Induced protein degradation of anaplastic lymphoma kinase (ALK) by proteolysis targeting chimera (PROTAC)
Kang, Chung Hyo, Lee, Dong Ho, Lee, Chong Ock, Du Ha, Jae, Park, Chi Hoon, Hwang, Jong Yeon
Published in Biochemical and biophysical research communications (28.10.2018)
Published in Biochemical and biophysical research communications (28.10.2018)
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Design and characterization of cereblon-mediated androgen receptor proteolysis-targeting chimeras
Takwale, Akshay D., Jo, Seung-Hyun, Jeon, Yeong Uk, Kim, Hyung Soo, Shin, Choong Hoon, Lee, Heung Kyoung, Ahn, Sunjoo, Lee, Chong Ock, Du Ha, Jae, Kim, Jeong-Hoon, Hwang, Jong Yeon
Published in European journal of medicinal chemistry (15.12.2020)
Published in European journal of medicinal chemistry (15.12.2020)
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Combination Treatment with GSK126 and Pomalidomide Induces B-Cell Differentiation in EZH2 Gain-of-Function Mutant Diffuse Large B-Cell Lymphoma
Park, Sungryul, Jo, Seung-Hyun, Kim, Jong-Hwan, Kim, Seon-Young, Ha, Jae Du, Hwang, Jong Yeon, Lee, Myeong Youl, Kang, Jong Soon, Han, Tae-Su, Park, Sung Goo, Kim, Sunhong, Park, Byoung Chul, Kim, Jeong-Hoon
Published in Cancers (01.09.2020)
Published in Cancers (01.09.2020)
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Synthesis and biological evaluation of rhodanine derivatives as PRL-3 inhibitors
Ahn, Jin Hee, Kim, Seung Jun, Park, Woul Seong, Cho, Sung Yun, Ha, Jae Du, Kim, Sung Soo, Kang, Seung Kyu, Jeong, Dae Gwin, Jung, Suk-Kyeong, Lee, Sang-Hyeup, Kim, Hwan Mook, Park, Song Kyu, Lee, Ki Ho, Lee, Chang Woo, Ryu, Seong Eon, Choi, Joong-Kwon
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
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Augmentation of the antitumor effects of PARP inhibitors in triple-negative breast cancer via degradation by hydrophobic tagging modulation
Go, Ahra, Jang, Jeong Woon, Lee, Woori, Ha, Jae Du, Kim, Hyun Jin, Nam, Hye Jin
Published in European journal of medicinal chemistry (15.10.2020)
Published in European journal of medicinal chemistry (15.10.2020)
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Synthesis and structure–activity relationship of aminopyridines with substituted benzoxazoles as c-Met kinase inhibitors
Lee, Jongkook, Han, Sun-Young, Jung, Heejung, Yang, Jeon, Choi, Jie-Won, Chae, Chong Hack, Park, Chi Hoon, Choi, Sang Un, Lee, Kwangho, Ha, Jae Du, Lee, Chong Ock, Ryu, Jae Wook, Kim, Hyoung Rae, Koh, Jong Sung, Cho, Sung Yun
Published in Bioorganic & medicinal chemistry letters (15.06.2012)
Published in Bioorganic & medicinal chemistry letters (15.06.2012)
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Cereblon contributes to cardiac dysfunction by degrading Cav1.2α
Park, Nammi, Marquez, Jubert, Pham, Trong Kha, Ko, Tae Hee, Youm, Jae Boum, Kim, Min, Choi, Seung Hak, Moon, Jiyoung, Flores, Jessa, Ko, Kyung Soo, Rhee, Byoung Doo, Shimizu, Ippei, Minamino, Tohru, Ha, Jae Du, Hwang, Jong Yeon, Yang, Seung Joo, Park, Chul-Seung, Kim, Hyoung Kyu, Han, Jin
Published in European heart journal (21.05.2022)
Published in European heart journal (21.05.2022)
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A Novel Series of Highly Potent Small Molecule Inhibitors of Rhinovirus Replication
Kim, Jinwoo, Jung, Yu Kyoung, Kim, Chonsaeng, Shin, Jin Soo, Scheers, Els, Lee, Joo-Youn, Han, Soo Bong, Lee, Chong-Kyo, Neyts, Johan, Ha, Jae-Du, Jung, Young-Sik
Published in Journal of medicinal chemistry (13.07.2017)
Published in Journal of medicinal chemistry (13.07.2017)
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Discovery of aminopyridines substituted with benzoxazole as orally active c-Met kinase inhibitors
Cho, Sung Yun, Han, Sun-Young, Ha, Jae Du, Ryu, Jae Wook, Lee, Chong Ock, Jung, Heejung, Kang, Nam Sook, Kim, Hyoung Rae, Koh, Jong Sung, Lee, Jongkook
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
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Disordered region of cereblon is required for efficient degradation by proteolysis-targeting chimera
Kim, Kidae, Lee, Dong Ho, Park, Sungryul, Jo, Seung-Hyun, Ku, Bonsu, Park, Sung Goo, Park, Byoung Chul, Jeon, Yeong Uk, Ahn, Sunjoo, Kang, Chung Hyo, Hwang, Daehee, Chae, Sehyun, Ha, Jae Du, Kim, Sunhong, Hwang, Jong Yeon, Kim, Jeong-Hoon
Published in Scientific reports (23.12.2019)
Published in Scientific reports (23.12.2019)
