Evolution of the Thienopyridine Class of Inhibitors of IκB Kinase-β: Part I: Hit-to-Lead Strategies
Morwick, Tina, Berry, Angela, Brickwood, Janice, Cardozo, Mario, Catron, Katrina, DeTuri, Molly, Emeigh, Jonathan, Homon, Carol, Hrapchak, Matt, Jacober, Stephen, Jakes, Scott, Kaplita, Paul, Kelly, Terence A, Ksiazek, John, Liuzzi, Michel, Magolda, Ronald, Mao, Can, Marshall, Daniel, McNeil, Daniel, Prokopowicz, Anthony, Sarko, Christopher, Scouten, Erika, Sledziona, Cynthia, Sun, Sanxing, Watrous, Jane, Wu, Jiang Ping, Cywin, Charles L
Published in Journal of medicinal chemistry (18.05.2006)
Published in Journal of medicinal chemistry (18.05.2006)
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The discovery of thienopyridine analogues as potent IκB kinase β inhibitors. Part II
Wu, Jiang-Ping, Fleck, Roman, Brickwood, Janice, Capolino, Alison, Catron, Katrina, Chen, Zhidong, Cywin, Charles, Emeigh, Jonathan, Foerst, Melissa, Ginn, John, Hrapchak, Matt, Hickey, Eugene, Hao, Ming-Hong, Kashem, Mohammed, Li, Jun, Liu, Weimin, Morwick, Tina, Nelson, Richard, Marshall, Daniel, Martin, Leslie, Nemoto, Peter, Potocki, Ian, Liuzzi, Michel, Peet, Gregory W., Scouten, Erika, Stefany, David, Turner, Michael, Weldon, Steve, Zimmitti, Clare, Spero, Denise, Kelly, Terence A.
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
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The discovery of thienopyridine analogues as potent I[kappa]B kinase beta inhibitors. Part II
Wu, Jiang-Ping, Fleck, Roman, Brickwood, Janice, Capolino, Alison, Catron, Katrina, Chen, Zhidong, Cywin, Charles, Emeigh, Jonathan, Foerst, Melissa, Ginn, John, Hrapchak, Matt, Hickey, Eugene, Hao, Ming-Hong, Kashem, Mohammed, Li, Jun, Liu, Weimin, Morwick, Tina, Nelson, Richard, Marshall, Daniel, Martin, Leslie, Nemoto, Peter, Potocki, Ian, Liuzzi, Michel, Peet, Gregory W, Scouten, Erika, Stefany, David, Turner, Michael, Weldon, Steve, Zimmitti, Clare, Spero, Denise, Kelly, Terence A
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
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Second-Generation Lymphocyte Function-Associated Antigen-1 Inhibitors: 1H-Imidazo[1,2-α]imidazol-2-one Derivatives
Wu, Jiang-Ping, Emeigh, Jonathan, Gao, Donghong A, Goldberg, Daniel R, Kuzmich, Daniel, Miao, Clara, Potocki, Ian, Qian, Kevin C, Sorcek, Ronald J, Jeanfavre, Deborah D, Kishimoto, Kei, Mainolfi, Elizabeth A, Nabozny, Gerald, Peng, Charline, Reilly, Patricia, Rothlein, Robert, Sellati, Rosemarie H, Woska, Joseph R, Chen, Shirlynn, Gunn, Jocelyn A, O'Brien, Drane, Norris, Stephen H, Kelly, Terence A
Published in Journal of medicinal chemistry (21.10.2004)
Published in Journal of medicinal chemistry (21.10.2004)
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Journal Article
Evolution of the thienopyridine class of inhibitors of IkappaB kinase-beta: part I: hit-to-lead strategies
Morwick, Tina, Berry, Angela, Brickwood, Janice, Cardozo, Mario, Catron, Katrina, DeTuri, Molly, Emeigh, Jonathan, Homon, Carol, Hrapchak, Matt, Jacober, Stephen, Jakes, Scott, Kaplita, Paul, Kelly, Terence A, Ksiazek, John, Liuzzi, Michel, Magolda, Ronald, Mao, Can, Marshall, Daniel, McNeil, Daniel, Prokopowicz, 3rd, Anthony, Sarko, Christopher, Scouten, Erika, Sledziona, Cynthia, Sun, Sanxing, Watrous, Jane, Wu, Jiang Ping, Cywin, Charles L
Published in Journal of medicinal chemistry (18.05.2006)
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Published in Journal of medicinal chemistry (18.05.2006)
Journal Article
Second-Generation Lymphocyte Function-Associated Antigen-1 Inhibitors: 1 H -Imidazo[1,2-α]imidazol-2-one Derivatives
Wu, Jiang-Ping, Emeigh, Jonathan, Gao, Donghong A., Goldberg, Daniel R., Kuzmich, Daniel, Miao, Clara, Potocki, Ian, Qian, Kevin C., Sorcek, Ronald J., Jeanfavre, Deborah D., Kishimoto, Kei, Mainolfi, Elizabeth A., Nabozny, Gerald, Peng, Charline, Reilly, Patricia, Rothlein, Robert, Sellati, Rosemarie H., Woska, Joseph R., Chen, Shirlynn, Gunn, Jocelyn A., O'Brien, Drane, Norris, Stephen H., Kelly, Terence A.
