Assessment of the Effect of Organ Impairment on the Pharmacokinetics of 2'-MOE and Phosphorothioate Modified Antisense Oligonucleotides
Wang, Yanfeng, Diep, John K, Yu, Rosie Z, Hurh, Eunju, Karwatowska-Prokopczuk, Ewa, Schneider, Eugene, Henry, Scott, Bhanot, Sanjay, Geary, Richard S
Published in Journal of clinical pharmacology (01.01.2023)
Published in Journal of clinical pharmacology (01.01.2023)
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Journal Article
Population pharmacokinetics of sonidegib (LDE225), an oral inhibitor of hedgehog pathway signaling, in healthy subjects and in patients with advanced solid tumors
Goel, Varun, Hurh, Eunju, Stein, Andrew, Nedelman, Jerry, Zhou, Jocelyn, Chiparus, Ovidiu, Huang, Pai-Hsi, Gogov, Sven, Sellami, Dalila
Published in Cancer chemotherapy and pharmacology (01.04.2016)
Published in Cancer chemotherapy and pharmacology (01.04.2016)
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Assessment of efficacy and safety of volanesorsen for treatment of metabolic complications in patients with familial partial lipodystrophy: Results of the BROADEN study: Volanesorsen in FPLD; The BROADEN Study
Oral, Elif A, Garg, Abhimanyu, Tami, Joseph, Huang, Eric A, O'Dea, Louis St L, Schmidt, Hartmut, Tiulpakov, Anatoly, Mertens, Ann, Alexander, Veronica J, Watts, Lynnetta, Hurh, Eunju, Witztum, Joseph L, Geary, Richard S, Tsimikas, Sotirios
Published in Journal of clinical lipidology (01.11.2022)
Published in Journal of clinical lipidology (01.11.2022)
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Journal Article
Abstract 6046: CFT8634, a BRD9 BiDAC™ degrader, is active in a subset of multiple myeloma cell line models and synergistic when combined with pomalidomide or dexamethasone
Poling, Laura L., Cocozziello, David, he, Minsng, Hurh, Eunju, Lobbardi, Riadh, Jackson, Katrina L., Fisher, Stewart L., Pollock, Roy M.
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Quantitative Prediction of Human Pharmacokinetics for Monoclonal Antibodies: Retrospective Analysis of Monkey as a Single Species for First-in-Human Prediction
Dong, Jennifer Q., Salinger, David H., Endres, Christopher J., Gibbs, John P., Hsu, Cheng-Pang, Stouch, Brian J., Hurh, Eunju, Gibbs, Megan
Published in Clinical pharmacokinetics (01.02.2011)
Published in Clinical pharmacokinetics (01.02.2011)
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Abstract 1658: CFT1946, a potent, selective BRAF V600X mutant-specific degrader demonstrates superior activity as a single agent to clinically approved BRAF inhibitors and standard of care combinations in preclinical models of BRAF V600X melanoma, CRC, NSCLC, and brain metastasis
Kreger, Bridget, Stephenson, Jacob R., Sowa, Mathew E., Perino, Samantha A., Poling, Laura L., Hurh, Eunju, Thomenius, Michael J., Liang, Yanke, Fisher, Stewart L., Pollock, Roy M.
