An inhibitor of NADPH oxidase-4 attenuates established pulmonary fibrosis in a rodent disease model
Jarman, Elizabeth R, Khambata, Valerie S, Cope, Claire, Jones, Peter, Roger, Jan, Ye, Li Yun, Duggan, Nicholas, Head, Denise, Pearce, Andrew, Press, Neil J, Bellenie, Ben, Sohal, Bindi, Jarai, Gabor
Published in American journal of respiratory cell and molecular biology (01.01.2014)
Published in American journal of respiratory cell and molecular biology (01.01.2014)
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Imatinib Attenuates Hypoxia-induced Pulmonary Arterial Hypertension Pathology via Reduction in 5-Hydroxytryptamine through Inhibition of Tryptophan Hydroxylase 1 Expression
CIUCLAN, Loredana, HUSSEY, Martin J, KONSTANTINOVA, Irena, PEARCE, Andrew, ROWLANDS, David J, JARAI, Gabor, WESTWICK, John, MACLEAN, Margaret R, THOMAS, Matthew, BURTON, Victoria, GOOD, Robert, DUGGAN, Nicholas, BEACH, Sarah, JONES, Peter, FOX, Roy, CLAY, Leuan, BONNEAU, Olivier
Published in American journal of respiratory and critical care medicine (2013)
Published in American journal of respiratory and critical care medicine (2013)
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The Development of Oculomotor Suppression of Salient Distractors in Children
Blakley, Emily C., Duggan, Nicholas, Gaspelin, Nicholas, Gerhardstein, Peter
Published in Journal of vision (Charlottesville, Va.) (27.09.2021)
Published in Journal of vision (Charlottesville, Va.) (27.09.2021)
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A Novel Murine Model of Severe Pulmonary Arterial Hypertension
CIUCLAN, Loredana, BONNEAU, Olivier, WALKER, Christoph, WESTWICK, John, THOMAS, Matthew, HUSSEY, Martin, DUGGAN, Nicholas, HOLMES, Alan M, GOOD, Robert, STRINGER, Rowan, JONES, Peter, MORRELL, Nicholas W, JARAI, Gabor
Published in American journal of respiratory and critical care medicine (15.11.2011)
Published in American journal of respiratory and critical care medicine (15.11.2011)
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Treatment with Anti–Gremlin 1 Antibody Ameliorates Chronic Hypoxia/SU5416–Induced Pulmonary Arterial Hypertension in Mice
Ciuclan, Loredana, Sheppard, KellyAnn, Dong, Liqun, Sutton, Daniel, Duggan, Nicholas, Hussey, Martin, Simmons, Jenny, Morrell, Nicholas W, Jarai, Gabor, Edwards, Matthew, DuBois, Gerald, Thomas, Matthew, Van Heeke, Gino, England, Karen
Published in The American journal of pathology (01.11.2013)
Published in The American journal of pathology (01.11.2013)
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Novel ROCK inhibitors for the treatment of pulmonary arterial hypertension
Shaw, Duncan, Hollingworth, Greg, Soldermann, Nicolas, Sprague, Elizabeth, Schuler, Walter, Vangrevelinghe, Eric, Duggan, Nicholas, Thomas, Matthew, Kosaka, Takatoshi, Waters, Nigel, van Eis, Maurice J.
Published in Bioorganic & medicinal chemistry letters (15.10.2014)
Published in Bioorganic & medicinal chemistry letters (15.10.2014)
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Activin-Like Kinase 5 (ALK5) Mediates Abnormal Proliferation of Vascular Smooth Muscle Cells from Patients with Familial Pulmonary Arterial Hypertension and Is Involved in the Progression of Experimental Pulmonary Arterial Hypertension Induced by Monocrotaline
Thomas, Matthew, Docx, Cerys, Holmes, Alan M, Beach, Sarah, Duggan, Nicholas, England, Karen, Leblanc, Catherine, Lebret, Clemence, Schindler, Francis, Raza, Farheen, Walker, Christoph, Crosby, Alexi, Davies, Rachel J, Morrell, Nicholas W, Budd, David C
Published in The American journal of pathology (01.02.2009)
Published in The American journal of pathology (01.02.2009)
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Journal Article
Discovery of Fevipiprant (NVP-QAW039), a Potent and Selective DP2 Receptor Antagonist for Treatment of Asthma
Sandham, David A, Barker, Lucy, Brown, Lyndon, Brown, Zarin, Budd, David, Charlton, Steven J, Chatterjee, Devnandan, Cox, Brian, Dubois, Gerald, Duggan, Nicholas, Hall, Edward, Hatto, Julia, Maas, Janet, Manini, Jodie, Profit, Rachael, Riddy, Darren, Ritchie, Catherine, Sohal, Bindi, Shaw, Duncan, Stringer, Rowan, Sykes, David A, Thomas, Matthew, Turner, Katharine L, Watson, Simon J, West, Ryan, Willard, Elisabeth, Williams, Gareth, Willis, Jennifer
