivariate QSAR study on the antimutagenic activity of flavonoids against 3-NFA on Salmonella typhimurium TA98
Borges de Melo, Eduardo, Ataide Martins, João Paulo, Marinho Jorge, Teresa Cristina, Friozi, Marcelo Couto, Castro Ferreira, Márcia Miguel
Published in European journal of medicinal chemistry (01.10.2010)
Published in European journal of medicinal chemistry (01.10.2010)
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A structure-activity relationship study of the toxicity of ionic liquids using an adapted Ferreira-Kiralj hydrophobicity parameterElectronic supplementary information (ESI) available: Table S1 - SMILES strings, chemical abstracts service (CAS) code and log EC50 for each sample of dataset; Table S2 - molecular descriptors used in this study; Table S3 - values of Crippen and Mannhold log P; Table S4 - the observed and predicted activities for models 1, 2 and 3 in the external validation; and Fig.
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Inibidores da HIV-integrase: potencial abordagem farmacológica para tratamento da AIDS
Melo, Eduardo Borges de, Bruni, Aline Thaís, Ferreira, Márcia Miguel Castro
Published in Química Nova (01.06.2006)
Published in Química Nova (01.06.2006)
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Pharmacophore modeling, molecular docking, and molecular dynamics studies to identify new 5-HT2AR antagonists with the potential for design of new atypical antipsychotics
Martins, Allana Faustino, de Campos, Luana Janaína, Conda-Sheridan, Martin, de Melo, Eduardo Borges
Published in Molecular diversity (01.10.2023)
Published in Molecular diversity (01.10.2023)
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Multivariate QSAR, similarity search and ADMET studies based in a set of methylamine derivatives described as dopamine transporter inhibitors
de Oliveira, Luiz Henrique Dias, Cruz, Jorddy Neves, dos Santos, Cleydson Breno Rodrigues, de Melo, Eduardo Borges
Published in Molecular diversity (06.09.2023)
Published in Molecular diversity (06.09.2023)
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