Direct Nucleophilic SN1-Type Reactions of Alcohols
Emer, Enrico, Sinisi, Riccardo, Capdevila, Montse Guiteras, Petruzziello, Diego, De Vincentiis, Francesco, Cozzi, Pier Giorgio
Published in European Journal of Organic Chemistry (01.02.2011)
Published in European Journal of Organic Chemistry (01.02.2011)
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Book Review
Journal Article
SN1-Type Reactions in the Presence of Water: Indium(III)-Promoted Highly Enantioselective Organocatalytic Propargylation of Aldehydes
Sinisi, Riccardo, Vita, Maria Victoria, Gualandi, Andrea, Emer, Enrico, Cozzi, Pier Giorgio
Published in Chemistry : a European journal (27.06.2011)
Published in Chemistry : a European journal (27.06.2011)
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Journal Article
Innovative Catalytic Protocols for the Ring-Closing Friedel-Crafts-Type Alkylation and Alkenylation of Arenes
Bandini, Marco, Emer, Enrico, Tommasi, Simona, Umani-Ronchi, Achille
Published in European Journal of Organic Chemistry (01.08.2006)
Published in European Journal of Organic Chemistry (01.08.2006)
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Book Review
Journal Article
Synthesis of SMT022357 enantiomers and in vivo evaluation in a Duchenne muscular dystrophy mouse model
Babbs, Arran, Berg, Adam, Chatzopoulou, Maria, Davies, Kay E., Davies, Stephen G., Edwards, Benjamin, Elsey, David J., Emer, Enrico, Figuccia, Aude L.A., Fletcher, Ai M., Guiraud, Simon, Harriman, Shawn, Moir, Lee, Robinson, Neil, Rowley, Jessica A., Russell, Angela J., Squire, Sarah E., Thomson, James E., Tinsley, Jonathon M., Wilson, Francis X., Wynne, Graham M.
Published in Tetrahedron (10.01.2020)
Published in Tetrahedron (10.01.2020)
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Journal Article
Derisking the Cu-Mediated 18F‑Fluorination of Heterocyclic Positron Emission Tomography Radioligands
Taylor, Nicholas J, Emer, Enrico, Preshlock, Sean, Schedler, Michael, Tredwell, Matthew, Verhoog, Stefan, Mercier, Joel, Genicot, Christophe, Gouverneur, Véronique
Published in Journal of the American Chemical Society (21.06.2017)
Published in Journal of the American Chemical Society (21.06.2017)
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Journal Article
Derisking the Cu-Mediated F-18-Fluorination of Heterocyclic Positron Emission Tomography Radioligands
Taylor, Nicholas J., Emer, Enrico, Preshlock, Sean, Schedler, Michael, Tredwell, Matthew, Verhoog, Stefan, Mercier, Joel, Genicot, Christophe, Gouverneur, Veronique
Published in Journal of the American Chemical Society (21.06.2017)
Published in Journal of the American Chemical Society (21.06.2017)
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Journal Article
Diversity-Oriented Approach to CF3CHF-, CF3CFBr-, CF3CF2-, (CF3)(2)CH-, and CF3(SCF3)CH-Substituted Arenes from 1-(Diazo-2,2,2-trifluoroethyl)arenes
Emer, Enrico, Twilton, Jack, Tredwell, Matthew, Calderwood, Samuel, Collier, Thomas Lee, Liegault, Benoit, Taillefer, Marc, Gouvemeur, Veronique
Published in Organic letters (21.11.2014)
Published in Organic letters (21.11.2014)
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Journal Article
Atroposelective Organocatalysis
Cozzi, Pier Giorgio, Emer, Enrico, Gualandi, Andrea
Published in Angewandte Chemie (International ed.) (18.04.2011)
Published in Angewandte Chemie (International ed.) (18.04.2011)
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Journal Article
Diversity-Oriented Approach to CF3CHF‑, CF3CFBr‑, CF3CF2‑, (CF3)2CH‑, and CF3(SCF3)CH-Substituted Arenes from 1‑(Diazo-2,2,2-trifluoroethyl)arenes
Emer, Enrico, Twilton, Jack, Tredwell, Matthew, Calderwood, Samuel, Collier, Thomas Lee, Liégault, Benoît, Taillefer, Marc, Gouverneur, Véronique
