The first highly potent and selective non-peptide neuropeptide Y Y1 receptor antagonist : BIBP3226
RUDOLF, K, EBERLEIN, W, ENGEL, W, WIELAND, H. A, WILLIM, K. D, ENTZEROTH, M, WIENEN, W, BECK-SICKINGER, A. G, DOODS, H. N
Published in European journal of pharmacology (27.12.1994)
Published in European journal of pharmacology (27.12.1994)
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BIBP 3226, the first selective neuropeptide Y1 receptor antagonist: A review of its pharmacological properties
Doods, Henri N., Wieland, Heike A., Engel, Wolfhard, Eberlein, Wolfgang, Willim, Klaus-Dieter, Entzeroth, Michael, Wienen, Wolfgang, Rudolf, Klaus
Published in Regulatory peptides (27.08.1996)
Published in Regulatory peptides (27.08.1996)
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Specific bradycardic agents. 1. Chemistry, pharmacology, and structure-activity relationships of substituted benzazepinones, a new class of compounds exerting antiischemic properties
Reiffen, Manfred, Eberlein, Wolfgang, Mueller, Peter, Psiorz, Manfred, Noll, Klaus, Heider, Joachim, Lillie, Christian, Kobinger, Walter, Luger, Peter
Published in Journal of medicinal chemistry (01.05.1990)
Published in Journal of medicinal chemistry (01.05.1990)
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Development of Human Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonists. 1. Potent and Selective Small Molecule CGRP Antagonists. 1-[N 2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1- piperidinyl]carbonyl]-d-tyrosyl]-l-lysyl]-4-(4-pyridinyl)piperazine: The First CGRP Antagonist for Clinical Trials in Acute Migraine
Rudolf, Klaus, Eberlein, Wolfgang, Engel, Wolfhard, Pieper, Helmut, Entzeroth, Michael, Hallermayer, Gerhard, Doods, Henri
Published in Journal of medicinal chemistry (22.09.2005)
Published in Journal of medicinal chemistry (22.09.2005)
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Tricyclic compounds as selective muscarinic receptor antagonists. 3. Structure-selectivity relationships in a series of cardioselective (M2) antimuscarinics
Engel, Wolfhard W, Eberlein, Wolfgang G, Mihm, Gerhard, Hammer, Rudolf, Trummlitz, Guenter
Published in Journal of medicinal chemistry (01.08.1989)
Published in Journal of medicinal chemistry (01.08.1989)
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BIIE0246: A selective and high affinity neuropeptide Y Y2 receptor antagonist
Doods, Henri, Gaida, Wolfram, Wieland, Heike A, Dollinger, Horst, Schnorrenberg, Gerd, Esser, Franz, Engel, Wolfhard, Eberlein, Wolfgang, Rudolf, Klaus
Published in European journal of pharmacology (19.11.1999)
Published in European journal of pharmacology (19.11.1999)
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Tricyclic compounds as selective antimuscarinics. 2. Structure-activity relationships of M1-selective antimuscarinics related to pirenzepine
Eberlein, Wolfgang G, Engel, Wolfhard W, Trummlitz, Guenter, Schmidt, Guenther, Hammer, Rudolf
Published in Journal of medicinal chemistry (01.06.1988)
Published in Journal of medicinal chemistry (01.06.1988)
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METHOD FOR PRODUCING A PRODUCT FROM ROLLED STRIP MATERIAL
BRECHT JOERG DIETER, MUHR THOMAS, SCHNEIDER CHRISTOPH, BUTZKAMM JUERGEN, STEFFENS HUBERTUS JOSEF, HAHN CHRISTOPH, EBERLEIN WOLFGANG
Year of Publication 24.02.2016
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Year of Publication 24.02.2016
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Tricyclic compounds as selective antimuscarinics. 1. Structural requirements for selectivity towards the muscarinic acetylcholine receptor in a series of pirenzepine and imipramine analogs
Eberlein, Wolfgang G, Trummlitz, Guenter, Engel, Wolfhard W, Schmidt, Guenther, Pelzer, Helmut, Mayer, Norbert
Published in Journal of medicinal chemistry (01.08.1987)
Published in Journal of medicinal chemistry (01.08.1987)
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Characterisation of calcitonin gene-related peptide receptors in rat atrium and vas deferens: evidence for a [Cys(Et) 2,7]hCGRP-preferring receptor
Wu, Dongmei, Eberlein, Wolfgang, Rudolf, Klaus, Engel, Wolfhard, Hallermayer, Gerhard, Doods, Henri
Published in European journal of pharmacology (21.07.2000)
Published in European journal of pharmacology (21.07.2000)
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