Discovery of BAY 94-8862: A Nonsteroidal Antagonist of the Mineralocorticoid Receptor for the Treatment of Cardiorenal Diseases
Bärfacker, Lars, Kuhl, Alexander, Hillisch, Alexander, Grosser, Rolf, Figueroa-Pérez, Santiago, Heckroth, Heike, Nitsche, Adam, Ergüden, Jens-Kerim, Gielen-Haertwig, Heike, Schlemmer, Karl-Heinz, Mittendorf, Joachim, Paulsen, Holger, Platzek, Johannes, Kolkhof, Peter
Published in ChemMedChem (01.08.2012)
Published in ChemMedChem (01.08.2012)
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Discovery of Molidustat (BAY 85‐3934): A Small‐Molecule Oral HIF‐Prolyl Hydroxylase (HIF‐PH) Inhibitor for the Treatment of Renal Anemia
Beck, Hartmut, Jeske, Mario, Thede, Kai, Stoll, Friederike, Flamme, Ingo, Akbaba, Metin, Ergüden, Jens‐Kerim, Karig, Gunter, Keldenich, Jörg, Oehme, Felix, Militzer, Hans‐Christian, Hartung, Ingo V., Thuss, Uwe
Published in ChemMedChem (23.05.2018)
Published in ChemMedChem (23.05.2018)
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Cover Picture: Discovery of BAY 94-8862: A Nonsteroidal Antagonist of the Mineralocorticoid Receptor for the Treatment of Cardiorenal Diseases (ChemMedChem 8/2012)
Bärfacker, Lars, Kuhl, Alexander, Hillisch, Alexander, Grosser, Rolf, Figueroa-Pérez, Santiago, Heckroth, Heike, Nitsche, Adam, Ergüden, Jens-Kerim, Gielen-Haertwig, Heike, Schlemmer, Karl-Heinz, Mittendorf, Joachim, Paulsen, Holger, Platzek, Johannes, Kolkhof, Peter
Published in ChemMedChem (01.08.2012)
Published in ChemMedChem (01.08.2012)
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A Novel Route to 6-Substituted Piperidin-3-ols via Domino Cyclization of 2-Hydroxy-6-phosphinyl-5-hexenyl Tosylates with Primary Amines: Synthesis of (+/-)-Pseudoconhydrine and (+/-)-epi-Pseudoconhydrine
Scherner, Cathrin, Ergueden, Jens-Kerim, Adiwidjaja, Gunadi, Schaumann, Ernst
Published in Synthesis (Stuttgart) (2014)
Published in Synthesis (Stuttgart) (2014)
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Selective Indole-Based ECE Inhibitors: Synthesis and Pharmacological Evaluation
Brands, Michael, Ergüden, Jens-Kerim, Hashimoto, Kentaro, Heimbach, Dirk, Krahn, Thomas, Schröder, Christian, Siegel, Stephan, Stasch, Johannes-Peter, Tsujishita, Hideki, Weigand, Stefan, Yoshida, Nagahiro H.
Published in ChemMedChem (01.01.2006)
Published in ChemMedChem (01.01.2006)
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Novel, selective indole-based ECE inhibitors: Lead optimization via solid-phase and classical synthesis
Brands, Michael, Ergüden, Jens-Kerim, Hashimoto, Kentaro, Heimbach, Dirk, Schröder, Christian, Siegel, Stephan, Stasch, Johannes-Peter, Weigand, Stefan
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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Front Cover: Discovery of Molidustat (BAY 85‐3934): A Small‐Molecule Oral HIF‐Prolyl Hydroxylase (HIF‐PH) Inhibitor for the Treatment of Renal Anemia (ChemMedChem 10/2018)
Beck, Hartmut, Jeske, Mario, Thede, Kai, Stoll, Friederike, Flamme, Ingo, Akbaba, Metin, Ergüden, Jens‐Kerim, Karig, Gunter, Keldenich, Jörg, Oehme, Felix, Militzer, Hans‐Christian, Hartung, Ingo V., Thuss, Uwe
Published in ChemMedChem (23.05.2018)
Published in ChemMedChem (23.05.2018)
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SUBSTITUTED DIHYDROPYRAZOLONES AND THEIR USE
OEHME, FELIX, AKBABA, METIN, ERGUDEN, JENS-KERIM, FLAMME, INGO, WILD, HANNO, KELDENICH, JORG, THEDE, KAI, STOLL, FRIEDERIKE, JESKE, MARIO, SCHUMACHER, JOACHIM, KOLKHOF, PETER, BECK, HARTMUT
Year of Publication 22.04.2019
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Year of Publication 22.04.2019
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DIHIDROPIRAZOLONAS SUSTITUIDAS PARA EL TRATAMIENTO DE ENFERMEDADES CARDIOVASCULARES Y HEMATOLÓGICAS
