AKF-D52, a Synthetic Phenoxypyrimidine-Urea Derivative, Triggers Extrinsic/Intrinsic Apoptosis and Cytoprotective Autophagy in Human Non-Small Cell Lung Cancer Cells
Gil, Hyo-Sun, Lee, Jeong-Hun, Farag, Ahmed K., Hassan, Ahmed H. E., Chung, Kyung-Sook, Choi, Jung-Hye, Roh, Eun-Joo, Lee, Kyung-Tae
Published in Cancers (22.11.2021)
Published in Cancers (22.11.2021)
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MRS2500 [2-Iodo-N6-methyl-(N)-methanocarba-2â²-deoxyadenosine-3â²,5â²-bisphosphate], a Potent, Selective, and Stable Antagonist of the Platelet P2Y1 Receptor with Strong Antithrombotic Activity in Mice
Hechler, Béatrice, Nonne, Christelle, Roh, Eun Joo, Cattaneo, Marco, Cazenave, Jean-Pierre, Lanza, François, Jacobson, Kenneth A, Gachet, Christian
Published in The Journal of pharmacology and experimental therapeutics (01.02.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2006)
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P2Y1 Antagonists: Combining Receptor-Based Modeling and QSAR for a Quantitative Prediction of the Biological Activity Based on Consensus Scoring
Costanzi, Stefano, Tikhonova, Irina G, Ohno, Michihiro, Roh, Eun Joo, Joshi, Bhalchandra V, Colson, Anny-Odile, Houston, Dayle, Maddileti, Savitri, Harden, T. Kendall, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (12.07.2007)
Published in Journal of medicinal chemistry (12.07.2007)
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Diabetes mellitus: Classification, mediators, and complications; A gate to identify potential targets for the development of new effective treatments
Antar, Samar A., Ashour, Nada A., Sharaky, Marwa, Khattab, Muhammad, Ashour, Naira A., Zaid, Roaa T., Roh, Eun Joo, Elkamhawy, Ahmed, Al-Karmalawy, Ahmed A.
Published in Biomedicine & pharmacotherapy (01.12.2023)
Published in Biomedicine & pharmacotherapy (01.12.2023)
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Trifluoperazine, a Well-Known Antipsychotic, Inhibits Glioblastoma Invasion by Binding to Calmodulin and Disinhibiting Calcium Release Channel IP3R
Kang, Seokmin, Hong, Jinpyo, Lee, Jung Moo, Moon, Hyo Eun, Jeon, Borami, Choi, Jungil, Yoon, Nal Ae, Paek, Sun Ha, Roh, Eun Joo, Lee, C Justin, Kang, Sang Soo
Published in Molecular cancer therapeutics (01.01.2017)
Published in Molecular cancer therapeutics (01.01.2017)
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Design, Synthesis and Biological Evaluation of 1,3,5-Triazine Derivatives Targeting hA1 and hA3 Adenosine Receptor
Park, Sujin, Ahn, Yujin, Kim, Yongchan, Roh, Eun Joo, Lee, Yoonji, Han, Chaebin, Yoo, Hee Min, Yu, Jinha
Published in Molecules (Basel, Switzerland) (22.06.2022)
Published in Molecules (Basel, Switzerland) (22.06.2022)
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Sulfonamide-based 4-anilinoquinoline derivatives as novel dual Aurora kinase (AURKA/B) inhibitors: Synthesis, biological evaluation and in silico insights
Al-Sanea, Mohammad M., Elkamhawy, Ahmed, Paik, Sora, Lee, Kyeong, El Kerdawy, Ahmed M., Syed Nasir Abbas, Bukhari, Joo Roh, Eun, Eldehna, Wagdy M., Elshemy, Heba A.H., Bakr, Rania B, Ali Farahat, Ibrahim, Alzarea, Abdulaziz I., Alzarea, Sami I., Alharbi, Khalid S., Abdelgawad, Mohamed A.
