Pilot Plant Preparation of an αvβ3 Integrin Antagonist. Part 1. Process Research and Development of a (S)-β-Amino Acid Ester Intermediate: Synthesis via a Scalable, Diastereoselective Imino-Reformatsky Reaction
Clark, Jerry D, Weisenburger, Gerald A, Anderson, D. Keith, Colson, Pierre-Jean, Edney, Albert D, Gallagher, Donald J, Kleine, H. Peter, Knable, Carl M, Lantz, Melissa K, Moore, Christine M. V, Murphy, James B, Rogers, Thomas E, Ruminski, Peter G, Shah, Ajit S, Storer, Neil, Wise, Bruce E
Published in Organic process research & development (16.01.2004)
Published in Organic process research & development (16.01.2004)
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Journal Article
Pilot-Plant Preparation of an α v β 3 Integrin Antagonist: Process Development of a Carbonyldiimidazole Peptide Coupling
Weisenburger, Gerald A., Anderson, D. Keith, Clark, Jerry D., Edney, Albert D., Karbin, Puneh S., Gallagher, Donald J., Knable, Carl M., Pietz, Mark A.
Published in Organic process research & development (16.01.2009)
Published in Organic process research & development (16.01.2009)
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Journal Article
Pilot Plant Preparation of an α v β 3 Integrin Antagonist. Part 1. Process Research and Development of a ( S )-β-Amino Acid Ester Intermediate: Synthesis via a Scalable, Diastereoselective Imino-Reformatsky Reaction
Clark, Jerry D., Weisenburger, Gerald A., Anderson, D. Keith, Colson, Pierre-Jean, Edney, Albert D., Gallagher, Donald J., Kleine, H. Peter, Knable, Carl M., Lantz, Melissa K., Moore, Christine M. V., Murphy, James B., Rogers, Thomas E., Ruminski, Peter G., Shah, Ajit S., Storer, Neil, Wise, Bruce E.
Published in Organic process research & development (01.01.2004)
Published in Organic process research & development (01.01.2004)
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Journal Article
Process for making substituted pyrazoles
ALLEN KIMBERLEY C.,ANDERSON DENNIS K.,BALDUS JOHNE.,BOEHLOW TODD,CLARK JERRY D.,DUKESHERER DANIEL R.,EDNEY ALBERT D.,FEVIG TOM,KUNDRA SASTRY,LAWSON JON P.,LAU PATRICK H.,MCDERMOTT LISA L.,MAO MICHAEL, IN,SELNESS SHAUN R
Year of Publication 28.06.2006
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Year of Publication 28.06.2006
Patent
Pilot-Plant Preparation of an αvβ3 Integrin Antagonist: Process Development of a Carbonyldiimidazole Peptide Coupling
Weisenburger, Gerald A, Anderson, D. Keith, Clark, Jerry D, Edney, Albert D, Karbin, Puneh S, Gallagher, Donald J, Knable, Carl M, Pietz, Mark A
Published in Organic process research & development (16.01.2009)
Published in Organic process research & development (16.01.2009)
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Journal Article
Process for making substituted pyrazoles
DAN R. DUKESHERER, WIN NAING, LISA L MCDERMOTT, SHEKHAR VISWANATH, JERRY D CLARK, PATRICK H LAU, JOHN E BALDUS, JODI L MOE, SHAUN R SELNESS, MICHAEL K. MAO, JOHN K WALKER, KIMBERLEY C ALLEN, ALBERT D EDNEY, DENNIS K ANDERSON, CHRISTINE B SEYMOUR, PARTHA S MUDIPALLI
Year of Publication 08.11.2007
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Year of Publication 08.11.2007
Patent
PROCESS FOR MAKING SUBSTITUTED PYRAZOLE
NAING WIN, EDNEY ALBERT D, MOE JODI L, SEYMOUR CHRISTINE B, SELNESS SHAUN D, YALAMANCHILI GOPICHAND, FEVIG TOM, VISWANATH SHEKHAR, ALLEN KIMBERLEY C, BOEHLOW TODD, DUKESHERER DANIEL R, WALKER JOHN K, CLARK JERRY D, MCDERMOTT LISA L, KUNDA SASTRY, MUDIPALLI PARTHA, SCHILKE TOBIN C, LAU PATRICK H, MAO MICHAEL K, BALDUS JOHN E, ANDERSON DENNIS K, LAWSON JON P
