Adherence to assigned dosing regimen and sustained virological response among chronic hepatitis C genotype 1 patients treated with boceprevir plus peginterferon alfa‐2b/ribavirin
Gordon, S. C., Yoshida, E. M., Lawitz, E. J., Bacon, B. R., Sulkowski, M. S., Davis, M., Poordad, F., Bronowicki, J.‐P., Esteban, R., Sniukiene, V., Burroughs, M. H., Deng, W., Dutko, F. J., Brass, C. A., Albrecht, J. K., Rajender Reddy, K.
Published in Alimentary Pharmacology & Therapeutics (Suppl) (01.07.2013)
Published in Alimentary Pharmacology & Therapeutics (Suppl) (01.07.2013)
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Safety and efficacy of the fixed-dose combination regimen of MK-3682/grazoprevir/ruzasvir in cirrhotic or non-cirrhotic patients with chronic HCV GT1 infection who previously failed a direct-acting antiviral regimen (C-SURGE)
Wedemeyer, H, Wyles, D, Reddy, R, Luetkemeyer, A, Jacobson, I, Vierling, J.M, Gordon, S, Nahass, R, Zeuzem, S, Wahl, J, Barr, E, Nguyen, B.-Y.T, Robertson, M, Joeng, H.-K, Liu, H, Jumes, P, Dutko, F, Martin, E
Published in Journal of hepatology (2017)
Published in Journal of hepatology (2017)
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Efficacy and safety of the fixed-dose combination regimen of MK3 [MK-3682/grazoprevir/ruzasvir] with or without ribavirin in non-cirrhotic or cirrhotic patients with chronic HCV GT1, 2, 3, 4 or 6 infection (Parts A & B of C-CREST-1 & 2)
Lawitz, E, Yoshida, E.M, Buti, M, Vierling, J.M, Almasio, P.L, Bruno, S, Ruane, P.J, Hassanein, T.I, Mullhaupt, B, Pearlman, B, Jancoriene, L, Gao, W, Huang, H.-C, Shepherd, A, Tannenbaum, B, Fernsler, D, Li, J.J, Grandhi, A, Liu, H, Su, M, Dutko, F, Yeh, W.W, Plank, R, Nguyen, B.-Y.T, Wahl, J, Barr, E, Butterton, J.R
Published in Journal of hepatology (2017)
Published in Journal of hepatology (2017)
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High sustained virologic response rates in patients with chronic hepatitis C virus GT1, 2 or 3 infection following 16 weeks of MK-3682/grazoprevir/ruzasvir plus ribavirin after having failed 8 weeks of a triplet drug regimen (Part C of C-CREST-1 & 2)
Serfaty, L, Pianko, S, Ari, Z.B, Laursen, A.L, Hansen, J, Gane, E.J, Huang, H.-C, Jin, S, Bourque, J, Liu, H, Grandhi, A, Su, M, Gendrano, N, Fernsler, D, Dutko, F, Nguyen, B.-Y.T, Wahl, J, Barr, E, Yeh, W, Plank, R, Butterton, J.R
Published in Journal of hepatology (2017)
Published in Journal of hepatology (2017)
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High Efficacy of an 8-Week 3-Drug Regimen of Grazoprevir/MK-8408/MK-3682 in HCV Genotype 1, 2 and 3-Infected Patients: SVR24 Data from the Phase 2 C-Crest 1 and 2 Studies
Gane, E.J, Pianko, S, Roberts, S.K, Thompson, A.J, Zeuzem, S, Zuckerman, E, Ari, Z.B, Foster, G.R, Agarwal, K, Laursen, A.L, Gerstoft, J, Gao, W, Huang, H.-C, Fitzgerald, B, Li, J.J, Wan, S, Dutko, F, Nguyen, B.-Y.T, Wahl, J, Barr, E, Butterton, J.R, Esteban, R
Published in Journal of hepatology (2016)
Published in Journal of hepatology (2016)
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Conformational change in the floor of the human rhinovirus canyon blocks adsorption to HeLa cell receptors
PEVEAR, D. C, FANCHER, M. J, FELOCK, P. J, ROSSMANN, M. G, MILLER, M. S, DIANA, G, TREASURYWALA, A. M, MCKINLAY, M. A, DUTKO, F. J
Published in Journal of Virology (01.05.1989)
Published in Journal of Virology (01.05.1989)
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Picornavirus Inhibitors: Trifluoromethyl Substitution Provides a Global Protective Effect against Hepatic Metabolism
Diana, Guy D, Rudewicz, Patrick, Pevear, Daniel C, Nitz, Theodore J, Aldous, Suzanne C, Aldous, David J, Robinson, David T, Draper, Tandy, Dutko, Frank J
Published in Journal of medicinal chemistry (01.04.1995)
Published in Journal of medicinal chemistry (01.04.1995)
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Crystal structure of human rhinovirus serotype 1A (HRV1A)
Kim, Sangsoo, Smith, Thomas J., Chapman, Michael S., Rossmann, Michael G., Pevear, Daniel C., Dutko, Frank J., Felock, Peter J., Diana, Guy D., McKinlay, Mark A.
