Novel Sulfonamide-Based Carbamates as Selective Inhibitors of BChE
Magar, Pratibha, Parravicini, Oscar, Štěpánková, Šárka, Svrčková, Katarina, Garro, Adriana D., Jendrzejewska, Izabela, Pauk, Karel, Hošek, Jan, Jampílek, Josef, Enriz, Ricardo D., Imramovský, Aleš
Published in International journal of molecular sciences (01.09.2021)
Published in International journal of molecular sciences (01.09.2021)
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Synthesis and antifungal activity of ( Z)-5-arylidenerhodanines
Sortino, Maximiliano, Delgado, Paula, Juárez, Sabina, Quiroga, Jairo, Abonía, Rodrigo, Insuasty, Braulio, Nogueras, Manuel, Rodero, Laura, Garibotto, Francisco M., Enriz, Ricardo D., Zacchino, Susana A.
Published in Bioorganic & medicinal chemistry (2007)
Published in Bioorganic & medicinal chemistry (2007)
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Synthesis, Analysis, Cholinesterase-Inhibiting Activity and Molecular Modelling Studies of 3-(Dialkylamino)-2-hydroxypropyl 4-[(Alkoxy-carbonyl)amino]benzoates and Their Quaternary Ammonium Salts
Padrtova, Tereza, Marvanova, Pavlina, Odehnalova, Klara, Kubinova, Renata, Parravicini, Oscar, Garro, Adriana, Enriz, Ricardo D, Humpa, Otakar, Oravec, Michal, Mokry, Petr
Published in Molecules (Basel, Switzerland) (23.11.2017)
Published in Molecules (Basel, Switzerland) (23.11.2017)
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Pentameric models as alternative molecular targets for the design of new antiaggregant agents
Barrera Guisasola, Exequiel E, Gutierrez, Lucas J, Andujar, Sebastián A, Angelina, Emilio, Rodríguez, Ana M, Enriz, Ricardo D
Published in Current protein & peptide science (01.03.2016)
Published in Current protein & peptide science (01.03.2016)
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Arylated analogues of cypronazole: fungicidal effect and activity on human fibroblasts. Docking analysis and molecular dynamics simulations
Herrera Cano, Natividad, Andujar, Sebastian A., Theoduloz, Cristina, Wunderlin, Daniel A., Santiago, Ana N., Schmeda-Hirschmann, Guillermo, Enriz, Ricardo D., Feresin, Gabriela E.
Published in Natural products and bioprospecting (01.12.2022)
Published in Natural products and bioprospecting (01.12.2022)
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Structural requirements for the antifungal activities of natural drimane sesquiterpenes and analogues, supported by conformational and electronic studies
Derita, Marcos, Montenegro, Iván, Garibotto, Francisco, Enriz, Ricardo D, Fritis, Mauricio Cuellar, Zacchino, Susana A
Published in Molecules (Basel, Switzerland) (05.02.2013)
Published in Molecules (Basel, Switzerland) (05.02.2013)
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Benzopyran hydrazones with dual PPARα/γ or PPARα/δ agonism and an anti-inflammatory effect on human THP-1 macrophages
García, Ainhoa, Vila, Laura, Duplan, Isabelle, Schiel, María Ayelén, Enriz, Ricardo D., Hennuyer, Nathalie, Staels, Bart, Cabedo, Nuria, Cortes, Diego
Published in European journal of medicinal chemistry (05.02.2024)
Published in European journal of medicinal chemistry (05.02.2024)
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Synthesis of a new 2-prenylated quinoline as potential drug for metabolic syndrome with pan-PPAR activity and anti-inflammatory effects
Villarroel-Vicente, Carlos, García, Ainhoa, Zibar, Khamis, Schiel, María Ayelén, Ferri, Jordi, Hennuyer, Nathalie, Enriz, Ricardo D., Staels, Bart, Cortes, Diego, Cabedo, Nuria
Published in Bioorganic & medicinal chemistry letters (01.07.2024)
Published in Bioorganic & medicinal chemistry letters (01.07.2024)
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Structure–activity relationship study of homoallylamines and related derivatives acting as antifungal agents
Suvire, Fernando D., Sortino, Maximiliano, Kouznetsov, Vladimir V., Vargas M, Leonor Y., Zacchino, Susana A., Cruz, Uriel Mora, Enriz, Ricardo D.
