Activating the Wnt/β-Catenin Pathway for the Treatment of Melanoma--Application of LY2090314, a Novel Selective Inhibitor of Glycogen Synthase Kinase-3
Atkinson, Jennifer M, Rank, Kenneth B, Zeng, Yi, Capen, Andrew, Yadav, Vipin, Manro, Jason R, Engler, Thomas A, Chedid, Marcio
Published in PloS one (27.04.2015)
Published in PloS one (27.04.2015)
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A robust high-content imaging approach for probing the mechanism of action and phenotypic outcomes of cell-cycle modulators
Sutherland, Jeffrey J, Low, Jonathan, Blosser, Wayne, Dowless, Michele, Engler, Thomas A, Stancato, Louis F
Published in Molecular cancer therapeutics (01.02.2011)
Published in Molecular cancer therapeutics (01.02.2011)
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The Glycogen Synthase Kinase-3β Inhibitor LSN 2105786 Promotes Zebrafish Fin Regeneration
Sarmah, Swapnalee, Curtis, Courtney, Mahin, Jennifer, Farrell, Mark, Engler, Thomas A, Sanchez-Felix, Manuel V, Sato, Masahiko, Ma, Yanfai Linda, Chu, Shaoyou, Marrs, James A
Published in Biomedicines (19.04.2019)
Published in Biomedicines (19.04.2019)
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Changes in Osteoblast, Chondrocyte, and Adipocyte Lineages Mediate the Bone Anabolic Actions of PTH and Small Molecule GSK-3 Inhibitor
Kulkarni, Nalini H., Wei, Tao, Kumar, Amar, Dow, Ernst R., Stewart, Trent R., Shou, Jianyong, N'cho, Mathias, Sterchi, Diane L., Gitter, Bruce D., Higgs, Richard E., Halladay, David L., Engler, Thomas A., Martin, T. John, Bryant, Henry U., Ma, Yanfei L., Onyia, Jude E.
Published in Journal of cellular biochemistry (15.12.2007)
Published in Journal of cellular biochemistry (15.12.2007)
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Chemical Proteomic Characterization of a Covalent KRASG12C Inhibitor
Wijeratne, Aruna, Xiao, Junpeng, Reutter, Christopher, Furness, Kelly W, Leon, Rebecca, Zia-Ebrahimi, Mohammad, Cavitt, Rachel N, Strelow, John M, Van Horn, Robert D, Peng, Sheng-Bin, Barda, David A, Engler, Thomas A, Chalmers, Michael J
Published in ACS medicinal chemistry letters (14.06.2018)
Published in ACS medicinal chemistry letters (14.06.2018)
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The development of potent and selective bisarylmaleimide GSK3 inhibitors
Engler, Thomas A., Malhotra, Sushant, Burkholder, Timothy P., Henry, James R., Mendel, David, Porter, Warren J., Furness, Kelly, Diefenbacher, Clive, Marquart, Angela, Reel, Jon K., Li, Yihong, Clayton, Joshua, Cunningham, Brian, McLean, Johnathan, O’Toole, John C., Brozinick, Joseph, Hawkins, Eric, Misener, Elizabeth, Briere, Daniel, Brier, Richard A., Wagner, Jill R., Campbell, Robert M., Anderson, Bryan D., Vaughn, Renee, Bennett, Donald B., Meier, Timothy I., Cook, James A.
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
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Synthesis of 1,7-annulated indoles and their applications in the studies of cyclin dependent kinase inhibitors
Zhu, Guoxin, Conner, Scott E., Zhou, Xun, Chan, Ho-Kit, Shih, Chuan, Engler, Thomas A., Al-awar, Rima S., Brooks, Harold B., Watkins, Scott A., Spencer, Charles D., Schultz, Richard M., Dempsey, Jack A., Considine, Eileen L., Patel, Bharvin R., Ogg, Catherine A., Vasudevan, Vasu, Lytle, Michelle L.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Synthetic Approaches to Indolo[6,7-a]pyrrolo[3,4-c]carbazoles: Potent Cyclin D1/CDK4 Inhibitors
Faul, Margaret M, Engler, Thomas A, Sullivan, Kevin A, Grutsch, John L, Clayton, Marcella T, Martinelli, Michael J, Pawlak, Joseph M, LeTourneau, Michael, Coffey, D. Scott, Pedersen, Steven W, Kolis, Stanley P, Furness, Kelly, Malhotra, Sushant, Al-awar, Rima S, Ray, James E
Published in Journal of organic chemistry (30.04.2004)
Published in Journal of organic chemistry (30.04.2004)
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Asymmetric Reactions of 2-Methoxy-1,4-benzoquinones with Styrenyl Systems: Enantioselective Syntheses of 8-Aryl-3-methoxybicyclo[4.2.0]oct-3-en-2,5-diones, 7-Aryl-3-hydroxybicyclo[3.2.1]oct-3-en-2,8-diones, 2-Aryl-6-methoxy-2,3-dihydrobenzofuran-5-ols, and Pterocarpans
Engler, Thomas A, Letavic, Michael A, Iyengar, Rajesh, LaTessa, Kenneth O, Reddy, Jayachandra P
Published in Journal of organic chemistry (02.04.1999)
Published in Journal of organic chemistry (02.04.1999)
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Lewis Acid-Controlled Regioselectivity in Reactions of Styrenyl Systems with Benzoquinone Monoimides: New Regioselective Syntheses of Substituted 2-Aryl-2,3-dihydrobenzofurans, 2-Aryl-2,3-dihydroindoles, and 2-Arylindoles
Engler, Thomas A, Chai, Wenying, LaTessa, Kenneth O
Published in Journal of organic chemistry (27.12.1996)
Published in Journal of organic chemistry (27.12.1996)
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Stereospecific Lewis Acid-Promoted Reactions of Styrenyl Systems with 2-Alkoxy-(6-Alkyl)-1,4-Benzoquinones: Scope, Limitations, and Synthetic Applications
Engler, Thomas A, Combrink, Keith D, Letavic, Michael A, Lynch, Kenneth O, Ray, James E
Published in Journal of organic chemistry (01.11.1994)
Published in Journal of organic chemistry (01.11.1994)
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Tandem 5 + 2/3 + 2 and 5 + 2/3 + 3 Cycloaddition Reactions
Engler, Thomas A, Scheibe, Cynthia M, Iyengar, Rajesh
Published in Journal of organic chemistry (28.11.1997)
Published in Journal of organic chemistry (28.11.1997)
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Lewis Acid-Promoted Reactions of Unsymmetrically Substituted Stilbenes with 2-Methoxy-1,4-benzoquinones: Stereoselective Synthesis of trans-2,3-Diaryl-2,3-dihydrobenzofurans
Engler, Thomas A, Gfesser, Gregory A, Draney, Bill W
Published in Journal of organic chemistry (01.06.1995)
Published in Journal of organic chemistry (01.06.1995)
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