Published in Journal of molecular biology (05.11.1989)
Published in Journal of molecular biology (05.11.1989)
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Efficacy and safety of 12 weeks versus 18 weeks of treatment with grazoprevir (MK-5172) and elbasvir (MK-8742) with or without ribavirin for hepatitis C virus genotype 1 infection in previously untreated patients with cirrhosis and patients with previous null response with or without cirrhosis (C-WORTHY): a randomised, open-label phase 2 trial
Lawitz, Eric, Prof, Gane, Edward, Prof, Pearlman, Brian, Prof, Tam, Edward, MD, Ghesquiere, Wayne, Prof, Guyader, Dominique, Prof, Alric, Laurent, MD, Bronowicki, Jean-Pierre, Prof, Lester, Laura, MSN, Sievert, William, Prof, Ghalib, Reem, MD, Balart, Luis, MD, Sund, Fredrik, MD, Lagging, Martin, Prof, Dutko, Frank, PhD, Shaughnessy, Melissa, MS, Hwang, Peggy, PhD, Howe, Anita Y M, PhD, Wahl, Janice, MD, Robertson, Michael, MD, Barr, Eliav, MD, Haber, Barbara, MD
Published in The Lancet (British edition) (21.03.2015)
Published in The Lancet (British edition) (21.03.2015)
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Genetic and molecular analyses of spontaneous mutants of human rhinovirus 14 that are resistant to an antiviral compound
HEINZ, B. A, RUECKERT, R. R, SHEPARD, D. A, DUTKO, F. J, MCKINLAY, M. A, FANCHER, M, ROSSMANN, M. G, BADGER, J, SMITH, T. J
Published in Journal of Virology (01.06.1989)
Published in Journal of Virology (01.06.1989)
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Oxadiazoles as Ester Bioisosteric Replacements in Compounds Related to Disoxaril. Antirhinovirus Activity
Diana, Guy D, Volkots, Deborah L, Nitz, Theodore J, Bailey, Thomas R, Long, Melody A, Vescio, Niranjan, Aldous, Suzanne, Pevear, Daniel C, Dutko, Frank J
Published in Journal of medicinal chemistry (01.07.1994)
Published in Journal of medicinal chemistry (01.07.1994)
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Efficacy of oral WIN 54954 for prophylaxis of experimental rhinovirus infection
Turner, R B, Dutko, F J, Goldstein, N H, Lockwood, G, Hayden, F G
Published in Antimicrobial Agents and Chemotherapy (01.02.1993)
Published in Antimicrobial Agents and Chemotherapy (01.02.1993)
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Structural Analysis of a Series of Antiviral Agents Complexed with Human Rhinovirus 14
Badger, John, Minor, Iwona, Kremer, Marcia J., Oliveira, Marcos A., Smith, Thomas J., Griffith, James P., Diego M. A. Guerin, Krishnaswamy, S., Luo, Ming, Rossmann, Michael G., McKinlay, Mark A., Diana, Guy D., Dutko, Frank J., Fancher, Marilyn, Rueckert, Roland R., Heinz, Beverly A.
Published in Proceedings of the National Academy of Sciences - PNAS (01.05.1988)
Published in Proceedings of the National Academy of Sciences - PNAS (01.05.1988)
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In vitro and in vivo activities of WIN 54954, a new broad-spectrum antipicornavirus drug
WOODS, M. G, DIANA, G. D, ROGGE, M. C, OTTO, M. J, DUTKO, F. J, MCKINLAY, M. A
Published in Antimicrobial Agents and Chemotherapy (01.12.1989)
Published in Antimicrobial Agents and Chemotherapy (01.12.1989)
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The structure of human rhinovirus 16
Oliveira, Marcos A, Zhao, Rui, Lee, Wai-Ming, Kremer, Marcia J, Minor, Iwona, Rueckert, Roland R, Diana, Guy D, Pevear, Daniel C, Dutko, Frank J, McKinlay, Mark A, Rossmann, Michael G
Published in Structure (London) (15.09.1993)
Published in Structure (London) (15.09.1993)
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Efficacy and safety of 8 weeks of elbasvir/grazoprevir in HCV GT4-infected treatment-naīve participants
Asselah, T., Pol, S., Hezode, C., Loustaud-Ratti, V., Leroy, V., Ahmed, S.N.S., Ozenne, V., Bronowicki, J.-P., Larrey, D., Tran, A., Alric, L., Nguyen-Khac, E., Robertson, M., Hanna, G., Brown, D., Asante-Appiah, E., Ludmerer, S., Su, M., Hwang, P., Klopfer, S., Dutko, F., Guidoum, A., Hagen, K., Haber, B., Talwani, R., Serfaty, L.
Published in Journal of hepatology (01.04.2018)
Published in Journal of hepatology (01.04.2018)
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