Orally Active MMP-1 Sparing α-Tetrahydropyranyl and α-Piperidinyl Sulfone Matrix Metalloproteinase (MMP) Inhibitors with Efficacy in Cancer, Arthritis, and Cardiovascular Disease
Becker, Daniel P, Barta, Thomas E, Bedell, Louis J, Boehm, Terri L, Bond, Brian R, Carroll, Jeffery, Carron, Chris P, DeCrescenzo, Gary A, Easton, Alan M, Freskos, John N, Funckes-Shippy, Chris L, Heron, Marcia, Hockerman, Susan, Howard, Carol Pearcy, Kiefer, James R, Li, Madeleine H, Mathis, Karl J, McDonald, Joseph J, Mehta, Pramod P, Munie, Grace E, Sunyer, Teresa, Swearingen, Craig A, Villamil, Clara I, Welsch, Dean, Williams, Jennifer M, Yu, Ying, Yao, Jun
Published in Journal of medicinal chemistry (23.09.2010)
Published in Journal of medicinal chemistry (23.09.2010)
Get full text
Journal Article
MMP-13 selective α-sulfone hydroxamates: A survey of P1′ heterocyclic amide isosteres
Barta, Thomas E., Becker, Daniel P., Bedell, Louis J., Easton, Alan M., Hockerman, Susan L., Kiefer, James, Munie, Grace E., Mathis, Karl J., Li, Madeleine H., Rico, Joseph G., Villamil, Clara I., Williams, Jennifer M.
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Get full text
Journal Article
Saturation Mutagenesis of Human Interleukin-3 (∗)
Olins, Peter O., Bauer, S. Christopher, Braford-Goldberg, Sarah, Sterbenz, Kris, Polazzi, Joseph O., Caparon, Maire H., Klein, Barbara K., Easton, Alan M., Paik, Kumnan, Klover, Jon A., Thiele, Barrett R., McKearn, John P.
Published in The Journal of biological chemistry (06.10.1995)
Published in The Journal of biological chemistry (06.10.1995)
Get full text
Journal Article
Use of combinatorial mutagenesis to select for multiply substituted human interleukin-3 variants with improved pharmacologic properties
Klein, Barbara K., Olins, Peter O., Bauer, S.Christopher, Caparon, Maire H., Easton, Alan M., Braford, Sarah R., Abrams, Mark A., Klover, Jon A., Paik, Kumnan, Thomas, John W., Hood, William F., Shieh, Jeng-Jong, Polazzi, Joseph O., Donnelly, Ann M., Zeng, David L., Welply, Joseph K., McKearn, John P.
Published in Experimental hematology (01.12.1999)
Published in Experimental hematology (01.12.1999)
Get full text
Journal Article
Production of bovine insulin-like growth factor 2 (bIGF2) in Escherichia coli
Easton, Alan M., Gierse, James K., Seetharam, Ramnath, Klein, Barbara K., Kotts, Claire E.
Published in Gene (30.05.1991)
Published in Gene (30.05.1991)
Get full text
Journal Article
11 alpha hydroxylase and oxidoreductase
Bolten, Suzanne L, Clayton, Robert A, Easton, Alan M, Engel, Leslie C, Messing, Dean M, Ng, John S, Reitz, Beverly, Walker, Mark C, Wang, Ping T
Year of Publication 03.07.2007
Get full text
Year of Publication 03.07.2007
Patent
Aspergillus ochraceus 11 alpha hydroxylase and oxidoreductase
ENGEL LESLIE C, CLAYTON ROBERT A, BOLTEN SUZANNE L, WANG PING T, EASTON ALAN M, NG JOHN S, REITZ BEVERLY, MESSING DEAN M, WALKER MARK C
Year of Publication 03.07.2007
Get full text
Year of Publication 03.07.2007
Patent
Aspergillus ochraceus 11 alpha hydroxylase and oxidoreductase
Bolten, Suzanne L, Clayton, Robert A, Easton, Alan M, Engel, Leslie C, Messing, Dean M, Ng, John S, Reitz, Beverly, Walker, Mark C, Wang, Ping T
Year of Publication 25.04.2006
Get full text
Year of Publication 25.04.2006
Patent
Aspergillus ochraceus 11 alpha hydroxylase and oxidoreductase
ENGEL LESLIE C, CLAYTON ROBERT A, BOLTEN SUZANNE L, WANG PING T, EASTON ALAN M, NG JOHN S, REITZ BEVERLY, MESSING DEAN M, WALKER MARK C
Year of Publication 25.04.2006
Get full text
Year of Publication 25.04.2006
Patent
Aspergillus ochraceus 11 alpha hydroxylase and oxidoreductase
ENGEL LESLIE C, CLAYTON ROBERT A, BOLTEN SUZANNE L, WANG PING T, EASTON ALAN M, NG JOHN S, REITZ BEVERLY, MESSING DEAN M, WALKER MARK C
Year of Publication 06.01.2005
Get full text
Year of Publication 06.01.2005
Patent
Interleukin-3 (IL-3) multiple mutation polypeptides
KLEIN BARBARA K, MCKEARN JOHN P, BRAFORD-GOLDBERG SARAH R, ABRAMS MARK A, EASTON ALAN M, PAIK KUMNAN, BAUER S. C, OLINS PETER, THOMAS JOHN W, CAPARON MAIRE H
Year of Publication 03.11.2005
Get full text
Year of Publication 03.11.2005
Patent
Aspergillus ochraceus 11 alpha hydroxylase and oxidoreductase
ENGEL LESLIE C, CLAYTON ROBERT A, WANG PING T, EASTON ALAN M, NG JOHN S, REITZ BEVERLY, SUZANNE BOLTEN L, MESSING DEAN M, WALKER MARK C
Year of Publication 07.08.2003
Get full text
Year of Publication 07.08.2003
Patent
Therapeutic methods using interleukin-3 (IL-3) human/murine hybrid polypeptides
EASTON; ALAN M, KLEIN; BARBARA K, BRAFORD-GOLDBERG; SARAH R, MCKEARN; JOHN P, OLINS; PETER O
Year of Publication 06.08.1996
Get full text
Year of Publication 06.08.1996
Patent