Published in Organic letters (21.11.2014)
Published in Organic letters (21.11.2014)
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Journal Article
Highly Enantioselective α Alkylation of Aldehydes with 1,3-Benzodithiolylium Tetrafluoroborate: A Formal Organocatalytic α Alkylation of Aldehydes by the Carbenium Ion
Gualandi, Andrea, Emer, Enrico, Capdevila, Montse Guiteras, Cozzi, Pier Giorgio
Published in Angewandte Chemie (International ed.) (16.08.2011)
Published in Angewandte Chemie (International ed.) (16.08.2011)
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Journal Article
S(N)1-Type Reactions in the Presence of Water: Indium(III)-Promoted Highly Enantioselective Organocatalytic Propargylation of Aldehydes
Sinisi, Riccardo, Vita, Maria Victoria, Gualandi, Andrea, Emer, Enrico, Cozzi, Pier Giorgio
Published in Chemistry : a European journal (27.06.2011)
Published in Chemistry : a European journal (27.06.2011)
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Journal Article
His-tagged Horse Liver Alcohol Dehydrogenase: Immobilization and application in the bio-based enantioselective synthesis of (S)-arylpropanols
Quaglia, Daniela, Pori, Matteo, Galletti, Paola, Emer, Enrico, Paradisi, Francesca, Giacomini, Daria
Published in Process biochemistry (1991) (01.06.2013)
Published in Process biochemistry (1991) (01.06.2013)
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Journal Article
Structure-activity relationships of 2-pyrimidinecarbohydrazides as utrophin modulators for the potential treatment of Duchenne muscular dystrophy
Chatzopoulou, Maria, Conole, Daniel, Emer, Enrico, Rowley, Jessica A., Willis, Nicky J., Squire, Sarah E., Gill, Becky, Brough, Steve, Wilson, Francis X., Wynne, Graham M., Davies, Stephen G., Davies, Kay E., Russell, Angela J.
Published in Bioorganic & medicinal chemistry (01.09.2022)
Published in Bioorganic & medicinal chemistry (01.09.2022)
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Journal Article
Chemoenzymatic synthesis of (2S)-2-arylpropanols through a dynamic kinetic resolution of 2-arylpropanals with alcohol dehydrogenases
Galletti, Paola, Emer, Enrico, Gucciardo, Gabriele, Quintavalla, Arianna, Pori, Matteo, Giacomini, Daria
Published in Organic & biomolecular chemistry (21.09.2010)
Published in Organic & biomolecular chemistry (21.09.2010)
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Journal Article
2‑Arylbenzo[d]oxazole Phosphinate Esters as Second-Generation Modulators of Utrophin for the Treatment of Duchenne Muscular Dystrophy
Babbs, Arran, Berg, Adam, Chatzopoulou, Maria, Davies, Kay E, Davies, Stephen G, Edwards, Benjamin, Elsey, David J, Emer, Enrico, Guiraud, Simon, Harriman, Shawn, Lecci, Cristina, Moir, Lee, Peters, David, Robinson, Neil, Rowley, Jessica A, Russell, Angela J, Squire, Sarah E, Tinsley, Jonathon M, Wilson, Francis X, Wynne, Graham M
Published in Journal of medicinal chemistry (23.07.2020)
Published in Journal of medicinal chemistry (23.07.2020)
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Journal Article
Isolation, Structural Identification, Synthesis, and Pharmacological Profiling of 1,2-trans-Dihydro-1,2-diol Metabolites of the Utrophin Modulator Ezutromid
Chatzopoulou, Maria, Claridge, Tim D. W, Davies, Kay E, Davies, Stephen G, Elsey, David J, Emer, Enrico, Fletcher, Ai M, Harriman, Shawn, Robinson, Neil, Rowley, Jessica A, Russell, Angela J, Tinsley, Jonathon M, Weaver, Richard, Wilkinson, Isabel V. L, Willis, Nicky J, Wilson, Francis X, Wynne, Graham M
Published in Journal of medicinal chemistry (12.03.2020)
Published in Journal of medicinal chemistry (12.03.2020)
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Journal Article