Novel conformationally constrained analogues of agomelatine as new melatoninergic ligands
Rami, Marouan, Landagaray, Elodie, Ettaoussi, Mohamed, Boukhalfa, Koussayla, Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Published in Molecules (Basel, Switzerland) (24.12.2012)
Published in Molecules (Basel, Switzerland) (24.12.2012)
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Journal Article
Melatonin MT1 receptor as a novel target in neuropsychopharmacology: MT1 ligands, pathophysiological and therapeutic implications, and perspectives
Comai, Stefano, Lopez-Canul, Martha, De Gregorio, Danilo, Posner, Ada, Ettaoussi, Mohamed, Guarnieri, Fabrizia Claudia, Gobbi, Gabriella
Published in Pharmacological research (01.06.2019)
Published in Pharmacological research (01.06.2019)
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Selective Enhancement of REM Sleep in Male Rats through Activation of Melatonin MT 1 Receptors Located in the Locus Ceruleus Norepinephrine Neurons
López-Canul, Martha, He, Qianzi, Sasson, Tania, Ettaoussi, Mohamed, Gregorio, Danilo De, Ochoa-Sanchez, Rafael, Catoire, Helene, Posa, Luca, Rouleau, Guy, Beaulieu, Jean Martin, Comai, Stefano, Gobbi, Gabriella
Published in The Journal of neuroscience (17.07.2024)
Published in The Journal of neuroscience (17.07.2024)
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Journal Article
Selective Enhancement of REM Sleep in Male Rats through Activation of Melatonin MT1 Receptors Located in the Locus Ceruleus Norepinephrine Neurons
López-Canul, Martha, He, Qianzi, Sasson, Tania, Ettaoussi, Mohamed, De Gregorio, Danilo, Ochoa-Sanchez, Rafael, Catoire, Helene, Posa, Luca, Rouleau, Guy, Beaulieu, Jean Martin, Comai, Stefano, Gobbi, Gabriella
Published in The Journal of neuroscience (17.07.2024)
Published in The Journal of neuroscience (17.07.2024)
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Journal Article
Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine
Bolteau, Raphaël, Descamps, Florian, Ettaoussi, Mohamed, Caignard, Daniel H., Delagrange, Philippe, Melnyk, Patricia, Yous, Saïd
Published in European journal of medicinal chemistry (01.03.2020)
Published in European journal of medicinal chemistry (01.03.2020)
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Journal Article
Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT1/MT2) and serotoninergic (5-HT2C) dual ligands
Duroux, Romain, Rami, Marouan, Landagaray, Elodie, Ettaoussi, Mohamed, Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Yous, Saïd
Published in European journal of medicinal chemistry (01.12.2017)
Published in European journal of medicinal chemistry (01.12.2017)
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Journal Article
Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitors
Kufareva, Irina, Bestgen, Benoit, Brear, Paul, Prudent, Renaud, Laudet, Béatrice, Moucadel, Virginie, Ettaoussi, Mohamed, Sautel, Celine F, Krimm, Isabelle, Engel, Matthias, Filhol, Odile, Borgne, Marc Le, Lomberget, Thierry, Cochet, Claude, Abagyan, Ruben
Published in Scientific reports (04.11.2019)
Published in Scientific reports (04.11.2019)
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Journal Article
Synthesis and SAR Studies of Isoquinoline and Tetrahydroisoquinoline Derivatives as Melatonin Receptor Ligands
Ettaoussi, Mohamed, Laversin, Amélie, Vreulz, Brandon, Rami, Marouane, Lebegue, Nicolas, Delagrange, Philippe, Caignard, Daniel Henri, Melnyk, Patricia, Liberelle, Maxime, Yous, Saïd
Published in ChemMedChem (04.02.2022)
Published in ChemMedChem (04.02.2022)
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Journal Article
New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation
Landagaray, Elodie, Ettaoussi, Mohamed, Rami, Marouan, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Berthelot, Pascal, Yous, Saïd
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
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Journal Article
