The coumarin osthole is a non-electrophilic agonist of TRPA1
Torres, Karen V., Pantke, Sebastian, Rudolf, Daniel, Eberhardt, Mirjam M., Leffler, Andreas
Published in Neuroscience letters (15.10.2022)
Published in Neuroscience letters (15.10.2022)
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Journal Article
Molecular mechanisms of MrgprA3‐independent activation of the transient receptor potential ion channels TRPA1 and TRPV1 by chloroquine
Fricke, Tabea C., Pantke, Sebastian, Lüttmann, Bjarne, Echtermeyer, Frank G., Herzog, Christine, Eberhardt, Mirjam J., Leffler, Andreas
Published in British journal of pharmacology (01.09.2023)
Published in British journal of pharmacology (01.09.2023)
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Journal Article
Oxidation of methionine residues activates the high-threshold heat-sensitive ion channel TRPV2
Fricke, Tabea C., Echtermeyer, Frank, Zielke, Johannes, de la Roche, Jeanne, Filipovic, Milos R., Claverol, Stéphane, Herzog, Christine, Tominaga, Makoto, Pumroy, Ruth A., Moiseenkova-Bell, Vera Y., Zygmunt, Peter M., Leffler, Andreas, Eberhardt, Mirjam J.
Published in Proceedings of the National Academy of Sciences - PNAS (26.11.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (26.11.2019)
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Journal Article
Methylglyoxal activates nociceptors through transient receptor potential channel A1 (TRPA1): a possible mechanism of metabolic neuropathies
Eberhardt, Mirjam J, Filipovic, Milos R, Leffler, Andreas, de la Roche, Jeanne, Kistner, Katrin, Fischer, Michael J, Fleming, Thomas, Zimmermann, Katharina, Ivanovic-Burmazovic, Ivana, Nawroth, Peter P, Bierhaus, Angelika, Reeh, Peter W, Sauer, Susanne K
Published in The Journal of biological chemistry (17.08.2012)
Published in The Journal of biological chemistry (17.08.2012)
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Journal Article
The Molecular Basis for Species-specific Activation of Human TRPA1 Protein by Protons Involves Poorly Conserved Residues within Transmembrane Domains 5 and 6
de la Roche, Jeanne, Eberhardt, Mirjam J., Klinger, Alexandra B., Stanslowsky, Nancy, Wegner, Florian, Koppert, Wolfgang, Reeh, Peter W., Lampert, Angelika, Fischer, Michael J.M., Leffler, Andreas
Published in The Journal of biological chemistry (12.07.2013)
Published in The Journal of biological chemistry (12.07.2013)
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Journal Article
Human TRPA1 is a heat sensor displaying intrinsic U-shaped thermosensitivity
Moparthi, Lavanya, Kichko, Tatjana I, Eberhardt, Mirjam, Högestätt, Edward D, Kjellbom, Per, Johanson, Urban, Reeh, Peter W, Leffler, Andreas, Filipovic, Milos R, Zygmunt, Peter M
Published in Scientific reports (28.06.2016)
Published in Scientific reports (28.06.2016)
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Journal Article
Quaternary Lidocaine Derivative QX-314 Activates and Permeates Human TRPV1 and TRPA1 to Produce Inhibition of Sodium Channels and Cytotoxicity
Stueber, Thomas, Eberhardt, Mirjam J, Hadamitzky, Christoph, Jangra, Annette, Schenk, Stefan, Dick, Felicia, Stoetzer, Carsten, Kistner, Katrin, Reeh, Peter W, Binshtok, Alexander M, Leffler, Andreas
Published in Anesthesiology (Philadelphia) (01.05.2016)
Published in Anesthesiology (Philadelphia) (01.05.2016)
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Journal Article
Reactive metabolites of acetaminophen activate and sensitize the capsaicin receptor TRPV1
Eberhardt, Mirjam J, Schillers, Florian, Eberhardt, Esther M, Risser, Linus, de la Roche, Jeanne, Herzog, Christine, Echtermeyer, Frank, Leffler, Andreas
Published in Scientific reports (06.10.2017)
Published in Scientific reports (06.10.2017)
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Journal Article
Distinct Mechanisms Account for In Vitro Activation and Sensitization of TRPV1 by the Porphyrin Hemin
Palmaers, Natalie E., Wiegand, Steffen B., Herzog, Christine, Echtermeyer, Frank G., Eberhardt, Mirjam J., Leffler, Andreas
Published in International journal of molecular sciences (01.10.2021)
Published in International journal of molecular sciences (01.10.2021)
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Journal Article
