Ligand Binding Mechanism in Steroid Receptors: From Conserved Plasticity to Differential Evolutionary Constraints
Edman, Karl, Hosseini, Ali, Bjursell, Magnus K., Aagaard, Anna, Wissler, Lisa, Gunnarsson, Anders, Kaminski, Tim, Köhler, Christian, Bäckström, Stefan, Jensen, Tina J., Cavallin, Anders, Karlsson, Ulla, Nilsson, Ewa, Lecina, Daniel, Takahashi, Ryoji, Grebner, Christoph, Geschwindner, Stefan, Lepistö, Matti, Hogner, Anders C., Guallar, Victor
Published in Structure (London) (01.12.2015)
Published in Structure (London) (01.12.2015)
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Preclinical pharmacology of AZD9977: A novel mineralocorticoid receptor modulator separating organ protection from effects on electrolyte excretion
Bamberg, Krister, Johansson, Ulrika, Edman, Karl, William-Olsson, Lena, Myhre, Susanna, Gunnarsson, Anders, Geschwindner, Stefan, Aagaard, Anna, Björnson Granqvist, Anna, Jaisser, Frédéric, Huang, Yufeng, Granberg, Kenneth L, Jansson-Löfmark, Rasmus, Hartleib-Geschwindner, Judith
Published in PloS one (23.02.2018)
Published in PloS one (23.02.2018)
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AZD9567 versus prednisolone in patients with active rheumatoid arthritis: A phase IIa, randomized, double‐blind, efficacy, and safety study
Laar, Jacob M., Lei, Alejhandra, Safy‐Khan, Mary, Almquist, Joachim, Belfield, Graham, Edman, Karl, Öberg, Lisa, Angermann, Bastian R., Dillmann, Inken, Berntsson, Pia, Etal, Damla, Dainty, Ian, Astbury, Carol, Belvisi, Maria G., Nemes, Szilárd, Platt, Adam, Prothon, Susanne, Samuelsson, Sara, Svanberg, Petter, Keen, Christina, Jacobs, J. W. G., Kaan, Ellen, Tubergen, Astrid, Hermans, Kasper, Vonkeman, Harald, Moghadam, Marjan Ghiti, Gjertsson, Inger, Ekwall, Anna‐Karin, Kapetanovic, Meliha, Einarsson, Jon Thorkell, Axelsson, Lena T., Olsson, Richard, Myrbäck, Tove Hegelund, Taib, Ziad, Vikman, Kerstin
Published in Clinical and translational science (01.12.2023)
Published in Clinical and translational science (01.12.2023)
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Bacteriorhodopsin: a high-resolution structural view of vectorial proton transport
Neutze, Richard, Pebay-Peyroula, Eva, Edman, Karl, Royant, Antoine, Navarro, Javier, Landau, Ehud M.
Published in BBA - Biomembranes (11.10.2002)
Published in BBA - Biomembranes (11.10.2002)
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Helix deformation is coupled to vectorial proton transport in the photocycle of bacteriorhodopsin
Pebay-Peyroula, Eva, Neutze, Richard, Edman, Karl, Landau, Ehud M, Royant, Antoine, Ursby, Thomas
Published in Nature (London) (10.08.2000)
Published in Nature (London) (10.08.2000)
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High-resolution X-ray structure of an early intermediate in the bacteriorhodopsin photocycle
Landau, Ehud M, Edman, Karl, Nollert, Peter, Royant, Antoine, Belrhali, Hassan, Pebay-Peyroula, Eva, Hajdu, Janos, Neutze, Richard
Published in Nature (London) (21.10.1999)
Published in Nature (London) (21.10.1999)
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Deformation of Helix C in the Low Temperature L-intermediate of Bacteriorhodopsin
Edman, Karl, Royant, Antoine, Larsson, Gisela, Jacobson, Frida, Taylor, Tom, van der Spoel, David, Landau, Ehud M., Pebay-Peyroula, Eva, Neutze, Richard
Published in The Journal of biological chemistry (16.01.2004)
Published in The Journal of biological chemistry (16.01.2004)
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Early Structural Rearrangements in the Photocycle of an Integral Membrane Sensory Receptor
Edman, Karl, Royant, Antoine, Nollert, Peter, Maxwell, Carrie A, Pebay-Peyroula, Eva, Navarro, Javier, Neutze, Richard, Landau, Ehud M
Published in Structure (London) (01.04.2002)
Published in Structure (London) (01.04.2002)
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Structural insight into allosteric modulation of protease-activated receptor 2
