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Published in European journal of medicinal chemistry (15.11.2021)
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Design, synthesis, and in vitro biological evaluation of meta-sulfonamidobenzamide-based antibacterial LpxH inhibitors
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Published in European journal of medicinal chemistry (15.11.2024)
Published in European journal of medicinal chemistry (15.11.2024)
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Antibiotic class with potent in vivo activity targeting lipopolysaccharide synthesis in Gram-negative bacteria
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Published in Proceedings of the National Academy of Sciences - PNAS (09.04.2024)
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Boronic ester-linked macrocyclic lipopeptides as serine protease inhibitors targeting Escherichia coli type I signal peptidase
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Published in European journal of medicinal chemistry (05.09.2018)
Published in European journal of medicinal chemistry (05.09.2018)
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Published in European journal of organic chemistry (07.02.2019)
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Discovery of 3-Cyano-N-(3-(1-isobutyrylpiperidin-4-yl)-1-methyl-4-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-5-yObenzamide: A Potent, Selective, and Orally Bioavailable Retinoic Acid Receptor Related Orphan Receptor C2 Inverse Agonist
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Published in Journal of medicinal chemistry (13.12.2018)
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Design, synthesis and in vitro biological evaluation of oligopeptides targeting E. coli type I signal peptidase (LepB)
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Published in Journal of medicinal chemistry (27.11.2008)
Published in Journal of medicinal chemistry (27.11.2008)
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A critical survey of the structure-function of the antisense oligo/RNA heteroduplex as substrate for RNase H
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The first example of sequence-specific non-uniformly 13C5 labelled RNA: Synthesis of the 29mer HIV-1 TAR RNA with 13C Relaxation Window
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Published in Tetrahedron (01.05.1999)
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