Design, Synthesis, In Vitro, and In Silico Studies of New N5-Substituted-pyrazolo[3,4-d]pyrimidinone Derivatives as Anticancer CDK2 Inhibitors
Zaki, Waheed A., El-Sayed, Selwan M., Alswah, Mohamed, El-Morsy, Ahmed, Bayoumi, Ashraf H., Mayhoub, Abrahman S., Moustafa, Walaa H., Awaji, Aeshah A., Roh, Eun Joo, Hassan, Ahmed H.E., Mahmoud, Kazem
Published in Pharmaceuticals (Basel, Switzerland) (11.11.2023)
Published in Pharmaceuticals (Basel, Switzerland) (11.11.2023)
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Highly Potent, Selective, and Competitive Indole-Based MAO-B Inhibitors Protect PC12 Cells against 6-Hydroxydopamine- and Rotenone-Induced Oxidative Stress
Elsherbeny, Mohamed H, Kim, Jushin, Gouda, Noha A, Gotina, Lizaveta, Cho, Jungsook, Pae, Ae Nim, Lee, Kyeong, Park, Ki Duk, Elkamhawy, Ahmed, Roh, Eun Joo
Published in Antioxidants (19.10.2021)
Published in Antioxidants (19.10.2021)
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Correction: Elsherbeny et al. 2-(3-Bromophenyl)-8-fluoroquinazoline-4-carboxylic Acid as a Novel and Selective Aurora A Kinase Inhibitory Lead with Apoptosis Properties: Design, Synthesis, In Vitro and In Silico Biological Evaluation. Life 2022, 12 , 876
Elsherbeny, Mohamed H, Ammar, Usama M, Abdellattif, Magda H, Abourehab, Mohammed A S, Abdeen, Ahmed, Ibrahim, Samah F, Abdelrahaman, Doaa, Mady, Wessam, Roh, Eun Joo, Elkamhawy, Ahmed
Published in Life (Basel, Switzerland) (22.03.2024)
Published in Life (Basel, Switzerland) (22.03.2024)
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Development of New Meridianin/Leucettine-Derived Hybrid Small Molecules as Nanomolar Multi-Kinase Inhibitors with Antitumor Activity
Elsherbeny, Mohamed H., Elkamhawy, Ahmed, Nada, Hossam, Abdellattif, Magda H., Lee, Kyeong, Roh, Eun Joo
Published in Biomedicines (01.09.2021)
Published in Biomedicines (01.09.2021)
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Novel Rhodanine Derivative, 5-[4-(4-Fluorophenoxy) phenyl]methylene-3-{4-[3-(4-methylpiperazin-1-yl) propoxy]phenyl}-2-thioxo-4-thiazolidinone dihydrochloride, Induces Apoptosis via Mitochondria Dysfunction and Endoplasmic Reticulum Stress in Human Colon Cancer Cells
Jung, Hye-Uk, Lee, Jeong-Hun, Chung, Kyung-Sook, Hong, Joo Young, Choi, Jung-Hye, Kim, Soo-Dong, Roh, Eun Joo, Shin, Kye Jung, Lee, Kyung-Tae
Published in Molecules (Basel, Switzerland) (06.11.2018)
Published in Molecules (Basel, Switzerland) (06.11.2018)
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Integrating computational methods guided the discovery of phytochemicals as potential Pin1 inhibitors for cancer: pharmacophore modeling, molecular docking, MM-GBSA calculations and molecular dynamics studies
Alzain, Abdulrahim A, Elbadwi, Fatima A, Shoaib, Tagyedeen H, Sherif, Asmaa E, Osman, Wadah, Ashour, Ahmed, Mohamed, Gamal A, Ibrahim, Sabrin R M, Roh, Eun Joo, Hassan, Ahmed H E
Published in Frontiers in chemistry (2024)
Published in Frontiers in chemistry (2024)
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Exploring the sedative properties of natural molecules from hop cones ( Humulus lupulus ) as promising natural anxiolytics through GABA receptors and the human serotonin transporter
Belal, Amany, Elballal, Mohammed S, Al-Karmalawy, Ahmed A, Hassan, Ahmed H E, Roh, Eun Joo, Ghoneim, Mohammed M, Ali, Mohamed A M, Obaidullah, Ahmad J, Alotaibi, Jawaher M, Shaaban, Salwa, Elanany, Mohamed A