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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INHIBITION OF APOLIPOPROTEIN C-III WITH GALNAC CONJUGATED ANTISENSE DRUG POTENTLY LOWERS FASTING SERUM APOLIPOPROTEIN C-III AND TRIGLYCERIDE LEVELS IN HEALTHY VOLUNTEERS WITH ELEVATED TRIGLYCERIDES
Alexander, Veronica J., Digenio, Andres, Xia, Shuting, Hurh, Eunju, Hughes, Steve, Geary, Richard S., Witztum, Joseph L., Tsimikas, Sotirios
Published in Journal of the American College of Cardiology (10.03.2018)
Published in Journal of the American College of Cardiology (10.03.2018)
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Treatment with Volanesorsen, a 2′-O-Methoxyethyl-Modified Antisense Oligonucleotide Targeting APOC3 mRNA, Does Not Affect the QTc Interval in Healthy Volunteers
Watts, Lynnetta M, Karwatowska-Prokopczuk, Ewa, Hurh, Eunju, Alexander, Veronica J, Balogh, Kristin, O'Dea, Louis, Geary, Richard S, Tsimikas, Sotirios
Published in Nucleic acid therapeutics (01.08.2020)
Published in Nucleic acid therapeutics (01.08.2020)
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Journal Article
AMG 386, a selective angiopoietin 1/2-neutralizing peptibody, inhibits angiogenesis in models of ocular neovascular diseases
Oliner, Jonathan D, Bready, James, Nguyen, Linh, Estrada, Juan, Hurh, Eunju, Ma, Hongjin, Pretorius, James, Fanslow, William, Nork, T Michael, Leedle, Robert A, Kaufman, Stephen, Coxon, Angela
Published in Investigative ophthalmology & visual science (24.04.2012)
Published in Investigative ophthalmology & visual science (24.04.2012)
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Journal Article
Absorption, distribution, metabolism, and excretion (ADME) of super(14)C-sonidegib (LDE225) in healthy volunteers
Zollinger, Markus, Lozac'h, Frederic, Hurh, Eunju, Emotte, Corinne, Bauly, Hounayda, Swart, Piet
Published in Cancer chemotherapy and pharmacology (01.07.2014)
Published in Cancer chemotherapy and pharmacology (01.07.2014)
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Journal Article
Absorption, distribution, metabolism, and excretion (ADME) of ^sup 14^C-sonidegib (LDE225) in healthy volunteers
Zollinger, Markus, Lozac'h, Frédéric, Hurh, Eunju, Emotte, Corinne, Bauly, Hounayda, Swart, Piet
Published in Cancer chemotherapy and pharmacology (01.07.2014)
Published in Cancer chemotherapy and pharmacology (01.07.2014)
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Journal Article
Phase 1b Dose-Escalation Study of Sonidegib (LDE225) in Combination with Ruxolitinib (INC424) in Patients with Myelofibrosis
Gupta, Vikas, Koschmieder, Steffen, Harrison, Claire N., Cervantes, Francisco, Heidel, Florian H, Drummond, Mark, Rey, Jerome, Hurh, Eunju, Bao, Weichao, Rampersad, Anita, Kalambakas, Stacey, Vannucchi, Alessandro Maria
Published in Blood (06.12.2014)
Published in Blood (06.12.2014)
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Journal Article
Effects of physostigmine on the pharmacokinetics of intravenous parathion in rats
Hurh, Eunju, Lee, Eun J., Kim, Yoon G., Kim, Sung Y., Kim, So H., Kim, Young C., Lee, Myung G.
Published in Biopharmaceutics & drug disposition (01.11.2000)
Published in Biopharmaceutics & drug disposition (01.11.2000)
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Journal Article
Assessment of the Drug Interaction Potential of Unconjugated and GalNAc 3 -Conjugated 2'-MOE-ASOs
Shemesh, Colby S, Yu, Rosie Z, Warren, Mark S, Liu, Michael, Jahic, Mirza, Nichols, Brandon, Post, Noah, Lin, Song, Norris, Daniel A, Hurh, Eunju, Huang, Jane, Watanabe, Tanya, Henry, Scott P, Wang, Yanfeng
Published in Molecular therapy. Nucleic acids (15.12.2017)
Published in Molecular therapy. Nucleic acids (15.12.2017)
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A phase I/II study of LDE225, a smoothened (Smo) antagonist, in pediatric patients with recurrent medulloblastoma (MB) or other solid tumors
Geoerger, Birgit, Aerts, Isabelle, Casanova, Michela, Chisholm, Julia C., Hargrave, Darren R, Leary, Sarah, Ashley, David M, Bouffet, Eric, MacDonald, Tobey, Hurh, Eunju, Dey, Jyotirmoy, Kalambakas, Stacey, Amakye, Dereck Dokyi, Kieran, Mark W.
Published in Journal of clinical oncology (20.05.2012)
Published in Journal of clinical oncology (20.05.2012)
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2-Arylthiazolidine-4-carboxylic acid amides (ATCAA) target dual pathways in cancer cells: 5'-AMP-activated protein kinase (AMPK)/mTOR and PI3K/Akt/mTOR pathways
LI, Chien-Ming, RAMESHNARAYANAN, YANLU, HURH, Eunju, COSS, Christopher C, BARRETT, Christina M, MILLER, Duane D, DALTON, James T
Published in International journal of oncology (01.10.2010)
Published in International journal of oncology (01.10.2010)
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