Search Results - "Edmondson, S D" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Pharmacological Characterization of a Novel Beta 3 Adrenergic Agonist, Vibegron: Evaluation of Antimuscarinic Receptor Selectivity for Combination Therapy for Overactive Bladder

Pharmacological Characterization of a Novel Beta 3 Adrenergic Agonist, Vibegron: Evaluation of Antimuscarinic Receptor Selectivity for Combination Therapy for Overactive Bladder

by Di Salvo, J, Nagabukuro, H, Wickham, L A, Abbadie, C, DeMartino, J A, Fitzmaurice, A, Gichuru, L, Kulick, A, Donnelly, M J, Jochnowitz, N, Hurley, A L, Pereira, A, Sanfiz, A, Veronin, G, Villa, K, Woods, J, Zamlynny, B, Zycband, E, Salituro, G M, Frenkl, T, Weber, A E, Edmondson, S D, Struthers, M
Published in The Journal of pharmacology and experimental therapeutics (01.02.2017)

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Journal Article

A concise route to the tetracyclic core of phorbol

A concise route to the tetracyclic core of phorbol

by Paquette, Leo A., Sauer, Daryl R., Edmondson, Scott D., Friedrich, Dirk
Published in Tetrahedron (04.04.1994)

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Journal Article

Analysis of the Conformational Nature, Resolvability, and Thermal Racemization of Hetero 2,3-Dispiro Cyclohexanones. The Weighting of Carbonyl/C-X Stabilization Relative to the Electronic Interaction between the Vicinal Electronegative Substituents

Analysis of the Conformational Nature, Resolvability, and Thermal Racemization of Hetero 2,3-Dispiro Cyclohexanones. The Weighting of Carbonyl/C-X Stabilization Relative to the Electronic Interaction between the Vicinal Electronegative Substituents

by Paquette, Leo A, Branan, Bruce M, Friedrich, Dirk, Edmondson, Scott D, Rogers, Robin D
Published in Journal of the American Chemical Society (01.01.1994)

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Journal Article

Crystal Structure of Human Phosphodiesterase 3B: Atomic Basis for Substrate and Inhibitor Specificity

Crystal Structure of Human Phosphodiesterase 3B: Atomic Basis for Substrate and Inhibitor Specificity

by Scapin, Giovanna, Patel, Sangita B, Chung, Christine, Varnerin, Jeffrey P, Edmondson, Scott D, Mastracchio, Anthony, Parmee, Emma R, Singh, Suresh B, Becker, Joseph W, Van der Ploeg, Lex H. T, Tota, Michael R
Published in Biochemistry (Easton) (25.05.2004)

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Journal Article

Palladium-Catalyzed Coupling of Vinylogous Amides with Aryl Halides: Applications to the Synthesis of Heterocycles

Palladium-Catalyzed Coupling of Vinylogous Amides with Aryl Halides: Applications to the Synthesis of Heterocycles

by Edmondson, Scott D, Mastracchio, Anthony, Parmee, Emma R
Published in Organic letters (20.04.2000)

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Journal Article

The Total Synthesis of Spirotryprostatin A

The Total Synthesis of Spirotryprostatin A

by Edmondson, Scott D., Danishefsky, Samuel J.
Published in Angewandte Chemie (International ed.) (04.05.1998)

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Journal Article

Discovery of potent and selective orally bioavailable β-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors

Discovery of potent and selective orally bioavailable β-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors

by Edmondson, Scott D., Mastracchio, Anthony, Duffy, Joseph L., Eiermann, George J., He, Huaibing, Ita, Ida, Leiting, Barbara, Leone, Joseph F., Lyons, Kathryn A., Makarewicz, Amanda M., Patel, Reshma A., Petrov, Aleksandr, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (15.06.2005)

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Journal Article

Potent and selective proline derived dipeptidyl peptidase IV inhibitors

Potent and selective proline derived dipeptidyl peptidase IV inhibitors

by Edmondson, Scott D., Mastracchio, Anthony, Beconi, Maria, Colwell, Lawrence F., Habulihaz, Bahanu, He, Huaibing, Kumar, Sanjeev, Leiting, Barbara, Lyons, Kathryn A., Mao, Ann, Marsilio, Frank, Patel, Reshma A., Wu, Joseph K., Zhu, Lan, Thornberry, Nancy A., Weber, Ann E., Parmee, Emma R.
Published in Bioorganic & medicinal chemistry letters (18.10.2004)

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Journal Article

Crystallization and X-ray analysis of the catalytic domain of human PDE 3B

Crystallization and X-ray analysis of the catalytic domain of human PDE 3B

by Patel, S. B., Varnerin, J. P., Tota, M. R., Edmondson, S. D., Parmee, E. R., Chung, C., Singh, S. B., Mastracchio, A., Becker, J. W., Scapin, G.
Published in Acta crystallographica. Section A, Foundations of crystallography (23.08.2005)