Published in Bioorganic & medicinal chemistry (01.07.2020)
Published in Bioorganic & medicinal chemistry (01.07.2020)
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Discovery of N-benzylbenzamide-based allosteric inhibitors of Aurora kinase A
Lee, Hyomin, Kim, Euijung, Hwang, Narae, Yoo, Jesik, Nam, Yunju, Hwang, Injeoung, Park, Jin-Gyeong, Park, Sang-Eun, Chung, Kyung-Sook, Won Chung, Hwan, Song, Chiman, Ji, Mi-Jung, Park, Hyun-Mee, Lee, In-Kyun, Lee, Kyung-Tae, Joo Roh, Eun, Hur, Wooyoung
Published in Bioorganic & medicinal chemistry (15.03.2024)
Published in Bioorganic & medicinal chemistry (15.03.2024)
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Scaffold Repurposing of In-House Small Molecule Candidates Leads to Discovery of First-in-Class CDK-1/HER-2 Dual Inhibitors: In Vitro and In Silico Screening
Elkamhawy, Ahmed, Ammar, Usama M., Paik, Sora, Abdellattif, Magda H., Elsherbeny, Mohamed H., Lee, Kyeong, Roh, Eun Joo
Published in Molecules (Basel, Switzerland) (01.09.2021)
Published in Molecules (Basel, Switzerland) (01.09.2021)
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Novel topoisomerase II/EGFR dual inhibitors: design, synthesis and docking studies of naphtho[2′,3′:4,5]thiazolo[3,2-a]pyrimidine hybrids as potential anticancer agents with apoptosis inducing activity
Mourad, Mai A. E., Abo Elmaaty, Ayman, Zaki, Islam, Mourad, Ahmed A. E., Hofni, Amal, Khodir, Ahmed E., Aboubakr, Esam M., Elkamhawy, Ahmed, Roh, Eun Joo, Al-Karmalawy, Ahmed A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
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Reprofiling of pyrimidine-based DAPK1/CSF1R dual inhibitors: identification of 2,5-diamino-4-pyrimidinol derivatives as novel potential anticancer lead compounds
Farag, Ahmed K., Hassan, Ahmed H. E., Ahn, Byung Sun, Park, Ki Duk, Roh, Eun Joo
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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EGFR inhibitors from cancer to inflammation: Discovery of 4-fluoro-N-(4-(3-(trifluoromethyl)phenoxy)pyrimidin-5-yl)benzamide as a novel anti-inflammatory EGFR inhibitor
Elkamhawy, Ahmed, Hassan, Ahmed H.E., Paik, Sora, Sup Lee, Yong, Lee, Hwi-Ho, Shin, Ji-Sun, Lee, Kyung-Tae, Roh, Eun Joo
Published in Bioorganic chemistry (01.05.2019)
Published in Bioorganic chemistry (01.05.2019)
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Discovery of N-(1-(3-fluorobenzoyl)-1H-indol-5-yl)pyrazine-2-carboxamide: a novel, selective, and competitive indole-based lead inhibitor for human monoamine oxidase B
Elkamhawy, Ahmed, Paik, Sora, Kim, Hyeon Jeong, Park, Jong-Hyun, Londhe, Ashwini M., Lee, Kyeong, Pae, Ae Nim, Park, Ki Duk, Roh, Eun Joo
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Synthesis and structure–activity relationships of tri-substituted thiazoles as RAGE antagonists for the treatment of Alzheimer’s disease
Lee, Yun Suk, Kim, Hee, Kim, Young-Ho, Roh, Eun Joo, Han, Hogyu, Shin, Kye Jung
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
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Novel potent blockers for TWIK-1/TREK-1 heterodimers as potential antidepressants
Lee, Elliot H., Park, Jung-eun, Gotina, Lizaveta, Han, Young-Eun, Viswanath, Ambily Nath Indu, Yoo, Seonguk, Moon, Bongjin, Hwang, Jin-Young, Park, Woo Kyu, Cho, Yoonjeong, Song, Chiman, Min, Sun-Joon, Hwang, Eun Mi, Lee, Hyunbeom, Pae, Ae Nim, Roh, Eun Joo, Oh, Soo-Jin
Published in Biomedicine & pharmacotherapy (01.09.2023)
Published in Biomedicine & pharmacotherapy (01.09.2023)
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Identification of Novel Aryl Carboxamide Derivatives as Death-Associated Protein Kinase 1 (DAPK1) Inhibitors with Anti-Proliferative Activities: Design, Synthesis, In Vitro, and In Silico Biological Studies
Elkamhawy, Ahmed, Paik, Sora, Ali, Eslam M. H, Hassan, Ahmed H. E, Kang, So Jin, Lee, Kyeong, Roh, Eun Joo
Published in Pharmaceuticals (Basel, Switzerland) (25.08.2022)
Published in Pharmaceuticals (Basel, Switzerland) (25.08.2022)
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Caffeine-Mediated Inhibition of Calcium Release Channel Inositol 1,4,5-Trisphosphate Receptor Subtype 3 Blocks Glioblastoma Invasion and Extends Survival
SANG SOO KANG, HAN, Kyung-Seok, SEUNG HYUN YOO, CHUN KEE CHUNG, PARK, Sung-Hye, SUN HA PAEK, EUN JOO ROH, SUNG JOONG LEE, PARK, Jae-Yong, TRAYNELIS, Stephen F, LEE, C. Justin, BO MI KU, YEON KYUNG LEE, HONG, Jinpyo, HYE YOUNG SHIN, ALMONTE, Antoine G, DONG HO WOO, BRAT, Daniel J, EUN MI HWANG
Published in Cancer research (Chicago, Ill.) (01.02.2010)
Published in Cancer research (Chicago, Ill.) (01.02.2010)
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Melatonin Analogues Potently Inhibit MAO-B and Protect PC12 Cells against Oxidative Stress
Elkamhawy, Ahmed, Woo, Jiyu, Gouda, Noha A., Kim, Jushin, Nada, Hossam, Roh, Eun Joo, Park, Ki Duk, Cho, Jungsook, Lee, Kyeong
Published in Antioxidants (12.10.2021)
Published in Antioxidants (12.10.2021)
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