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Published in ACS medicinal chemistry letters (14.11.2019)
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Lead Optimization of Thiazolo[5,4-c]piperidines: 3-Cyclobutoxy Linker as a Key Spacer for H3R Inverse Agonists
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Published in ChemMedChem (01.12.2012)
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Phenyl‐oxazoles, a New Family of Inverse Agonists at the H 3 Histamine Receptor
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Published in ChemMedChem (06.07.2009)
Published in ChemMedChem (06.07.2009)
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COMPOUNDS COMPRISING A CYCLOBUTOXY GROUP
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Year of Publication 18.11.2010
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Year of Publication 18.11.2010
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First dual M sub(3) antagonists-PDE4 inhibitors: Synthesis and SAR of 4,6- diaminopyrimidine derivatives
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Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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First dual M3 antagonists-PDE4 inhibitors : Synthesis and SAR of 4,6-diaminopyrimidine derivatives
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Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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Lead Optimization of Thiazolo[5,4‐ c ]piperidines: 3‐Cyclobutoxy Linker as a Key Spacer for H 3 R Inverse Agonists
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Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Phenyl-oxazoles, a New Family of Inverse Agonists at the H3 Histamine Receptor
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Published in ChemMedChem (01.02.2010)
Published in ChemMedChem (01.02.2010)
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First dual M 3 antagonists-PDE4 inhibitors: Synthesis and SAR of 4,6-diaminopyrimidine derivatives
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Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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COMPOUNDS COMPRISING A CYCLOBUTOXY GROUP
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Year of Publication 22.12.2011
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Year of Publication 22.12.2011
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Acetamide Scanning around Bicyclic Thiazoles: SAR at the H3 Receptor
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Published in ChemMedChem (05.09.2011)
Published in ChemMedChem (05.09.2011)
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Fused tricyclic benzimidazoles derivatives as modulators of TNF activity
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Year of Publication 03.04.2018
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Year of Publication 03.04.2018
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Compounds Comprising A Cyclobutoxy Group
CELANIRE SYLVAIN, DENONNE FREDERIC, DEFAYS SABINE, DURIEU VERONIQUE, VALADE ANNE
Year of Publication 18.11.2010
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Year of Publication 18.11.2010
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COMPOUNDS COMPRISING A CYCLOBUTOXY GROUP
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Year of Publication 13.10.2010
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Year of Publication 13.10.2010
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Compounds comprising a cyclobutoxy group
SYLVAIN CELANIRE, ANNE VALADE, FREDERIC DENONNE, SABINE DEFAYS, VERONIQUE DURIEU
Year of Publication 30.07.2009
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Year of Publication 30.07.2009
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Fused Tricyclic Benzimidazoles Derivatives As Modulators of TNF Activity
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Year of Publication 20.10.2016
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Year of Publication 20.10.2016
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Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists
Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van Houtvin, Nathalie
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Journal Article
Discovery of a New Class of Non-imidazole Oxazoline-Based Histamine H3 Receptor (H3R) Inverse Agonists
Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean-Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent
Published in ChemMedChem (06.07.2009)
Published in ChemMedChem (06.07.2009)
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