Design, synthesis and pharmacological evaluation of new series of naphthalenic analogues as melatoninergic (MT1/MT2) and serotoninergic 5-HT2C dual ligands (I)
Ettaoussi, Mohamed, Sabaouni, Ahmed, Rami, Marouan, Boutin, Jean A., Delagrange, Philippe, Renard, Pierre, Spedding, Michael, Caignard, Daniel-Henri, Berthelot, Pascal, Yous, Saïd
Published in European journal of medicinal chemistry (01.03.2012)
Published in European journal of medicinal chemistry (01.03.2012)
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Journal Article
New melatonin (MT1/MT2) ligands: Design and synthesis of (8,9-dihydro-7H-furo[3,2-f]chromen-1-yl) derivatives
Landagaray, Elodie, Ettaoussi, Mohamed, Leclerc, Véronique, Traoré, Balla, Perez, Valérie, Nosjean, Olivier, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Published in Bioorganic & medicinal chemistry (01.02.2014)
Published in Bioorganic & medicinal chemistry (01.02.2014)
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Journal Article
Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives
Landagaray, Elodie, Ettaoussi, Mohamed, Duroux, Romain, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Berthelot, Pascal, Yous, Saïd
Published in European journal of medicinal chemistry (15.02.2016)
Published in European journal of medicinal chemistry (15.02.2016)
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Journal Article
Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II)
Ettaoussi, Mohamed, Pérès, Basile, Errazani, Aïcha, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Berthelot, Pascal, Yous, Saïd
Published in European journal of medicinal chemistry (27.01.2015)
Published in European journal of medicinal chemistry (27.01.2015)
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Journal Article
Melatonin MT 1 receptor as a novel target in neuropsychopharmacology: MT 1 ligands, pathophysiological and therapeutic implications, and perspectives
Comai, Stefano, Lopez-Canul, Martha, De Gregorio, Danilo, Posner, Ada, Ettaoussi, Mohamed, Guarnieri, Fabrizia Claudia, Gobbi, Gabriella
Published in Pharmacological research (01.06.2019)
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Published in Pharmacological research (01.06.2019)
Journal Article
Synthesis and Pharmacological Evaluation of a series of the Agomelatine Analogues as Melatonin MT1/MT2 Agonist and 5-HT2C Antagonist
Ettaoussi, Mohamed, Sabaouni, Ahmed, Pérès, Basile, Landagaray, Elodie, Nosjean, Olivier, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Published in ChemMedChem (01.11.2013)
Published in ChemMedChem (01.11.2013)
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Journal Article
Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3
Leclerc, Veronique, Ettaoussi, Mohamed, Rami, Marouan, Farce, Amaury, Boutin, Jean Albert, Delagrange, Philippe, Caignard, Daniel-Henri, Renard, Pierre, Berthelot, Pascal, Yous, Said
Published in European journal of medicinal chemistry (01.05.2011)
Published in European journal of medicinal chemistry (01.05.2011)
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Journal Article
Synthesis and Pharmacological Evaluation of a series of the Agomelatine Analogues as Melatonin MT 1 /MT 2 Agonist and 5‐HT 2C Antagonist
Ettaoussi, Mohamed, Sabaouni, Ahmed, Pérès, Basile, Landagaray, Elodie, Nosjean, Olivier, Boutin, Jean A., Caignard, Daniel‐Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Published in ChemMedChem (01.11.2013)
Published in ChemMedChem (01.11.2013)
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Journal Article
Synthesis, chiral resolution, absolute configuration assignment and pharmacological evaluation of a series of melatoninergic ligandsElectronic supplementary information (ESI) available. See DOI: 10.1039/c4md00149d
Ettaoussi, Mohamed, Pérès, Basile, Jarry, Christian, Nosjean, Olivier, Boutin, Jean A, Gohier, Arnaud, Mannoury la Cour, Clotilde, Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Year of Publication 20.08.2014
Year of Publication 20.08.2014
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