Year of Publication 20.09.2007
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Year of Publication 20.09.2007
Patent
Process for making substituted pyrazoles
NAING WIN, EDNEY ALBERT D, MOE JODI L, SEYMOUR CHRISTINE B, DUKESHERER DAN R, SELNESS SHAUN R, YALAMANCHILI GOPICHAND, FEVIG TOM, VISWANATH SHEKHAR, ALLEN KIMBERLEY C, BOEHLOW TODD, WALKER JOHN K, CLARK JERRY D, MCDERMOTT LISA L, KUNDA SASTRY, MUDIPALLI PARTHA, SCHILKE TOBIN C, LAU PATRICK H, MAO MICHAEL K, BALDUS JOHN E, ANDERSON DENNIS K, LAWSON JON P
Year of Publication 06.06.2006
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Year of Publication 06.06.2006
Patent
Process for making substituted pyrazoles
Allen, Kimberley C, Anderson, Dennis K, Baldus, John E, Boehlow, Todd, Clark, Jerry D, Dukesherer, Dan R, Edney, Albert D, Fevig, Tom, Kunda, Sastry, Lawson, Jon P, Lau, Patrick H, McDermott, Lisa L, Mao, Michael K, Moe, Jodi L, Mudipalli, Partha, Naing, Win, Selness, Shaun R, Seymour, Christine B, Schilke, Tobin C, Viswanath, Shekhar, Walker, John K, Yalamanchili, Gopichand
Year of Publication 06.06.2006
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Year of Publication 06.06.2006
Patent
PROCESS FOR MAKING SUBSTITUTED PYRAZOLES
BOEHLOW, TODD, NAING, WIN, FEVIG, TOM, MUDIPALLI, PARTHA, ALLEN, KIMBERLEY C, SELNESS, SHAUN, D, CLARK, JERRY, D, MAO, MICHAEL, K, LAWSON, JON, P, EDNEY, ALBERT, D, DUKESHERER, DANIEL, R, MCDERMOTT, LISA, L, BALDUS, JOHN, E, SEYMOUR, CHRISTINE, B, WALKER, JOHN, K, SCHILKE, TOBIN, C, LAU, PATRICK, H, ANDERSON, DENNIS, K, MOE, JODI, L, KUNDA, SASTRY
Year of Publication 11.01.2006
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Year of Publication 11.01.2006
Patent
PROCESS FOR MAKING SUBSTITUTED PYRAZOLES
NAING WIN, EDNEY ALBERT D, MOE JODI L, SEYMOUR CHRISTINE B, SELNESS SHAUN R, YALAMANCHILI GOPICHAND, FEVIG TOM, VISWANATH SHEKHAR, ALLEN KIMBERLEY C, BOEHLOW TODD, DUKESHERER DANIEL R, WALKER JOHN K, CLARK JERRY D, MCDERMOTT LISA L, KUNDA SASTRY, MUDIPALLI PARTHA, SCHILKE TOBIN C, LAU PATRICK H, MAO MICHAEL K, BALDUS JOHN E, ANDERSON DENNIS K, LAWSON JON P
Year of Publication 09.11.2005
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Year of Publication 09.11.2005
Patent
Process for making substituted pyrazoles
WIN NAING, SHEKHAR VISWANATH, ALLEN, KIMBERLY, K, CLARK, JERRY, D, MAO, MICHAEL, K, DUKESHERER, DAN, R, EDNEY, ALBERT, D, MCDERMOTT, LISA, L, BALDUS, JOHN, E, MUDIPALLI, PARTHAN, S, SEYMOUR, CHRISTINE, B, WALKER, JOHN, K, SCHILKE, TOBIN, C, GOPI YALAMANCHILI, LAU, PATRICK, H, ANDERSON, DENNIS, K, MOE, JODI, L, SELNESS, SHAUN, R
Year of Publication 27.05.2005
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Year of Publication 27.05.2005
Patent
Process for making substituted pyrazoles
GOPICHAND YALAMANCHILI, DAN R. DUKESHERER, WIN NAING, SHEKHAR VISWANATH, DENNIS K. ANDERSON, MOE, CZARNIK, JODI, PATRICK H. LAU, TOBIN C. SCHILKE, JOHN K. WALKER, JERRY D. CLARK, CHRISTINE B. SEYMOUR, MICHAEL K. MAO, ALBERT D. EDNEY, PARTHA S. MUDIPALLI, KIMBERLEY C. ALLEN, LISA L. MCDERMOTT, SHAUN R. SELNESS, JOHN E. BALDUS
Year of Publication 29.04.2005
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Year of Publication 29.04.2005
Patent
PROCESS FOR MAKING SUBSTITUTED PYRAZOLES
NAING WIN, EDNEY ALBERT D, MOE JODI L, SEYMOUR CHRISTINE B, DUKESHERER DAN R, SELNESS SHAUN R, YALAMANCHILI GOPICHAND, VISWANATH SHEKHAR, ALLEN KIMBERLEY C, WALKER JOHN K, CLARK JERRY D, MCDERMOTT LISA L, MUDIPALLI PARTHA S, SCHILKE TOBIN C, LAU PATRICK H, MAO MICHAEL K, BALDUS JOHN E, ANDERSON DENNIS K
