Human Protein Tyrosine Phosphatase 1B (PTP1B): From Structure to Clinical Inhibitor Perspectives
Liu, Rongxing, Mathieu, Cécile, Berthelet, Jérémy, Zhang, Wenchao, Dupret, Jean-Marie, Rodrigues Lima, Fernando
Published in International journal of molecular sciences (24.06.2022)
Published in International journal of molecular sciences (24.06.2022)
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Structural characterization of a pathogenic mutant of human protein tyrosine phosphatase PTPN2 (Cys216Gly) that causes very early onset autoimmune enteropathy
Nian, Qing, Berthelet, Jérémy, Parlato, Marianna, Mechaly, Ariel E., Liu, Rongxing, Dupret, Jean‐Marie, Cerf‐Bensussan, Nadine, Haouz, Ahmed, Rodrigues Lima, Fernando
Published in Protein science (01.02.2022)
Published in Protein science (01.02.2022)
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Biochemical, Enzymatic, and Computational Characterization of Recurrent Somatic Mutations of the Human Protein Tyrosine Phosphatase PTP1B in Primary Mediastinal B Cell Lymphoma
Liu, Rongxing, Sun, Yujie, Berthelet, Jérémy, Bui, Linh-Chi, Xu, Ximing, Viguier, Mireille, Dupret, Jean-Marie, Deshayes, Frédérique, Rodrigues Lima, Fernando
Published in International journal of molecular sciences (24.06.2022)
Published in International journal of molecular sciences (24.06.2022)
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From arylamine N-acetyltransferase to folate-dependent acetyl CoA hydrolase: impact of folic acid on the activity of (HUMAN)NAT1 and its homologue (MOUSE)NAT2
Laurieri, Nicola, Dairou, Julien, Egleton, James E, Stanley, Lesley A, Russell, Angela J, Dupret, Jean-Marie, Sim, Edith, Rodrigues-Lima, Fernando
Published in PloS one (13.05.2014)
Published in PloS one (13.05.2014)
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Cisplatin causes covalent inhibition of protein-tyrosine phosphatase 1B (PTP1B) through reaction with its active site cysteine: Molecular, cellular and in vivo mice studies
Liu, Rongxing, Zhang, Wenchao, Gou, Panhong, Berthelet, Jérémy, Nian, Qing, Chevreux, Guillaume, Legros, Véronique, Moroy, Gautier, Bui, Linh-Chi, Wang, Li, Dupret, Jean-Marie, Deshayes, Frédérique, Rodrigues Lima, Fernando
Published in Biomedicine & pharmacotherapy (01.09.2022)
Published in Biomedicine & pharmacotherapy (01.09.2022)
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Xenobiotic‐metabolizing enzymes in Bacillus anthracis: molecular and functional analysis of a truncated arylamine N‐acetyltransferase isozyme
Kubiak, Xavier, Duval, Romain, Pluvinage, Benjamin, Chaffotte, Alain F, Dupret, Jean‐Marie, Rodrigues‐Lima, Fernando
Published in British journal of pharmacology (01.07.2017)
Published in British journal of pharmacology (01.07.2017)
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A readout of metabolic efficiency in arylamine N‐acetyltransferase‐deficient mice reveals minor energy metabolism changes
Denis, Raphaël G.P., Busi, Florent, Castel, Julien, Morel, Chloé, Zhang, Wenchao, Bui, Linh‐Chi, Sugamori, Kim S., Prokopec, Stephenie D., Boutros, Paul C., Grant, Denis M., Rodrigues‐Lima, Fernando, Luquet, Serge, Dupret, Jean‐Marie
Published in FEBS letters (01.04.2019)
Published in FEBS letters (01.04.2019)
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Carbon Black Nanoparticles Selectively Alter Follicle-Stimulating Hormone Expression in vitro and in vivo in Female Mice
Avet, Charlotte, Paul, Emmanuel N, Garrel, Ghislaine, Grange-Messent, Valérie, L'Hôte, David, Denoyelle, Chantal, Corre, Raphaël, Dupret, Jean-Marie, Lanone, Sophie, Boczkowski, Jorge, Simon, Violaine, Cohen-Tannoudji, Joëlle
Published in Frontiers in neuroscience (06.12.2021)
Published in Frontiers in neuroscience (06.12.2021)
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Biotransformation of Trichoderma spp. and Their Tolerance to Aromatic Amines, a Major Class of Pollutants