Published in ACS medicinal chemistry letters (11.05.2017)
Published in ACS medicinal chemistry letters (11.05.2017)
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Discovery and characterization of NVP-QAV680, a potent and selective CRTh2 receptor antagonist suitable for clinical testing in allergic diseases
Sandham, David A., Arnold, Nicola, Aschauer, Heinrich, Bala, Kamlesh, Barker, Lucy, Brown, Lyndon, Brown, Zarin, Budd, David, Cox, Brian, Docx, Cerys, Dubois, Gerald, Duggan, Nicholas, England, Karen, Everatt, Brian, Furegati, Marcus, Hall, Edward, Kalthoff, Frank, King, Anna, Leblanc, Catherine J., Manini, Jodie, Meingassner, Josef, Profit, Rachael, Schmidt, Alfred, Simmons, Jennifer, Sohal, Bindi, Stringer, Rowan, Thomas, Matthew, Turner, Katharine L., Walker, Christoph, Watson, Simon J., Westwick, John, Willis, Jennifer, Williams, Gareth, Wilson, Caroline
Published in Bioorganic & medicinal chemistry (01.11.2013)
Published in Bioorganic & medicinal chemistry (01.11.2013)
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Essential role of phosphoinositide 3-kinase gamma in eosinophil chemotaxis within acute pulmonary inflammation
Thomas, Matthew, Edwards, Matthew J, Sawicka, Elzbieta, Duggan, Nicholas, Hirsch, Emilio, Wymann, Matthias P, Owen, Charles, Trifilieff, Alexandre, Walker, Christoph, Westwick, John, Finan, Peter
Published in Immunology (01.03.2009)
Published in Immunology (01.03.2009)
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A translational preclinical model of interstitial pulmonary fibrosis and pulmonary hypertension: mechanistic pathways driving disease pathophysiology
Jarman, Elizabeth R., Khambata, Valerie S., Li, Yun Ye, Cheung, Kenneth, Thomas, Matthew, Duggan, Nicholas, Jarai, Gabor
Published in Physiological reports (01.09.2014)
Published in Physiological reports (01.09.2014)
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Journal Article
Correction to "Discovery of Fevipiprant (NVP-QAW039), a Potent and Selective DP 2 Receptor Antagonist for Treatment of Asthma"
Sandham, David A, Barker, Lucy, Brown, Lyndon, Brown, Zarin, Budd, David, Charlton, Steven J, Chatterjee, Devnandan, Cox, Brian, Dubois, Gerald, Duggan, Nicholas, Hall, Edward, Hatto, Julia, Leblanc, Catherine, Maas, Janet, Manini, Jodie, Profit, Rachael, Riddy, Darren, Ritchie, Catherine, Sohal, Bindi, Shaw, Duncan, Stringer, Rowan, Sykes, David A, Thomas, Matthew, Turner, Katharine L, Watson, Simon J, West, Ryan, Willard, Elisabeth, Williams, Gareth, Willis, Jennifer
Published in ACS medicinal chemistry letters (14.09.2017)
Published in ACS medicinal chemistry letters (14.09.2017)
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Journal Article
Correction to “Discovery of Fevipiprant (NVP-QAW039), a Potent and Selective DP2 Receptor Antagonist for Treatment of Asthma”
Sandham, David A, Barker, Lucy, Brown, Lyndon, Brown, Zarin, Budd, David, Charlton, Steven J, Chatterjee, Devnandan, Cox, Brian, Dubois, Gerald, Duggan, Nicholas, Hall, Edward, Hatto, Julia, Maas, Janet, Manini, Jodie, Profit, Rachael, Riddy, Darren, Ritchie, Catherine, Sohal, Bindi, Shaw, Duncan, Stringer, Rowan, Sykes, David A, Thomas, Matthew, Turner, Katharine L, Watson, Simon J, West, Ryan, Willard, Elisabeth, Williams, Gareth, Willis, Jennifer
Published in ACS medicinal chemistry letters (14.09.2017)
Published in ACS medicinal chemistry letters (14.09.2017)
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Journal Article
Discovery of Fevipiprant (NVP-QAW039), a Potent and Selective DP 2 Receptor Antagonist for Treatment of Asthma
Sandham, David A, Barker, Lucy, Brown, Lyndon, Brown, Zarin, Budd, David, Charlton, Steven J, Chatterjee, Devnandan, Cox, Brian, Dubois, Gerald, Duggan, Nicholas, Hall, Edward, Hatto, Julia, Maas, Janet, Manini, Jodie, Profit, Rachael, Riddy, Darren, Ritchie, Catherine, Sohal, Bindi, Shaw, Duncan, Stringer, Rowan, Sykes, David A, Thomas, Matthew, Turner, Katharine L, Watson, Simon J, West, Ryan, Willard, Elisabeth, Williams, Gareth, Willis, Jennifer
Published in ACS medicinal chemistry letters (11.05.2017)
Published in ACS medicinal chemistry letters (11.05.2017)
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Journal Article