ADO-RESISTANT CYSTEAMINE ANALOGS AND USES THEREOF
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Year of Publication 27.01.2022
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Year of Publication 27.01.2022
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PYRIMIDINE CYCLOHEXENYL GLUCOCORTICOID RECEPTOR MODULATORS
BAKER, Thomas Matthew, CREPIN, Damien Francis Philippe, HUNT, Hazel, DUFFY, Lorna, HILL-COUSINS, Joseph Thomas
Year of Publication 26.01.2022
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Year of Publication 26.01.2022
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COMPOUNDS
DUFFY, Lorna, WRIGGLESWORTH, Joseph, GEORGE, Pascal, NOVAK, Andrew, BIRCH, Louise, JONES, Geraint
Year of Publication 09.12.2021
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Year of Publication 09.12.2021
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N-(5-(6-ethoxypyrazin-2-yl)pyridin-2-yl)-4-(2-(methylsulfonamido)pyrimidin-4-yl) tetrahydro-2H-pyran-4-carboxamide derivatives and related compounds as human CTPS1 inhibitors for the treatment of proliferative diseases
Jones, Geraint, Birch, Louise, George, Pascal, Novak, Andrew, Blackham, Emma, Wrigglesworth, Joseph, Duffy, Lorna, Quddus, Abdul, Cousin, David, Ahmed, Saleh
Year of Publication 13.10.2022
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Year of Publication 13.10.2022
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Aminopyrimidine/pyrazine derivatives as CTPS1 inhibitors
BLACKHAM, Emma, DUFFY, Lorna, WRIGGLESWORTH, Joseph, GEORGE, Pascal, QUDDUS, Abdul, NOVAK, Andrew, COUSIN, David, AHMED, Saleh, BIRCH, Louise, JONES, Geraint
Year of Publication 08.09.2022
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Year of Publication 08.09.2022
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SULFONAMIDE INHIBITORS AS CTPS 1 INHIBITORS
BLACKHAM, Emma, DUFFY, Lorna, WRIGGLESWORTH, Joseph, GEORGE, Pascal, QUDDUS, Abdul, NOVAK, Andrew, COUSIN, David, AHMED, Saleh, BIRCH, Louise, JONES, Geraint
Year of Publication 17.08.2022
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Year of Publication 17.08.2022
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SULFONAMIDE DERIVATIVES AS CTPS1 INHIBITORS
BLACKHAM, Emma, DUFFY, Lorna, WRIGGLESWORTH, Joseph, GEORGE, Pascal, QUDDUS, Abdul, NOVAK, Andrew, COUSIN, David, AHMED, Saleh, BIRCH, Louise, JONES, Geraint
Year of Publication 17.08.2022
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Year of Publication 17.08.2022
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PYRIMIDINE CYCLOHEXENYL GLUCOCORTICOID RECEPTOR MODULATORS
BAKER, Thomas Matthew, CREPIN, Damien Francis Philippe, HUNT, Hazel, DUFFY, Lorna, HILL-COUSINS, Joseph Thomas
Year of Publication 05.08.2021
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Year of Publication 05.08.2021
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Aminothiazole compounds as inhibitors of CTPS1
Jones, Geraint, Birch, Louise, Chatzopoulou, Elli, Thomas, Jennifer, George, Pascal, Novak, Andrew, Blackham, Emma, Wrigglesworth, Joseph, Duffy, Lorna, Quddus, Abdul, Cousin, David, Ahmed, Saleh
Year of Publication 23.05.2023
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Year of Publication 23.05.2023
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N-(4-(5-chloropyridin-3-yl)phenyl)-2-(2-(cyclopropanesulfonamido)pyrimidin-4-yl) butanamide derivatives and related compounds as human CTPS1 inhibitors for the treatment of proliferative diseases
Jones, Geraint, Novak, Andrew, Blackham, Emma, Wrigglesworth, Joseph, Birch, Louise, Thomas, Jennifer, George, Pascal, Duffy, Lorna, Toschi, Gianna, Quddus, Abdul, Cousin, David, Chatzopoulou, Ellie, Ahmed, Saleh
Year of Publication 23.03.2023
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Year of Publication 23.03.2023
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N-(5-(6-ETHOXYPYRAZIN-2-YL)PYRIDIN-2-YL)-4-(2-(METHYLSULFONAMIDO)PYRIMIDIN-4-YL) TETRAHYDRO-2H-PYRAN-4-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS HUMAN CTPS1 INHIBITORS FOR THE TREATMENT OF PROLIFERATIVE DISEASES
BLACKHAM, Emma, DUFFY, Lorna, WRIGGLESWORTH, Joseph, GEORGE, Pascal, QUDDUS, Abdul, NOVAK, Andrew, COUSIN, David, AHMED, Saleh, BIRCH, Louise, JONES, Geraint
Year of Publication 13.04.2022
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Year of Publication 13.04.2022
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COMPOSITIONS AND METHODS OF USING THE SAME FOR TREATMENT OF NEURODEGENERATIVE AND MITOCHONDRIAL DISEASE
SULEMAN, Abid, HOBRATH, Varady, MCDONALD, Rory, DUFFY, Lorna, DEVITA, Robert, HERTZ, Nicholas, INCERTI-PRADILLOS, Celia, JOHNSTONE, Shawn, BARTHOLOMEUS, Johan, DITSWORTH, Dara
Year of Publication 23.02.2023
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Year of Publication 23.02.2023
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PYRIMIDINE CYCLOHEXENYL GLUCOCORTICOID RECEPTOR MODULATORS
BAKER, Thomas Matthew, CREPIN, Damien Francis Philippe, HUNT, Hazel, DUFFY, Lorna, HILL-COUSINS, Joseph Thomas
Year of Publication 14.04.2021
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Year of Publication 14.04.2021
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ADO-resistant cysteamine analogs and uses thereof
Phillips, Timothy, Gourdet, Benoit, Zankel, Todd C, Duffy, Lorna, Unitt, John
Year of Publication 02.02.2021
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Year of Publication 02.02.2021
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QUATERNARY INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS
PHILLIPS, Andrew William, HUNT, Hazel, DUFFY, Lorna, JOUANNEAU, Morgan, STRUTT, Ian, HORNSBY, Thomas, MILLS, Mark, WARD, Jon-Paul
Year of Publication 30.12.2021
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Year of Publication 30.12.2021
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QUATERNARY INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS
HUNT, HAZEL, DUFFY, LORNA, MILLS, MARK, HORNSBY, THOMAS, PHILLIPS, ANDREW WILLIAM, STRUTT, IAN, JOUANNEAU, MORGAN, WARD, JON-PAUL
Year of Publication 30.12.2021
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Year of Publication 30.12.2021
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Compounds
Jones, Geraint, Birch, Louise, George, Pascal, Novak, Andrew, Blackham, Emma, Wrigglesworth, Joseph, Duffy, Lorna, Quddus, Abdul, Cousin, David, Ahmed, Saleh
Year of Publication 16.12.2021
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Year of Publication 16.12.2021
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Pyrimidine cyclohexenyl glucocorticoid receptor modulators
BAKER, Thomas Matthew, CREPIN, Damien Francis Philippe, HUNT, Hazel, DUFFY, Lorna, HILL-COUSINS, Joseph Thomas
Year of Publication 07.01.2021
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Year of Publication 07.01.2021
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