Published in Journal of medicinal chemistry (01.10.2004)
Published in Journal of medicinal chemistry (01.10.2004)
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Journal Article
The discovery of thienopyridine analogues as potent IkappaB kinase beta inhibitors. Part II
Wu, Jiang-Ping, Fleck, Roman, Brickwood, Janice, Capolino, Alison, Catron, Katrina, Chen, Zhidong, Cywin, Charles, Emeigh, Jonathan, Foerst, Melissa, Ginn, John, Hrapchak, Matt, Hickey, Eugene, Hao, Ming-Hong, Kashem, Mohammed, Li, Jun, Liu, Weimin, Morwick, Tina, Nelson, Richard, Marshall, Daniel, Martin, Leslie, Nemoto, Peter, Potocki, Ian, Liuzzi, Michel, Peet, Gregory W, Scouten, Erika, Stefany, David, Turner, Michael, Weldon, Steve, Zimmitti, Clare, Spero, Denise, Kelly, Terence A
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
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IMIDAZOIMIDAZOLES AND TRIAZOLES AS ANTI - INFLAMMATORY AGENTS
WU JIANG - PING, EMEIGH JONATHAN, KELLY TERENCE, SORCEK RONALD, LEMIEUX RENE, GOLDBERG DANIEL
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Year of Publication 31.03.2010
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IMIDAZOIMIDAZOLE UND -TRIAZOLE ALS ENTZÜNDUNGSHEMMENDE MITTEL
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Year of Publication 15.11.2008
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SUBSTITUTED 3-AMINO-THIENO[2,3-B]PYRIDINE-2-CARBOXYLIC ACID AMIDE COMPOUNDS AND PROCESSES FOR PREPARING AND THEIR USES
MARSHALL, DANIEL R, NEMOTO, PETER ALLEN, HAO, MING HONG, LIU, WEIMIN W, HICKEY, EUGENE RICHARD, MORWICK, TINA M, CHEN, ZHIDONG, CYWIN, CHARLES L, FLECK, ROMAN WOLFGANG, WU, JIANG-PING, SORCEK, RONALD J, SUN, SANXING, EMEIGH, JONATHAN
Year of Publication 11.12.2012
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Small molecules useful in the treatment of inflammatory disease
Wu, Jiang-Ping, Kelly, Terence Alfred, Lemieux, Rene M, Goldberg, Daniel R, Emeigh, Jonathan Emillian, Sorcek, Ronald John
Year of Publication 23.06.2009
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Year of Publication 23.06.2009
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Small molecules useful in the treatment of inflammatory disease
LEMIEUX RENE M, GOLDBERG DANIEL R, SORCEK RONALD JOHN, EMEIGH JONATHAN EMILLIAN, KELLY TERENCE ALFRED, WU JIANG-PING
Year of Publication 23.06.2009
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Year of Publication 23.06.2009
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Imidazoimidazoler og triazoler som anti-inflammatoriske midler
KELLY, TERENCE, ALFRED, EMEIGH, JONATHAN, EMILIAN, LEMIEUX, RENE, M, WU, JIANG-PING, SORCEK, RONALD, J, GOLDBERG, DANIEL, R
Year of Publication 23.02.2009
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Year of Publication 23.02.2009
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IMIDAZOIMIDAZOLES AND TRIAZOLES AS ANTI-INFLAMMATORY AGENTS
KELLY, TERENCE, ALFRED, EMEIGH, JONATHAN, EMILIAN, LEMIEUX, RENE, M, WU, JIANG-PING, GOLDBERG, DANIEL, R, SORCEK, RONALD, J
Year of Publication 05.11.2008
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Year of Publication 05.11.2008
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ANTI-INFLAMMATORY COMPOSITIONS COMPRISING IMIDAZOIMIDAZOLES AND TRIAZOLES
LEMIEUX RENE M, GOLDBERG DANIEL R, KELLY TERENCE ALFRED, EMEIGH JONATHAN EMILIAN, WU JIANG PING, SORCEK RONALD J
Year of Publication 23.05.2007
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Year of Publication 23.05.2007
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