Anti-emetic Action of the Brain-Penetrating New Ghrelin Agonist, HM01, Alone and in Combination With the 5-HT3 Antagonist, Palonosetron and With the NK1 Antagonist, Netupitant, Against Cisplatin- and Motion-Induced Emesis in Suncus murinus (House Musk Shrew)
Rudd, John A., Chan, Sze W., Ngan, Man P., Tu, Longlong, Lu, Zengbing, Giuliano, Claudio, Lovati, Emanuela, Pietra, Claudio
Published in Frontiers in pharmacology (06.08.2018)
Published in Frontiers in pharmacology (06.08.2018)
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Profile of Antiemetic Activity of Netupitant Alone or in Combination with Palonosetron and Dexamethasone in Ferrets and Suncus murinus (House Musk Shrew)
Rudd, John A, Ngan, Man P, Lu, Zengbing, Higgins, Guy A, Giuliano, Claudio, Lovati, Emanuela, Pietra, Claudio
Published in Frontiers in pharmacology (31.08.2016)
Published in Frontiers in pharmacology (31.08.2016)
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Corrigendum: Anti-emetic Action of the Brain-Penetrating New Ghrelin Agonist, HM01, Alone and in Combination With the 5-HT3 Antagonist, Palonosetron and With the NK1 Antagonist, Netupitant, Against Cisplatin- and Motion-Induced Emesis in Suncus murinus (House Musk Shrew)
Rudd, John A., Chan, Sze W., Ngan, Man P., Tu, Longlong, Lu, Zengbing, Giuliano, Claudio, Lovati, Emanuela, Pietra, Claudio
Published in Frontiers in pharmacology (28.09.2018)
Published in Frontiers in pharmacology (28.09.2018)
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Netupitant, a Potent and Highly Selective NK1 Receptor Antagonist, Alleviates Acetic Acid-Induced Bladder Overactivity in Anesthetized Guinea-Pigs
Palea, Stefano, Guilloteau, Véronique, Rekik, Moéz, Lovati, Emanuela, Guerard, Marc, Guardia, Maria-Alba, Lluel, Philippe, Pietra, Claudio, Yoshiyama, Mitsuharu
Published in Frontiers in pharmacology (04.08.2016)
Published in Frontiers in pharmacology (04.08.2016)
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Genetic polymorphisms of the renin-angiotensin-aldosterone system in end-stage renal disease
Lovati, Emanuela, Richard, Alain, Frey, Brigitte M., Frey, Felix J., Ferrari, Paolo
Published in Kidney international (01.07.2001)
Published in Kidney international (01.07.2001)
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The growth hormone secretagogue receptor 1a agonists, anamorelin and ipamorelin, inhibit cisplatin-induced weight loss in ferrets: Anamorelin also exhibits anti-emetic effects via a central mechanism
Lu, Zengbing, Ngan, Man P., Liu, Julia Y.H, Yang, Lingqing, Tu, Longlong, Chan, Sze Wa, Giuliano, Claudio, Lovati, Emanuela, Pietra, Claudio, Rudd, John A.
Published in Physiology & behavior (01.10.2024)
Published in Physiology & behavior (01.10.2024)
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Abstract B009: The histone deacetylase inhibitor pracinostat and its metabolite SB991 are active as single agents and in combination with 5-azacitidine in acute myeloid leukemia cells
Mensah, Afua Adjeiwaa, Spriano, Filippo, Gaudio, Eugenio, Bonifacio, Annalisa, Lovati, Emanuela, Pietra, Claudio, Bertoni, Francesco
Published in Molecular cancer therapeutics (01.12.2019)
Published in Molecular cancer therapeutics (01.12.2019)
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Comparison of TAS0953/HM06 and selpercatinib in RET fusion-driven preclinical disease models of intracranial metastases
Odintsov, Igor, Lui, Allan J.W., Ishizawa, Kota, Miyazaki, Isao, Khodos, Inna, Wakayama, Kentaro, Vojnic, Morana, Hagen, Connor J., Chang, Qing, Bonifacio, Annalisa, Giuliano, Claudio, de Stanchina, Elisa, Lovati, Emanuela, Cheng, Emily, Ladanyi, Marc, Somwar, Romel
Published in Journal of clinical oncology (01.06.2022)
Published in Journal of clinical oncology (01.06.2022)
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Abstract P233: TAS0953/HM06 is effective in preclinical models of diverse tumor types driven by RET alterations
Odintsov, Igor, Kurth, Renate I., Ishizawa, Kota, Delasos, Lukas, Lui, Allan J.W., Khodos, Inna, Hagen, Connor J., Chang, Qing, Mattar, Marissa S., Vojnic, Morana, Kunte, Siddharth, Bonifacio, Annalisa, Giuliano, Claudio, De Stanchina, Elisa, Cheng, Emily, Lovati, Emanuela, Ladanyi, Marc, Somwar, Romel
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
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The brain‐penetrating, orally bioavailable, ghrelin receptor agonist HM01 ameliorates motion‐induced emesis in Suncus murinus (house musk shrew)
Tu, Longlong, Lu, Zengbing, Ngan, Man P., Lam, Francis F.Y., Giuliano, Claudio, Lovati, Emanuela, Pietra, Claudio, Rudd, John A.
