Solvent-Controlled, Site-Selective N‑Alkylation Reactions of Azolo-Fused Ring Heterocycles at N1‑, N2‑, and N3-Positions, Including Pyrazolo[3,4‑d]pyrimidines, Purines, [1,2,3]Triazolo[4,5]pyridines, and Related Deaza-Compounds
Bookser, Brett C, Weinhouse, Michael I, Burns, Aaron C, Valiere, Andrew N, Valdez, Lino J, Stanczak, Pawel, Na, Jim, Rheingold, Arnold L, Moore, Curtis E, Dyck, Brian
Published in Journal of organic chemistry (15.06.2018)
Published in Journal of organic chemistry (15.06.2018)
Get full text
Journal Article
Phosphodiesterase 1b (PDE1B) Regulates Spatial and Contextual Memory in Hippocampus
McQuown, Susan, Xia, Shouzhen, Baumgärtel, Karsten, Barido, Richard, Anderson, Gary, Dyck, Brian, Scott, Roderick, Peters, Marco
Published in Frontiers in molecular neuroscience (07.02.2019)
Published in Frontiers in molecular neuroscience (07.02.2019)
Get full text
Journal Article
Total Asymmetric Synthesis of the Putative Structure of the Cytotoxic Diterpenoid (−)-Sclerophytin A and of the Authentic Natural Sclerophytins A and B
Bernardelli, Patrick, Moradei, Oscar M, Friedrich, Dirk, Yang, Jiong, Gallou, Fabrice, Dyck, Brian P, Doskotch, Raymond W, Lange, Tim, Paquette, Leo A
Published in Journal of the American Chemical Society (19.09.2001)
Published in Journal of the American Chemical Society (19.09.2001)
Get full text
Journal Article
Studies on the structure–activity relationship of bicifadine analogs as monoamine transporter inhibitors
Zhang, Mingzhu, Jovic, Florence, Vickers, Troy, Dyck, Brian, Tamiya, Junko, Grey, Jonathan, Tran, Joe A., Fleck, Beth A., Pick, Rebecca, Foster, Alan C., Chen, Chen
Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
Get full text
Journal Article
Identification of 1S,2R-milnacipran analogs as potent norepinephrine and serotonin transporter inhibitors
TAMIYA, Junko, DYCK, Brian, FOSTER, Alan C, CHEN CHEN, MINGZHU ZHANG, PHAN, Kasey, FLECK, Beth A, APARICIO, Anna, JOVIC, Florence, TRAN, Joe A, VICKERS, Troy, GREY, Jonathan
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
Get full text
Journal Article
Studies on the SAR and pharmacophore of milnacipran derivatives as monoamine transporter inhibitors
Chen, Chen, Dyck, Brian, Fleck, Beth A., Foster, Alan C., Grey, Jonathan, Jovic, Florence, Mesleh, Michael, Phan, Kasey, Tamiya, Junko, Vickers, Troy, Zhang, Mingzhu
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
Get full text
Journal Article
Studies on a series of milnacipran analogs containing a heteroaromatic group as potent norepinephrine and serotonin transporter inhibitors
Vickers, Troy, Dyck, Brian, Tamiya, Junko, Zhang, Mingzhu, Jovic, Florence, Grey, Jonathan, Fleck, Beth A., Aparicio, Anna, Johns, Michael, Jin, Liping, Tang, Hui, Foster, Alan C., Chen, Chen
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
Get full text
Journal Article
Potent and orally active non-peptide antagonists of the human melanocortin-4 receptor based on a series of trans-2-disubstituted cyclohexylpiperazines
Tucci, Fabio C., White, Nicole S., Markison, Stacy, Joppa, Margaret, Tran, Joe A., Fleck, Beth A., Madan, Ajay, Dyck, Brian P., Parker, Jessica, Pontillo, Joseph, Melissa Arellano, L., Marinkovic, Dragan, Jiang, Wanlong, Chen, Caroline W., Gogas, Kathleen R., Goodfellow, Val S., Saunders, John, Foster, Alan C., Chen, Chen
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Get full text
Journal Article
Potent, Orally Active Corticotropin-Releasing Factor Receptor-1 Antagonists Containing a Tricyclic Pyrrolopyridine or Pyrazolopyridine Core
Dyck, Brian, Grigoriadis, Dimitri E, Gross, Raymond S, Guo, Zhiqiang, Haddach, Mustapha, Marinkovic, Dragan, McCarthy, James R, Moorjani, Manisha, Regan, Collin F, Saunders, John, Schwaebe, Michael K, Szabo, Tomas, Williams, John P, Zhang, Xiaohu, Bozigian, Haig, Chen, Ta Kung
Published in Journal of medicinal chemistry (16.06.2005)
Published in Journal of medicinal chemistry (16.06.2005)
Get full text
Journal Article
Potent imidazole and triazole CB 1 receptor antagonists related to SR141716
Dyck, Brian, Goodfellow, Val S., Phillips, Teresa, Grey, Jonathan, Haddach, Mustapha, Rowbottom, Martin, Naeve, Gregory S., Brown, Brock, Saunders, John
Published in Bioorganic & medicinal chemistry letters (01.03.2004)
Published in Bioorganic & medicinal chemistry letters (01.03.2004)
Get full text
Journal Article
PDE1 억제제로서의 치환된 푸라노피리미딘 화합물
CHUNG DEMICHAEL, BURNS AARON, TRAN JOE, DYCK BRIAN, KLEINKE ANDREW, RAFFAELE NICHOLAS, WEINHOUSE MICHAEL, KUMAR DANGE VIJAY, BOOKSER BRETT, BOTROUS IRINY, MCCARRICK MARGARET
Year of Publication 18.09.2020
Get full text
Year of Publication 18.09.2020
Patent