Cheng, Robert K Y, Fiez-Vandal, Cédric, Schlenker, Oliver, Edman, Karl, Aggeler, Birte, Brown, Dean G, Brown, Giles A, Cooke, Robert M, Dumelin, Christoph E, Doré, Andrew S, Geschwindner, Stefan, Grebner, Christoph, Hermansson, Nils-Olov, Jazayeri, Ali, Johansson, Patrik, Leong, Louis, Prihandoko, Rudi, Rappas, Mathieu, Soutter, Holly, Snijder, Arjan, Sundström, Linda, Tehan, Benjamin, Thornton, Peter, Troast, Dawn, Wiggin, Giselle, Zhukov, Andrei, Marshall, Fiona H, Dekker, Niek
Published in Nature (London) (04.05.2017)
Published in Nature (London) (04.05.2017)
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Unraveling the Allosteric Cross-Talk between the Coactivator Peptide and the Ligand-Binding Site in the Glucocorticoid Receptor
La Sala, Giuseppina, Gunnarsson, Anders, Edman, Karl, Tyrchan, Christian, Hogner, Anders, Frolov, Andrey I
Published in Journal of chemical information and modeling (26.07.2021)
Published in Journal of chemical information and modeling (26.07.2021)
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Exploring Binding Mechanisms in Nuclear Hormone Receptors by Monte Carlo and X-ray-derived Motions
Grebner, Christoph, Lecina, Daniel, Gil, Victor, Ulander, Johan, Hansson, Pia, Dellsen, Anita, Tyrchan, Christian, Edman, Karl, Hogner, Anders, Guallar, Victor
Published in Biophysical journal (28.03.2017)
Published in Biophysical journal (28.03.2017)
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Quaternary glucocorticoid receptor structure highlights allosteric interdomain communication
Postel, Sandra, Wissler, Lisa, Johansson, Carina A, Gunnarsson, Anders, Gordon, Euan, Collins, Barry, Castaldo, Marie, Köhler, Christian, Öling, David, Johansson, Patrik, Fröderberg Roth, Linda, Beinsteiner, Brice, Dainty, Ian, Delaney, Stephen, Klaholz, Bruno P, Billas, Isabelle M L, Edman, Karl
Published in Nature structural & molecular biology (01.03.2023)
Published in Nature structural & molecular biology (01.03.2023)
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Glucocorticoid receptor Thr524 phosphorylation by MINK1 induces interactions with 14-3-3 protein regulators
Munier, Claire C., De Maria, Leonardo, Edman, Karl, Gunnarsson, Anders, Longo, Marianna, MacKintosh, Carol, Patel, Saleha, Snijder, Arjan, Wissler, Lisa, Brunsveld, Luc, Ottmann, Christian, Perry, Matthew W.D.
Published in The Journal of biological chemistry (01.01.2021)
Published in The Journal of biological chemistry (01.01.2021)
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Designing Selective Drug-like Molecular Glues for the Glucocorticoid Receptor/14-3‑3 Protein–Protein Interaction
Pallesen, Jakob S., Munier, Claire C., Bosica, Francesco, Andrei, Sebastian A., Edman, Karl, Gunnarsson, Anders, La Sala, Giuseppina, Putra, Okky Dwichandra, Srdanović, Sonja, Wilson, Andrew J., Wissler, Lisa, Ottmann, Christian, Perry, Matthew W. D., O’Mahony, Gavin
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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The effect of AZD9567 vs. prednisolone on glycaemic control in patients with type 2 diabetes mellitus: Results from a phase 2a clinical trial
Ambery, Philip, Zajac, Grzegorz, Almquist, Joachim, Prothon, Susanne, Astbury, Carol, Brown, Mary N., Nemes, Szilard, Nsabimana, Joselyne, Edman, Karl, Öberg, Lisa, Lepistö, Matti, Edenro, Goran, Dillmann, Inken, Mitra, Suman, Belfield, Graham, Keen, Christina, Heise, Tim
Published in British journal of clinical pharmacology (01.08.2024)
Published in British journal of clinical pharmacology (01.08.2024)
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Correction to “Designing Selective Drug-like Molecular Glues for the Glucocorticoid Receptor/14-3‑3 Protein–Protein Interaction”
Pallesen, Jakob S., Munier, Claire C., Bosica, Francesco, Andrei, Sebastian A., Edman, Karl, Gunnarsson, Anders, La Sala, Giuseppina, Putra, Okky Dwichandra, Srdanović, Sonja, Wilson, Andrew J., Wissler, Lisa, Ottmann, Christian, Perry, Matthew W. D., O’Mahony, Gavin
Published in Journal of medicinal chemistry (09.02.2023)
Published in Journal of medicinal chemistry (09.02.2023)
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