Published in Frontiers in chemistry (10.07.2024)
Published in Frontiers in chemistry (10.07.2024)
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2-(3-Bromophenyl)-8-fluoroquinazoline-4-carboxylic Acid as a Novel and Selective Aurora A Kinase Inhibitory Lead with Apoptosis Properties: Design, Synthesis, In Vitro and In Silico Biological Evaluation
Elsherbeny, Mohamed H, Ammar, Usama M, Abdellattif, Magda H, Abourehab, Mohammed A S, Abdeen, Ahmed, Ibrahim, Samah F, Abdelrahaman, Doaa, Mady, Wessam, Roh, Eun Joo, Elkamhawy, Ahmed
Published in Life (Basel, Switzerland) (01.06.2022)
Published in Life (Basel, Switzerland) (01.06.2022)
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AF8c, a Multi-Kinase Inhibitor Induces Apoptosis by Activating DR5/Nrf2 via ROS in Colorectal Cancer Cells
Jeong, Soyeon, Farag, Ahmed K., Yun, Hye Kyeong, Jeong, Yoon A., Kim, Dae Yeong, Jo, Min Jee, Park, Seong Hye, Kim, Bo Ram, Kim, Jung Lim, Kim, Bu Gyeom, Lee, Dae-Hee, Roh, Eun Joo, Oh, Sang Cheul
Published in Cancers (21.06.2022)
Published in Cancers (21.06.2022)
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Trifluoperazine and Its Analog Suppressed the Tumorigenicity of Non-Small Cell Lung Cancer Cell; Applicability of Antipsychotic Drugs to Lung Cancer Treatment
Jeong, Joo Yeon, Park, Haangik, Yoo, Hong, Kim, Eun-Jin, Jeon, Borami, Lee, Jong Deog, Kang, Dawon, Lee, Changjoon Justin, Paek, Sun Ha, Roh, Eun Joo, Yi, Gwan-Su, Kang, Sang Soo
Published in Biomedicines (30.04.2022)
Published in Biomedicines (30.04.2022)
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Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamides as carbonic anhydrase isoforms I and II inhibitors
Al-Sanea, Mohammad M., Elkamhawy, Ahmed, Paik, Sora, Bua, Silvia, Ha Lee, So, Abdelgawad, Mohamed A., Roh, Eun Joo, Eldehna, Wagdy M., Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
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Discovery of potent and selective rhodanine type IKKβ inhibitors by hit-to-lead strategy
Song, Hyeseung, Lee, Yun Suk, Roh, Eun Joo, Seo, Jae Hong, Oh, Kwang-Seok, Lee, Byung Ho, Han, Hogyu, Shin, Kye Jung
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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Synthesis and biological evaluation of 4-piperidinecarboxylate and 4-piperidinecyanide derivatives for T-type calcium channel blockers
Woo, Hyun Min, Lee, Yun Suk, Roh, Eun Joo, Seo, Seon Hee, Song, Chi Man, Chung, Hye Jin, Pae, Ae Nim, Shin, Kye Jung
Published in Bioorganic & medicinal chemistry letters (01.10.2011)
Published in Bioorganic & medicinal chemistry letters (01.10.2011)
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Discovery of piperidinyl aminopyrimidine derivatives as IKK-2 inhibitors
Kim, Sora, Jung, Jin Kyo, Lee, Hyo Seon, Kim, Youngjae, Kim, Jiyoon, Choi, Kihang, Baek, Du-Jong, Moon, Bongjin, Oh, Kwang-Seok, Lee, Byung Ho, Shin, Kye Jung, Pae, Ae Nim, Nam, Ghilsoo, Roh, Eun Joo, Cho, Yong Seo, Choo, Hyunah
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Cr(salen) catalysed asymmetric ring opening reactions of epoxides in room temperature ionic liquids
Song, CE, Oh, CR, Roh, EJ, Choo, DJ
Published in Chemical communications (Cambridge, England) (01.01.2000)
Published in Chemical communications (Cambridge, England) (01.01.2000)
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