Published in Bioorganic & medicinal chemistry (15.03.2006)
Published in Bioorganic & medicinal chemistry (15.03.2006)
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Second generation of pyrimidin-quinolone hybrids obtained from virtual screening acting as sphingosine kinase 1 inhibitors and potential anticancer agents
Vettorazzi, Marcela, Díaz, Iván, Angelina, Emilio, Salido, Sofía, Gutierrez, Lucas, Alvarez, Sergio E., Cobo, Justo, Enriz, Ricardo D.
Published in Bioorganic chemistry (01.03.2024)
Published in Bioorganic chemistry (01.03.2024)
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Computer-aided structure-based optimization of 4,5,6,7-tetrahydrobenzo[]thiazole-2,6-diamine derivatives as DNA gyrase B inhibitors
Gutierrez, Lucas J, Vettorazzi, Marcela, Dernovšek, Jaka, Durcik, Martina, Maši, Lucija Peterlin, Tomaši, Tihomir, Enriz, Ricardo D
Published in New journal of chemistry (20.02.2023)
Published in New journal of chemistry (20.02.2023)
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New short cationic antibacterial peptides. Synthesis, biological activity and mechanism of action
Lima, Beatriz, Ricci, Maria, Garro, Adriana, Juhász, Tünde, Szigyártó, Imola Csilla, Papp, Zita I., Feresin, Gabriela, Garcia de la Torre, Jose, Lopez Cascales, Javier, Fülöp, Lívia, Beke-Somfai, Tamás, Enriz, Ricardo D.
Published in Biochimica et biophysica acta. Biomembranes (01.10.2021)
Published in Biochimica et biophysica acta. Biomembranes (01.10.2021)
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Conformational and electronic study of dopamine interacting with the D2 dopamine receptor
Tosso, Rodrigo D., Parravicini, Oscar, Zarycz, M. Natalia C., Angelina, Emilio, Vettorazzi, Marcela, Peruchena, Nélida, Andujar, Sebastián, Enriz, Ricardo D.
Published in Journal of computational chemistry (05.08.2020)
Published in Journal of computational chemistry (05.08.2020)
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Evaluating the conformational space of the active site of D 2 dopamine receptor. Scope and limitations of the standard docking methods
Tosso, Rodrigo D, Zarycz, M Natalia C, Schiel, Ayelén, Goicoechea Moro, Luisa, Baldoni, Héctor A, Angelina, Emilio, Enriz, Ricardo D
Published in Journal of computational chemistry (15.07.2022)
Published in Journal of computational chemistry (15.07.2022)
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The Mechanism of Antimicrobial Small-Cationic Peptides from Coarse-Grained Simulations
Frigini, Ezequiel N., Porasso, Rodolfo D., Beke-Somfai, Tamás, López Cascales, José Javier, Enriz, Ricardo D., Pantano, Sergio
Published in Journal of chemical information and modeling (13.11.2023)
Published in Journal of chemical information and modeling (13.11.2023)
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Anti-inflammatory effects and improved metabolic derangements in ob/ob mice by a newly synthesized prenylated benzopyran with pan-PPAR activity
Marques, Patrice, Villarroel-Vicente, Carlos, Collado, Aida, García, Ainhoa, Vila, Laura, Duplan, Isabelle, Hennuyer, Nathalie, Garibotto, Francisco, Enriz, Ricardo D., Dacquet, Catherine, Staels, Bart, Piqueras, Laura, Cortes, Diego, Sanz, María-Jesús, Cabedo, Nuria
Published in Pharmacological research (01.01.2023)
Published in Pharmacological research (01.01.2023)
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Targeting defective sphingosine kinase 1 in Niemann–Pick type C disease with an activator mitigates cholesterol accumulation
Newton, Jason, Palladino, Elisa N.D., Weigel, Cynthia, Maceyka, Michael, Gräler, Markus H., Senkal, Can E., Enriz, Ricardo D., Marvanova, Pavlina, Jampilek, Josef, Lima, Santiago, Milstien, Sheldon, Spiegel, Sarah
Published in The Journal of biological chemistry (03.07.2020)
Published in The Journal of biological chemistry (03.07.2020)
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Journal Article
Evaluating the conformational space of the active site of D2 dopamine receptor. Scope and limitations of the standard docking methods
Tosso, Rodrigo D., Zarycz, M. Natalia C., Schiel, Ayelén, Goicoechea Moro, Luisa, Baldoni, Héctor A., Angelina, Emilio, Enriz, Ricardo D.
Published in Journal of computational chemistry (15.07.2022)
Published in Journal of computational chemistry (15.07.2022)
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