Discovery of 1‑Butyl-3-chloro-4-(4-phenyl-1-piperidinyl)-(1H)‑pyridone (JNJ-40411813): A Novel Positive Allosteric Modulator of the Metabotropic Glutamate 2 Receptor
Cid, José María, Tresadern, Gary, Duvey, Guillaume, Lütjens, Robert, Finn, Terry, Rocher, Jean-Philippe, Poli, Sonia, Vega, Juan Antonio, de Lucas, Ana Isabel, Matesanz, Encarnación, Linares, María Lourdes, Andrés, José Ignacio, Alcazar, Jesús, Alonso, José Manuel, Macdonald, Gregor J, Oehlrich, Daniel, Lavreysen, Hilde, Ahnaou, Abdelah, Drinkenburg, Wilhelmus, Mackie, Claire, Pype, Stefan, Gallacher, David, Trabanco, Andrés A
Published in Journal of medicinal chemistry (14.08.2014)
Published in Journal of medicinal chemistry (14.08.2014)
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MGLU7 수용체의 음성 다른 자리 입체성 조절제로서의 축합된 헤테로사이클 유도체
PAPARIN JEAN LAURENT, DUVEY GUILLAUME, ROCHER JEAN PHILIPPE, FINN TERRY
Year of Publication 23.02.2024
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Year of Publication 23.02.2024
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An mGlu4‐Positive Allosteric Modulator Alleviates Parkinsonism in Primates
Charvin, Delphine, Di Paolo, Therese, Bezard, Erwan, Gregoire, Laurent, Takano, Akihiro, Duvey, Guillaume, Pioli, Elsa, Halldin, Christer, Medori, Rossella, Conquet, François
Published in Movement disorders (01.10.2018)
Published in Movement disorders (01.10.2018)
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MGLU7 수용체의 음성 다른 자리 입체성 조절제로서의 치환된 헤테로이환식 유도체
PAPARIN JEAN LAURENT, STACH TANJA, DUVEY GUILLAUME, TANG LAM, MAEDER PATRICK, ROCHER JEAN PHILIPPE
Year of Publication 20.02.2024
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Year of Publication 20.02.2024
Patent
Discovery of 1-Buty1-3-chloro-4-(4-pheny1-1-piperidiny1)(1H)-pyridone (JNJ-40411813): A Novel Positive Allosteric Modulator of the Metabotropic Glutamate 2 Receptor
Maria Cid, Jose, Tresadern, Gary, Duvey, Guillaume, Lutjens, Robert, Finn, Terry, Rocher, Jean-Philippe, Poli, Sonia, Antonio Vega, Juan, Isabel de Lucas, Ana, Matesanz, Encarnacion, Lourdes Linares, Maria, Ignacio Andres, Jose, Alcazar, Jesus, Manuel Alonso, Jose, Macdonald, Gregor J., Oehlrich, Daniel, Lavreysen, Hilde, Ahnaou, Abdelah, Drinkenburg, Wilhelmus, Mackie, Claire, Pype, Stefan, Gallacher, David, Trabanco, Andres A.