Published in British journal of pharmacology (01.04.2020)
Published in British journal of pharmacology (01.04.2020)
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Abstract 4735: The histone deacetylase inhibitor pracinostat modulates the transcriptome of diffuse large B-cell lymphoma cells and is active in combination with several targeted agents
Mensah, Afua A., Spriano, Filippo, Gaudio, Eugenio, Tarantelli, Chiara Chiara, Cascione, Luciano, Rinaldi, Andrea, Lovati, Emanuela, Zucca, Emanuele, Stathis, Anastasios, Pietra, Claudio, Bertoni, Francesco
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Abstract 799: The novel histone deacetylase inhibitor pracinostat is an effective anti-lymphoma agent
Mensah, Afua A., Spriano, Filippo, Gaudio, Eugenio, Tarantelli, Chiara, Cascione, Luciano, Aresu, Luca, Lovati, Emanuela, Zucca, Emanuele, Stathis, Anastasios, Pietra, Claudio, Bertoni, Francesco
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Abstract 4784: TAS0286/HM05, a novel highly selective RET inhibitor, prominently inhibits various RET defective tumor growth
Fujita, Hidenori, Miyazaki, Isao, Kato, Masanori, Yamada, Yukari, Ishida, Keiji, Haruma, Tomonori, Nagasaki, Haruka, Ito, Kenjiro, Hashimoto, Akihiro, Kodama, Yasuo, Funabashi, Kaoru, Lovati, Emanuela, Miyadera, Kazutaka, Matsuo, Kenichi, Iwasawa, Yoshikazu
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Abstract B157: Preclinical evaluation of the blood-brain barrier permeability and intracranial efficacy of the next-generation RET inhibitor Vepafestinib
Odintsov, Igor, Wakayama, Kentaro, Zhang, Tom, Iguchi, Satoru, Kato, Masanori, Lui, Allan JW, Khodos, Inna, Vojnic, Morana, Giuliano, Claudio, Bonifacio, Annalisa, Davare, Monika A, de Stanchina, Elisa, Lovati, Emanuela, Ladanyi, Marc, Miyazaki, Isao, Somwar, Romel
Published in Molecular cancer therapeutics (01.12.2023)
Published in Molecular cancer therapeutics (01.12.2023)
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In vitro and in vivo pharmacological characterization of Pronetupitant, a prodrug of the neurokinin 1 receptor antagonist Netupitant
Ruzza, Chiara, Rizzi, Anna, Malfacini, Davide, Molinari, Stefano, Giuliano, Claudio, Lovati, Emanuela, Pietra, Claudio, Calo’, Girolamo
Published in Peptides (New York, N.Y. : 1980) (01.07.2015)
Published in Peptides (New York, N.Y. : 1980) (01.07.2015)
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Study of the antilymphoma activity of pracinostat reveals different sensitivities of DLBCL cells to HDAC inhibitors
Mensah, Afua Adjeiwaa, Spriano, Filippo, Sartori, Giulio, Priebe, Valdemar, Cascione, Luciano, Gaudio, Eugenio, Tarantelli, Chiara, Civanelli, Elisa, Aresu, Luca, Rinaldi, Andrea, Damia, Giovanna, Lovati, Emanuela, Zucca, Emanuele, Stathis, Anastasios, Pietra, Claudio, Bertoni, Francesco
Published in Blood advances (25.05.2021)
Published in Blood advances (25.05.2021)
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Abstract 4007: Efficacy of vepafestinib in preclinical models of RET fusion-driven sarcoma models
Odintsov, Igor, Cheng, Ryan C., Lui, Allan J., Zhang, Tom, Lu, Yue C., Kurth, Renate I., Vojnic, Morana, Khodos, Inna, Chang, Qing, Chen, Kevin, Giuliano, Claudio, Bonifacio, Annalisa, Miyazaki, Isao, Stanchina, Elisa de, Lovati, Emanuela, Ladanyi, Marc, Somwar, Romel
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Journal Article
Anti-emetic Action of the Brain-Penetrating New Ghrelin Agonist, HM01, Alone and in Combination With the 5-HT 3 Antagonist, Palonosetron and With the NK 1 Antagonist, Netupitant, Against Cisplatin- and Motion-Induced Emesis in Suncus murinus (House Musk Shrew)
Rudd, John A, Chan, Sze W, Ngan, Man P, Tu, Longlong, Lu, Zengbing, Giuliano, Claudio, Lovati, Emanuela, Pietra, Claudio
Published in Frontiers in pharmacology (2018)
Get full text
Published in Frontiers in pharmacology (2018)
Journal Article
Corrigendum: Anti-emetic Action of the Brain-Penetrating New Ghrelin Agonist, HM01, Alone and in Combination With the 5-HT 3 Antagonist, Palonosetron and With the NK 1 Antagonist, Netupitant, Against Cisplatin- and Motion-Induced Emesis in Suncus murinus (House Musk Shrew)
Rudd, John A, Chan, Sze W, Ngan, Man P, Tu, Longlong, Lu, Zengbing, Giuliano, Claudio, Lovati, Emanuela, Pietra, Claudio
Published in Frontiers in pharmacology (2018)
Get full text
Published in Frontiers in pharmacology (2018)
Journal Article