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Journal Article

4-Amino cyclohexylglycine analogues as potent dipeptidyl peptidase IV inhibitors

4-Amino cyclohexylglycine analogues as potent dipeptidyl peptidase IV inhibitors

by Parmee, Emma R., He, Jiafang, Mastracchio, Anthony, Edmondson, Scott D., Colwell, Larry, Eiermann, George, Feeney, William P., Habulihaz, Bahanu, He, Huaibing, Kilburn, Ruth, Leiting, Barbara, Lyons, Kathryn, Marsilio, Frank, Patel, Reshma A., Petrov, Aleksandr, Di Salvo, Jerry, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (05.01.2004)

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Journal Article

Benzyl vinylogous amide substituted aryldihydropyridazinones and aryldimethylpyrazolones as potent and selective PDE3B inhibitors

Benzyl vinylogous amide substituted aryldihydropyridazinones and aryldimethylpyrazolones as potent and selective PDE3B inhibitors

by Edmondson, Scott D., Mastracchio, Anthony, He, Jiafang, Chung, Christine C., Forrest, Michael J., Hofsess, Scott, MacIntyre, Euan, Metzger, Joseph, O'Connor, Naphtali, Patel, Kajal, Tong, Xinchun, Tota, Michael R., Van der Ploeg, Lex H.T., Varnerin, Jeff P., Fisher, Michael H., Wyvratt, Matthew J., Weber, Ann E., Parmee, Emma R.
Published in Bioorganic & medicinal chemistry letters (17.11.2003)

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Journal Article

Discovery of potent, selective, and orally bioavailable pyridone-based dipeptidyl peptidase-4 inhibitors

Discovery of potent, selective, and orally bioavailable pyridone-based dipeptidyl peptidase-4 inhibitors

by Xu, Jinyou, Wei, Lan, Mathvink, Robert, Edmondson, Scott D., Mastracchio, Anthony, Eiermann, George J., He, Huaibing, Leone, Joseph F., Leiting, Barbara, Lyons, Kathryn A., Marsilio, Frank, Patel, Reshma A., Petrov, Aleksandr, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (01.03.2006)

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Journal Article

$Crystallization and preliminary X-ray diffraction analysis of the catalytic domain of recombinant human phosphodiesterase 3B$

Crystallization and preliminary X-ray diffraction analysis of the catalytic domain of recombinant human phosphodiesterase 3B

by Patel, Sangita B., Varnerin, Jeffrey P., Tota, Michael R., Edmondson, Scott D., Parmee, Emma R., Becker, Joseph W., Scapin, Giovanna
Published in Acta crystallographica. Section D, Biological crystallography. (01.01.2004)

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Journal Article

Studies Directed toward the Synthesis of the Unusual Antileukemic Diterpene Jatrophatrione. 1. A Solution to the Problem of Chirality Merger during Elaboration of the Entire Carbotricyclic Framework

Studies Directed toward the Synthesis of the Unusual Antileukemic Diterpene Jatrophatrione. 1. A Solution to the Problem of Chirality Merger during Elaboration of the Entire Carbotricyclic Framework

by Paquette, Leo A, Nakatani, Shogo, Zydowsky, Thomas M, Edmondson, Scott D, Sun, Li-Qiang, Skerlj, Renato
Published in Journal of organic chemistry (30.04.1999)

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Journal Article

Studies Directed toward the Synthesis of the Unusual Antileukemic Diterpene Jatrophatrione. 2. Functionalization of Advanced Polycyclic Precursors to the 9-Epi and 8,9-Dehydro Congeners

Studies Directed toward the Synthesis of the Unusual Antileukemic Diterpene Jatrophatrione. 2. Functionalization of Advanced Polycyclic Precursors to the 9-Epi and 8,9-Dehydro Congeners

by Paquette, Leo A, Edmondson, Scott D, Monck, Nathaniel, Rogers, Robin D
Published in Journal of organic chemistry (30.04.1999)

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Journal Article

Conformational Analysis of Poly(spirotetrahydrofuranyl)cyclohexyl Systems. The Preference of Multiple C−O Bonds for Equatorial Occupancy

Conformational Analysis of Poly(spirotetrahydrofuranyl)cyclohexyl Systems. The Preference of Multiple C−O Bonds for Equatorial Occupancy

by Paquette, Leo A, Stepanian, Marshall, Branan, Bruce M, Edmondson, Scott D, Bauer, Cary B, Rogers, Robin D
Published in Journal of the American Chemical Society (08.05.1996)

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Journal Article

Beta-Amino Tetrahydroimidazo (1, 2-A)Pyrazines And Tetrahydrotrioazolo (4, 3-A)Pyrazines as Dipeptidyl Peptidase Inhibitors for Treatment or Prevention of Diabetes

Beta-Amino Tetrahydroimidazo (1, 2-A)Pyrazines And Tetrahydrotrioazolo (4, 3-A)Pyrazines as Dipeptidyl Peptidase Inhibitors for Treatment or Prevention of Diabetes

by Parmee(US), Emma, R, Maccoss(US), Malcolm, Fisher (US), Michael, H, Edmondson (US), Scott, D, Weber (US), Ann, E, Kim (US), Dooseop, Xu(Us), Jinyou
Year of Publication 10.01.2006

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