Published in Journal of medicinal chemistry (14.08.2014)
Published in Journal of medicinal chemistry (14.08.2014)
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An m G lu4‐ P ositive A llosteric M odulator A lleviates P arkinsonism in P rimates
Charvin, Delphine, Di Paolo, Therese, Bezard, Erwan, Gregoire, Laurent, Takano, Akihiro, Duvey, Guillaume, Pioli, Elsa, Halldin, Christer, Medori, Rossella, Conquet, François
Published in Movement disorders (01.10.2018)
Published in Movement disorders (01.10.2018)
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Characterization of [11C]PXT012253 as a PET Radioligand for mGlu4 Allosteric Modulators in Nonhuman Primates
Takano, Akihiro, Nag, Sangram, Jia, Zhisheng, Jahan, Mahabuba, Forsberg, Anton, Arakawa, Ryosuke, Grybäck, Per, Duvey, Guillaume, Halldin, Christer, Charvin, Delphine
Published in Molecular imaging and biology (17.06.2019)
Published in Molecular imaging and biology (17.06.2019)
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Characterization of [ 11 C]PXT012253 as a PET Radioligand for mGlu 4 Allosteric Modulators in Nonhuman Primates
Takano, Akihiro, Nag, Sangram, Jia, Zhisheng, Jahan, Mahabuba, Forsberg, Anton, Arakawa, Ryosuke, Grybäck, Per, Duvey, Guillaume, Halldin, Christer, Charvin, Delphine
Published in Molecular imaging and biology (01.06.2019)
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Published in Molecular imaging and biology (01.06.2019)
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Discovery of 1,4-Disubstituted 3-Cyano-2-pyridones: A New Class of Positive Allosteric Modulators of the Metabotropic Glutamate 2 Receptor
Cid, Jose María, Duvey, Guillaume, Tresadern, Gary, Nhem, Vanthea, Furnari, Rocco, Cluzeau, Philippe, Vega, Juan Antonio, de Lucas, Ana Isabel, Matesanz, Encarnación, Alonso, José Manuel, Linares, María Lourdes, Andrés, José Ignacio, Poli, Sonia M, Lutjens, Robert, Himogai, Hassan, Rocher, Jean-Philippe, Macdonald, Gregor J, Oehlrich, Daniel, Lavreysen, Hilde, Ahnaou, Abdelah, Drinkenburg, Wilhelmus, Mackie, Claire, Trabanco, Andrés A
Published in Journal of medicinal chemistry (08.03.2012)
Published in Journal of medicinal chemistry (08.03.2012)
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A novel series of metabotropic glutamate receptor 5 negative allosteric modulators based on a 4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine core
Duvey, Guillaume, Perry, Benjamin, Le Poul, Emmanuel, Poli, Sonia, Bonnet, Beatrice, Lambeng, Nathalie, Charvin, Delphine, Donovan-Rodrigues, Tansy, Haddouk, Hasnaà, Gagliardi, Stefania, Rocher, Jean-Philippe
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
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Synthesis of 3-Fluoroazetidines
Van Brabandt, Willem, Verniest, Guido, De Smaele, Dirk, Duvey, Guillaume, De Kimpe, Norbert
Published in Journal of organic chemistry (01.09.2006)
Published in Journal of organic chemistry (01.09.2006)
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New positive allosteric modulators of the metabotropic glutamate receptor 2 (mGluR2): Identification and synthesis of N-propyl-8-chloro-6-substituted isoquinolones
Trabanco, Andrés A., Duvey, Guillaume, Cid, José María, Macdonald, Gregor J., Cluzeau, Philippe, Nhem, Vanthea, Furnari, Rocco, Behaj, Nadia, Poulain, Géraldine, Finn, Terry, Lavreysen, Hilde, Poli, Sonia, Raux, Alexandre, Thollon, Yves, Poirier, Nicolas, D’Addona, David, Andrés, José Ignacio, Lutjens, Robert, Poul, Emmanuel Le, Imogai, Hassan, Rocher, Jean-Philippe
Published in Bioorganic & medicinal chemistry letters (01.02.2011)
Published in Bioorganic & medicinal chemistry letters (01.02.2011)
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FUSED HETEROCYCLIC DERIVATIVES AS NEGATIVE ALLOSTERIC MODULATORS OF MGLU7 RECEPTOR
Finn, Terry, Paparin, Jean-Laurent, Duvey, Guillaume, Rocher, Jean-Philippe
Year of Publication 08.08.2024
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Year of Publication 08.08.2024
Patent
Discovery of 1,5-Disubstituted Pyridones: A New Class of Positive Allosteric Modulators of the Metabotropic Glutamate 2 Receptor
Cid, Jose María, Duvey, Guillaume, Cluzeau, Philippe, Nhem, Vanthea, Macary, Karim, Raux, Alexandre, Poirier, Nicolas, Muller, Jessica, Boléa, Christelle, Finn, Terry, Poli, Sonia, Epping-Jordan, Mark, Chamelot, Emilie, Derouet, Francis, Girard, Francoise, Macdonald, Gregor J, Vega, Juan Antonio, de Lucas, Ana Isabel, Matesanz, Encarnación, Lavreysen, Hilde, Linares, María Lourdes, Oehlrich, Daniel, Oyarzábal, Julen, Tresadern, Gary, Trabanco, Andrés A, Andrés, Jose Ignacio, Le Poul, Emmanuel, Imogai, Hassan, Lutjens, Robert, Rocher, Jean-Philippe
Published in ACS chemical neuroscience (15.12.2010)
Published in ACS chemical neuroscience (15.12.2010)
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