Year of Publication 18.04.2005
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Year of Publication 18.04.2005
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PROCESS FOR MAKING SUBSTITUTED PYRAZOLES
BOEHLOW, TODD, NAING, WIN, FEVIG, TOM, MUDIPALLI, PARTHA, CLARK, JERRY, D, MAO, MICHAEL, K, LAWSON, JON, P, VISWANATH, SHEKHAR, YALAMANCHILI, GOPICHAND, EDNEY, ALBERT, D, DUKESHERER, DANIEL, R, MCDERMOTT, LISA, L, ALLEN, KIMBERLEY, C, BALDUS, JOHN, E, SEYMOUR, CHRISTINE, B, WALKER, JOHN, K, SCHILKE, TOBIN, C, LAU, PATRICK, H, ANDERSON, DENNIS, K, MOE, JODI, L, KUNDA, SASTRY, SELNESS, SHAUN, R
Year of Publication 24.03.2005
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Year of Publication 24.03.2005
Patent
PROCESS FOR MAKING SUBSTITUTED PYRAZOLES
BOEHLOW, TODD, NAING, WIN, FEVIG, TOM, MUDIPALLI, PARTHA, CLARK, JERRY, D, MAO, MICHAEL, K, LAWSON, JON, P, VISWANATH, SHEKHAR, YALAMANCHILI, GOPICHAND, EDNEY, ALBERT, D, DUKESHERER, DANIEL, R, MCDERMOTT, LISA, L, ALLEN, KIMBERLEY, C, BALDUS, JOHN, E, SEYMOUR, CHRISTINE, B, WALKER, JOHN, K, SCHILKE, TOBIN, C, LAU, PATRICK, H, ANDERSON, DENNIS, K, MOE, JODI, L, KUNDA, SASTRY, SELNESS, SHAUN, R
Year of Publication 14.10.2004
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Year of Publication 14.10.2004
Patent
PROCESS FOR MAKING SUBSTITUTED PYRAZOLES
SELNESS, SHAUN R, BOEHLOW, TODD, NAING, WIN, FEVIG, TOM, LAWSON, JON P, DUKESHERER, DANIEL R, MUDIPALLI, PARTHA, ALLEN, KIMBERLEY C, VISWANATH, SHEKHAR, YALAMANCHILI, GOPICHAND, EDNEY, ALBERT D, MCDERMOTT, LISA L, BALDUS, JOHN E, SCHILKE, TOBIN C, SEYMOUR, CHRISTINE B, CLARK, JERRY D, LAU, PATRICK H, MOE, JODI L, WALKER, JOHN K, KUNDA, SASTRY, ANDERSON, DENNIS K, MAO, MICHAEL K
Year of Publication 14.10.2004
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Year of Publication 14.10.2004
Patent
Process for making substituted pyrazoles
JODI L. MOE, GOPICHAND YALAMANCHILI, WIN NAING, TODD BOEHLOW, SHEKHAR VISWANATH, DENNIS K. ANDERSON, JON P. LAWSON, PATRICK H. LAU, TOBIN C. SCHILKE, JOHN K. WALKER, TOM FEVIG, PARTHA MUDIPALLI, JERRY D. CLARK, CHRISTINE B. SEYMOUR, MICHAEL K. MAO, SASTRY KUNDA, ALBERT D. EDNEY, LISA L. MCDERMOTT, KIMBERLEY C. ALLEN, SHAUN R. SELNESS, DANIEL R. DUKESHERER, JOHN E. BALDUS
Year of Publication 14.10.2004
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Year of Publication 14.10.2004
Patent
PROCESS FOR MAKING SUBSTITUTED PYRAZOLES
NAING, WIN, CLARK, JERRY, D, MAO, MICHAEL, K, VISWANATH, SHEKHAR, MUDIPALLI, PARTHA, S, EDNEY, ALBERT, D, DUKESHERER, DAN, R, MCDERMOTT, LISA, L, ALLEN, KIMBERLEY, C, BALDUS, JOHN, E, SEYMOUR, CHRISTINE, B, WALKER, JOHN, K, LAU, PATRICK, H, YALAMANCHILI, GOPI, ANDERSON, DENNIS, K, MOE, JODI, L, SELNESS, SHAUN, R
Year of Publication 23.06.2004
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Year of Publication 23.06.2004
Patent
Process for making substituted pyrazoles
NAING WIN, KUNDRA SASTRY, EDNEY ALBERT D, MOE JODI L, SEYMOUR CHRISTINE B, SELNESS SHAUN R, YALAMANCHILI GOPICHAND, FEVIG TOM, VISWANATH SHEKHAR, ALLEN KIMBERLEY C, BOEHLOW TODD, DUKESHERER DANIEL R, WALKER JOHN K, CLARK JERRY D, MCDERMOTT LISA L, MUDIPALLI PARTHA, SCHILKE TOBIN C, LAU PATRICK H, MAO MICHAEL K, BALDUS JOHN E, ANDERSON DENNIS K, LAWSON JON P
Year of Publication 04.12.2003
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Year of Publication 04.12.2003
Patent