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Design and synthesis of triazolopyridazines substituted with methylisoquinolinone as selective c-Met kinase inhibitors
Ryu, Jae Wook, Han, Sun-Young, Yun, Jeong In, Choi, Sang-Un, Jung, Heejung, Ha, Jae Du, Cho, Sung Yun, Lee, Chong Ock, Kang, Nam Sook, Koh, Jong Sung, Kim, Hyoung Rae, Lee, Jongkook
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
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Synthesis and biological evaluation of N9-cis-cyclobutylpurine derivatives for use as cyclin-dependent kinase (CDK) inhibitors
Park, Sun Jun, Kim, Eunjin, Yoo, Miyoun, Lee, Joo-Youn, Park, Chi Hoon, Hwang, Jong Yeon, Ha, Jae Du
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
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cIAPs promote the proteasomal degradation of mutant SOD1 linked to familial amyotrophic lateral sclerosis
Choi, Jin Sun, Kim, Kidae, Lee, Do Hee, Cho, Sayeon, Ha, Jae Du, Park, Byoung Chul, Kim, Sunhong, Park, Sung Goo, Kim, Jeong-Hoon
Published in Biochemical and biophysical research communications (18.11.2016)
Published in Biochemical and biophysical research communications (18.11.2016)
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Synthesis and evaluation of novel 2,4-diaminopyrimidines bearing bicyclic aminobenzazepines for anaplastic lymphoma kinase (ALK) inhibitor
Kang, Ga Ae, Lee, Minji, Song, Dawn, Lee, Heung Kyoung, Ahn, Sunjoo, Park, Chi Hoon, Lee, Chong Ock, Yun, Chang Soo, Jung, Heejung, Kim, Pilho, Ha, Jae Du, Cho, Sung Yun, Kim, Hyoung Rae, Hwang, Jong Yeon
Published in Bioorganic & medicinal chemistry letters (15.09.2015)
Published in Bioorganic & medicinal chemistry letters (15.09.2015)
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Replacing the terminal piperidine in ceritinib with aliphatic amines confers activities against crizotinib-resistant mutants including G1202R
Mathi, Gangadhar Rao, Kang, Chung Hyo, Lee, Heung Kyoung, Achary, Raghavendra, Lee, Ha-Yeon, Lee, Joo-Youn, Ha, Jae Du, Ahn, Sunjoo, Park, Chi Hoon, Lee, Chong Ock, Hwang, Jong Yeon, Yun, Chang-Soo, Jung, Hee Jung, Cho, Sung Yun, Kim, Hyoung Rae, Kim, Pilho
Published in European journal of medicinal chemistry (27.01.2017)
Published in European journal of medicinal chemistry (27.01.2017)
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4-Substituted quinazoline derivatives as novel EphA2 receptor tyrosine kinase inhibitors
Lim, Chae Jo, Oh, Kwang-Seok, Ha, Jae Du, Lee, Jeong Hyun, Seo, Ho Won, Chae, Chong Hack, Kim, Dae-Ghon, Lee, Mi-Jin, Lee, Byung Ho
Published in Bioorganic & medicinal chemistry letters (01.09.2014)
Published in Bioorganic & medicinal chemistry letters (01.09.2014)
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Novel bis-ortho-alkoxy-para-piperazinesubstituted-2,4-dianilinopyrimidines (KRCA-0008) as potent and selective ALK inhibitors for anticancer treatment
Park, Chi Hoon, Choe, Hyeonjeong, Jang, In-Young, Kwon, So Yeong, Latif, Muhammad, Lee, Heung Kyoung, Lee, Hyeon Ji, Yang, Eun Hye, Yun, Jeong In, Chae, Chong Hak, Cho, Sung Yun, Choi, Sang Un, Ha, Jae Du, Jung, Heejung, Kim, Hyoung Rae, Kim, Pilho, Lee, Chong Ock, Yun, Chang-Soo, Lee, Kwangho
Published in Bioorganic & medicinal chemistry letters (15.11.2013)
Published in Bioorganic & medicinal chemistry letters (15.11.2013)
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Development of potent ALK inhibitor and its molecular inhibitory mechanism against NSCLC harboring EML4-ALK proteins
Kang, Chung Hyo, Yun, Jeong In, Lee, Kwangho, Lee, Chong Ock, Lee, Heung Kyoung, Yun, Chang-Soo, Hwang, Jong Yeon, Cho, Sung Yun, Jung, Heejung, Kim, Pilho, Ha, Jae Du, Jeon, Jeong Hee, Choi, Sang Un, Jeong, Hye Gwang, Kim, Hyoung Rae, Park, Chi Hoon
Published in Biochemical and biophysical research communications (28.08.2015)
Published in Biochemical and biophysical research communications (28.08.2015)
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Therapeutic Efficacy of ABN401, a Highly Potent and Selective MET Inhibitor, Based on Diagnostic Biomarker Test in MET-Addicted Cancer
Kim, Jooseok, Park, Kyung Eui, Jeong, Yoo-Seong, Kim, YeongMun, Park, Hayeon, Nam, Ji-Hye, Jung, Kyungsoo, Son, Woo Sung, Jung, Hun Soon, Lee, Jong-Hwa, Jeong, Seong Hoon, Kim, Nam Ah, Ha, Jae Du, Cho, Sung Yun, Choi, Yoon-La, Chung, Suk-Jae, Choi, Jun Young, Hong, Sungyoul, Shin, Young Kee
Published in Cancers (15.06.2020)
Published in Cancers (15.06.2020)
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