Continuous Synthesis and Purification by Coupling a Multistep Flow Reaction with Centrifugal Partition Chromatography
Örkényi, Róbert, Éles, János, Faigl, Ferenc, Vincze, Péter, Prechl, Anita, Szakács, Zoltán, Kóti, János, Greiner, István
Published in Angewandte Chemie International Edition (17.07.2017)
Published in Angewandte Chemie International Edition (17.07.2017)
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Design, synthesis and biological evaluation of novel cyclic malonamide derivatives as selective RIPK1 inhibitors
Petró, József Levente, Bényei, Gyula, Bana, Péter, Linke, Nikolett, Horti, Ferenc, Szabó, Judit Eszter, Szalai, Krisztina Katalin, Hornyánszky, Gábor, Greiner, István, Éles, János
Published in Bioorganic & medicinal chemistry letters (01.03.2024)
Published in Bioorganic & medicinal chemistry letters (01.03.2024)
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One-Step, Catalyst-Free Continuous-Flow Method for the Rapid and Safe Synthesis of 1‑Substituted 1H‑Tetrazoles
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Published in Organic process research & development (20.09.2024)
Published in Organic process research & development (20.09.2024)
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Environmentally Friendly Synthesis of Indoline Derivatives using Flow‐Chemistry Techniques
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Published in European journal of organic chemistry (01.12.2017)
Published in European journal of organic chemistry (01.12.2017)
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Evolution of flow-oriented design strategies in the continuous preparation of pharmaceuticals
Fülöp, Zsolt, Szemesi, Péter, Bana, Péter, Éles, János, Greiner, István
Published in Reaction chemistry & engineering (01.09.2020)
Published in Reaction chemistry & engineering (01.09.2020)
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hERG Optimization of Benzofuro−Pyridine and Pyrazino−Indole Derivatives as MCHR1 Antagonists
Huszár, József, Bozó, Éva, Beke, Gyula, Katalin Szalai, Krisztina, Kardos, Péter, Boros, András, Greiner, István, Éles, János
Published in ChemMedChem (05.04.2022)
Published in ChemMedChem (05.04.2022)
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Multistep batch-flow hybrid synthesis of a terbinafine precursor
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Published in Journal of flow chemistry (01.03.2022)
Published in Journal of flow chemistry (01.03.2022)
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Discovery of novel steroidal histamine H-3 receptor antagonists/inverse agonists. Part 2. Versatile steroidal carboxamide derivatives
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Published in Bioorganic & medicinal chemistry letters (15.10.2019)
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
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Vascular Action as the Primary Mechanism of Cognitive Effects of Cholinergic, CNS-Acting Drugs, a Rat phMRI BOLD Study
Kocsis, Pál, Gyertyán, István, Éles, János, Laszy, Judit, Hegedüs, Nikolett, Gajári, Dávid, Deli, Levente, Pozsgay, Zsófia, Dávid, Szabolcs, Tihanyi, Károly
Published in Journal of cerebral blood flow and metabolism (01.06.2014)
Published in Journal of cerebral blood flow and metabolism (01.06.2014)
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Bradykinin B1 receptor antagonists: a patent update 2009 - 2012
Bozó, Éva, Éles, János, Keserű, György M
Published in Expert opinion on therapeutic patents (01.12.2012)
Published in Expert opinion on therapeutic patents (01.12.2012)
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Multistep Continuous-Flow Synthesis of Condensed Benzothiazoles
Lövei, Klára, Greiner, István, Éles, János, Szigetvári, Áron, Dékány, Miklós, Lévai, Sándor, Novák, Zoltán, Túrós, György István
Published in Journal of flow chemistry (01.06.2015)
Published in Journal of flow chemistry (01.06.2015)
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Synthesis of vinca alkaloids and related compounds. 100. Stereoselective oxidation reactions of compounds with the aspidospermane and quebrachamine ring system. First synthesis of some alkaloids containing the epoxy ring
Eles, J, Kalaus, G, Greiner, Kajtar-Peredy, M, Szabo, P, Keseru, GM, Szabo, L, Szantay, C
Published in Journal of organic chemistry (18.10.2002)
Published in Journal of organic chemistry (18.10.2002)
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6-Aryl-quinazolines as novel GABA(B) receptor positive allosteric modulators
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Published in Bioorganic & medicinal chemistry letters (01.07.2022)
Published in Bioorganic & medicinal chemistry letters (01.07.2022)
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Discovery of novel positive allosteric modulators of the alpha 7 nicotinic acetylcholine receptor: Scaffold hopping approach
Ledneczki, Istvan, Tapolcsanyi, Pal, Gabor, Eszter, Visegrady, Andras, Vass, Marton, Eles, Janos, Holm, Patrik, Horvath, Anita, Pocsai, Aniko, Maho, Sandor, Greiner, Istvan, Kramos, Balazs, Beni, Zoltan, Koti, Janos, Kancz, Anna E., Than, Marta, Kolok, Sandor, Laszy, Judit, Balazs, Ottilia, Bugovits, Gyula, Nagy, Jozsef, Vastag, Monika, Szajli, Agota, Bozo, Eva, Levay, Gyorgy, Lendvai, Balazs, Nemethy, Zsolt
Published in European journal of medicinal chemistry (15.03.2021)
Published in European journal of medicinal chemistry (15.03.2021)
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Journal Article
Continuous Synthesis and Purification by Coupling a Multistep Flow Reaction with Centrifugal Partition Chromatography
Örkényi, Róbert, Éles, János, Faigl, Ferenc, Vincze, Péter, Prechl, Anita, Szakács, Zoltán, Kóti, János, Greiner, István
Published in Angewandte Chemie (17.07.2017)
Published in Angewandte Chemie (17.07.2017)
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HTS-based discovery and optimization of novel positive allosteric modulators of the alpha 7 nicotinic acetylcholine receptor
Ledneczki, Istvan, Horvath, Anita, Tapolcsanyi, Pal, Eles, Janos, Molnar, Katalin Dudas, Vago, Istvan, Visegrady, Andras, Kiss, Laszlo, Szigetvari, Aron, Koti, Janos, Kramos, Balazs, Maho, Sandor, Holm, Patrik, Kolok, Sandor, Fodor, Laszlo, Than, Marta, Kostyalik, Diana, Balazs, Ottilia, Vastag, Monika, Greiner, Istvan, Levay, Gyorgy, Lendvai, Balazs, Nemethy, Zsolt
Published in European journal of medicinal chemistry (15.10.2021)
Published in European journal of medicinal chemistry (15.10.2021)
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