KELDENICH, JÖRG, OEHME, FELIX, AKBABA, METIN, ERGUDEN, JENS-KERIM, FLAMME, INGO, SCHUHMACHER, JOACHIM, WILD, HANNO, THEDE, KAI, STOLL, FRIEDERIKE, JESKE, MARIO, KOLKHOF, PETER, BECK, HARTMUT
Year of Publication 26.12.2014
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Year of Publication 26.12.2014
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DIHIDROPIRAZOLONAS SUSTITUIDAS
OEHME, FELIX, AKBABA, METIN, ERGUDEN, JENS-KERIM, FLAMME, INGO, SCHUHMACHER, JOACHIM, WILD, HANNO, KELDENICH, JORG, THEDE, KAI, STOLL, FRIEDERIKE, JESKE, MARIO, KOLKHOF, PETER, BECK, HARTMUT
Year of Publication 16.09.2014
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Year of Publication 16.09.2014
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SUBSTITUTED DIHYDROPYRAZOLONES FOR TREATING CARDIOVASCULAR AND HAEMATOLOGICAL DISEASES
ERGUDEN, Jens-Kerim, JESKE, Mario, SCHUHMACHER, Joachim, THEDE, Kai, OEHME, Felix, KELDENICH, Jorg, FLAMME, Ingo, KOLKHOF, Peter, BECK, Hartmut, WILD, Hanno, AKBABA, Metin, STOLL, Friederike
Year of Publication 08.09.2014
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Year of Publication 08.09.2014
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Substituted dihydropyrazolones for treating cardiovascular and haematological diseases
OEHME, FELIX, AKBABA, METIN, ERGUDEN, JENS-KERIM, FLAMME, INGO, WILD, HANNO, KELDENICH, JORG, SCHUHMACHER, JOACHIM, THEDE, KAI, STOLL, FRIEDERIKE, JESKE, MARIO, BECK, HARTMUT, KOLKHOF, PETER
Year of Publication 07.11.2013
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Year of Publication 07.11.2013
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SUBSTITUTED DIHYDROPYRAZOLONES FOR TREATING CARDIOVASCULAR AND HAEMATOLOGICAL DISEASES
JESKE MARIO, SCHUHMACHER JOACHIM, FLAMME INGO, OEHME FELIX, ERGUDEN JENS-KERIM, AKBABA METIN, BECK HARTMUT, THEDE KAI, KOLKHOF PETER, STOLL FRIEDERIKE, WILD HANNO, KELDENICH JORG
Year of Publication 30.10.2013
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Year of Publication 30.10.2013
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SUBSTITUTED DIHYDROPYRAZOLONES FOR TREATING CARDIOVASCULAR AND HAEMATOLOGICAL DISEASES
OEHME, FELIX, AKBABA, METIN, ERGUDEN, JENS-KERIM, FLAMME, INGO, SCHUHMACHER, JOACHIM, WILD, HANNO, KELDENICH, JORG, THEDE, KAI, STOLL, FRIEDERIKE, JESKE, MARIO, KOLKHOF, PETER, BECK, HARTMUT
Year of Publication 31.05.2013
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Year of Publication 31.05.2013
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DIHIDROPIRAZOLONAS SUSTITUIDAS COMO INHIBIDORES DE HIF-PROPIL-4-HIDROXILASAS
OEHME, FELIX, AKBABA, METIN, ERGUDEN, JENS-KERIM, FLAMME, INGO, SCHUHMACHER, JOACHIM, WILD, HANNO, KELDENICH, JORG, THEDE, KAI, STOLL, FRIEDERIKE, JESKE, MARIO, KOLKHOF, PETER, BECK, HARTMUT
Year of Publication 27.05.2012
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Year of Publication 27.05.2012
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DIHIDROPIRAZOLONAS SUSTITUIDAS COMO INHIBIDORES DE HIF-PROPIL-4-HIDROXILASAS
OEHME, FELIX, AKBABA, METIN, ERGUDEN, JENS-KERIM, FLAMME, INGO, SCHUHMACHER, JOACHIM, WILD, HANNO, KELDENICH, JORG, THEDE, KAI, STOLL, FRIEDERIKE, JESKE, MARIO, KOLKHOF, PETER, BECK, HARTMUT
Year of Publication 20.05.2012
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Year of Publication 20.05.2012
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SUBSTITUTED DIHYDROPYRAZOLON FOR THE TREATMENT OF CARDIOVASCULAR AND HAEMATOLOGICAL DISEASES
OEHME, FELIX, AKBABA, METIN, ERGUDEN, JENS-KERIM, FLAMME, INGO, JESKE MARIO, SCHUHMACHER JOACHIM, WILD, HANNO, KELDENICH, JORG, THEDE, KAI, BECK HARTMUT, STOLL FRIEDERIKE, KOLKHOF, PETER
Year of Publication 25.04.2012
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Year of Publication 25.04.2012
Patent