Cocaign, Angélique, Bui, Linh-Chi, Silar, Philippe, Chan Ho Tong, Laetitia, Busi, Florent, Lamouri, Aazdine, Mougin, Christian, Rodrigues-Lima, Fernando, Dupret, Jean-Marie, Dairou, Julien
Published in Applied and Environmental Microbiology (01.08.2013)
Published in Applied and Environmental Microbiology (01.08.2013)
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The Structure and the Regulation of Glycogen Phosphorylases in Brain
Mathieu, Cécile, Dupret, Jean-Marie, Rodrigues-Lima, Fernando
Published in Advances in neurobiology (01.01.2019)
Published in Advances in neurobiology (01.01.2019)
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An acetyltransferase assay for CREB-binding protein based on reverse phase–ultra-fast liquid chromatography of fluorescent histone H3 peptides
Duval, Romain, Fritsch, Lauriane, Bui, Linh-Chi, Berthelet, Jérémy, Guidez, Fabien, Mathieu, Cécile, Dupret, Jean-Marie, Chomienne, Christine, Ait-Si-Ali, Slimane, Rodrigues-Lima, Fernando
Published in Analytical biochemistry (01.10.2015)
Published in Analytical biochemistry (01.10.2015)
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Structural and Biochemical Characterization of an Active Arylamine N-Acetyltransferase Possessing a Non-canonical Cys-His-Glu Catalytic Triad
Kubiak, Xavier, Li de la Sierra-Gallay, Inès, Chaffotte, Alain F., Pluvinage, Benjamin, Weber, Patrick, Haouz, Ahmed, Dupret, Jean-Marie, Rodrigues-Lima, Fernando
Published in The Journal of biological chemistry (02.08.2013)
Published in The Journal of biological chemistry (02.08.2013)
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Insight into cofactor recognition in arylamine N-acetyltransferase enzymes: structure of Mesorhizobium loti arylamine N-acetyltransferase in complex with coenzyme A
Xu, Ximing, Li de la Sierra-Gallay, Inés, Kubiak, Xavier, Duval, Romain, Chaffotte, Alain F., Dupret, Jean-Marie, Haouz, Ahmed, Rodrigues-Lima, Fernando
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2015)
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2015)
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Identification of the Xenobiotic-Metabolizing Enzyme Arylamine N-Acetyltransferase 1 as a New Target of Cisplatin in Breast Cancer Cells: Molecular and Cellular Mechanisms of Inhibition
Ragunathan, Nilusha, Dairou, Julien, Pluvinage, Benjamin, Martins, Marta, Petit, Emile, Janel, Nathalie, Dupret, Jean-Marie, Rodrigues-Lima, Fernando
Published in Molecular pharmacology (01.06.2008)
Published in Molecular pharmacology (01.06.2008)
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A novel color change mechanism for breast cancer biomarker detection: naphthoquinones as specific ligands of human arylamine N-acetyltransferase 1
Laurieri, Nicola, Egleton, James E, Varney, Amy, Thinnes, Cyrille C, Quevedo, Camilo E, Seden, Peter T, Thompson, Sam, Rodrigues-Lima, Fernando, Dairou, Julien, Dupret, Jean-Marie, Russell, Angela J, Sim, Edith
Published in PloS one (05.08.2013)
Published in PloS one (05.08.2013)
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Mechanisms and kinetics of human arylamine N-acetyltransferase 1 inhibition by disulfiram
Malka, Florence, Dairou, Julien, Ragunathan, Nilusha, Dupret, Jean-Marie, Rodrigues-Lima, Fernando
Published in The FEBS journal (01.09.2009)
Published in The FEBS journal (01.09.2009)
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Structural and functional characterization of an arylamine N-acetyltransferase from the pathogen Mycobacterium abscessus: differences from other mycobacterial isoforms and implications for selective inhibition
Cocaign, Angélique, Kubiak, Xavier, Xu, Ximing, Garnier, Guillaume, Li de la Sierra-Gallay, Inès, Chi-Bui, Linh, Dairou, Julien, Busi, Florent, Abuhammad, Areej, Haouz, Ahmed, Dupret, Jean-Marie, Herrmann, Jean-Louis, Rodrigues-Lima, Fernando
Published in Acta crystallographica. Section D, Biological crystallography. (01.11.2014)
Published in Acta crystallographica. Section D, Biological crystallography. (01.11.2014)
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