Differential cytotoxicity and intracellular calcium-signalling following activation of the calcium-permeable ion channels TRPV1 and TRPA1
Stueber, Thomas, Eberhardt, Mirjam J., Caspi, Yaki, Lev, Shaya, Binshtok, Alexander, Leffler, Andreas
Published in Cell calcium (Edinburgh) (01.12.2017)
Published in Cell calcium (Edinburgh) (01.12.2017)
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Journal Article
TRPA1 and Substance P Mediate Colitis in Mice
Engel, Matthias A, Leffler, Andreas, Niedermirtl, Florian, Babes, Alexandru, Zimmermann, Katharina, Filipović, Miloš R, Izydorczyk, Iwona, Eberhardt, Mirjam, Kichko, Tatjana I, Mueller–Tribbensee, Sonja M, Khalil, Mohammad, Siklosi, Norbert, Nau, Carla, Ivanović–Burmazović, Ivana, Neuhuber, Winfried L, Becker, Christoph, Neurath, Markus F, Reeh, Peter W
Published in Gastroenterology (New York, N.Y. 1943) (01.10.2011)
Published in Gastroenterology (New York, N.Y. 1943) (01.10.2011)
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Journal Article
HCN2 channels account for mechanical (but not heat) hyperalgesia during long-standing inflammation
Schnorr, Sabine, Eberhardt, Mirjam, Kistner, Katrin, Rajab, Hamsa, Käßer, Johannes, Hess, Andreas, Reeh, Peter, Ludwig, Andreas, Herrmann, Stefan
Published in Pain (Amsterdam) (01.06.2014)
Published in Pain (Amsterdam) (01.06.2014)
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Journal Article
The General Anesthetic Propofol Excites Nociceptors by Activating TRPV1 and TRPA1 Rather than GABAA Receptors
Fischer, Michael J.M., Leffler, Andreas, Niedermirtl, Florian, Kistner, Katrin, Eberhardt, Mirjam, Reeh, Peter W., Nau, Carla
Published in The Journal of biological chemistry (05.11.2010)
Published in The Journal of biological chemistry (05.11.2010)
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Journal Article
TRPA1 and TRPV1 are required for lidocaine-evoked calcium influx and neuropeptide release but not cytotoxicity in mouse sensory neurons
Eberhardt, Mirjam, Stueber, Thomas, de la Roche, Jeanne, Herzog, Christine, Leffler, Andreas, Reeh, Peter W, Kistner, Katrin
Published in PloS one (15.11.2017)
Published in PloS one (15.11.2017)
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Journal Article
Etomidate and propylene glycol activate nociceptive TRP ion channels
Niedermirtl, Florian, Eberhardt, Mirjam, Namer, Barbara, Leffler, Andreas, Nau, Carla, Reeh, Peter W, Kistner, Katrin
Published in Molecular pain (01.01.2018)
Published in Molecular pain (01.01.2018)
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Journal Article
Sea-Anemone Toxin ATX-II Elicits A-Fiber-Dependent Pain and Enhances Resurgent and Persistent Sodium Currents in Large Sensory Neurons
Klinger, Alexandra B, Eberhardt, Mirjam, Link, Andrea S, Namer, Barbara, Kutsche, Lisa K, Schuy, E Theresa, Sittl, Ruth, Hoffmann, Tali, Alzheimer, Christian, Huth, Tobias, Carr, Richard W, Lampert, Angelika
Published in Molecular pain (15.09.2012)
Published in Molecular pain (15.09.2012)
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Journal Article
Streptozotocin Stimulates the Ion Channel TRPA1 Directly
Andersson, David A., Filipović, Milos R., Gentry, Clive, Eberhardt, Mirjam, Vastani, Nisha, Leffler, Andreas, Reeh, Peter, Bevan, Stuart
Published in The Journal of biological chemistry (01.06.2015)
Published in The Journal of biological chemistry (01.06.2015)
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Journal Article
Methylglyoxal modification of Nav1.8 facilitates nociceptive neuron firing and causes hyperalgesia in diabetic neuropathy
Bierhaus, Angelika, Fleming, Thomas, Stoyanov, Stoyan, Leffler, Andreas, Babes, Alexandru, Neacsu, Cristian, Sauer, Susanne K, Eberhardt, Mirjam, Schnölzer, Martina, Lasitschka, Felix, Lasischka, Felix, Neuhuber, Winfried L, Kichko, Tatjana I, Konrade, Ilze, Elvert, Ralf, Mier, Walter, Pirags, Valdis, Lukic, Ivan K, Morcos, Michael, Dehmer, Thomas, Rabbani, Naila, Thornalley, Paul J, Edelstein, Diane, Nau, Carla, Forbes, Josephine, Humpert, Per M, Schwaninger, Markus, Ziegler, Dan, Stern, David M, Cooper, Mark E, Haberkorn, Uwe, Brownlee, Michael, Reeh, Peter W, Nawroth, Peter P
Published in Nature medicine (01.06.2012)
Published in Nature medicine (01.06.2012)
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Journal Article