Structural basis of ketamine action on human NMDA receptors
Zhang, Youyi, Ye, Fei, Zhang, Tongtong, Lv, Shiyun, Zhou, Liping, Du, Daohai, Lin, He, Guo, Fei, Luo, Cheng, Zhu, Shujia
Published in Nature (London) (12.08.2021)
Published in Nature (London) (12.08.2021)
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Identification and Assessments of Novel and Potent Small-Molecule Inhibitors of EED–EZH2 Interaction of Polycomb Repressive Complex 2 by Computational Methods and Biological Evaluations
Zhu, Kongkai, Du, Daohai, Yang, Rui, Tao, Hongrui, Zhang, Hua
Published in Chemical & pharmaceutical bulletin (01.01.2020)
Published in Chemical & pharmaceutical bulletin (01.01.2020)
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Astemizole Arrests the Proliferation of Cancer Cells by Disrupting the EZH2-EED Interaction of Polycomb Repressive Complex 2
Kong, Xiangqian, Chen, Limin, Jiao, Lianying, Jiang, Xiangrui, Lian, Fulin, Lu, Junyan, Zhu, Kongkai, Du, Daohai, Liu, Jingqiu, Ding, Hong, Zhang, Naixia, Shen, Jingshan, Zheng, Mingyue, Chen, Kaixian, Liu, Xin, Jiang, Hualiang, Luo, Cheng
Published in Journal of medicinal chemistry (26.11.2014)
Published in Journal of medicinal chemistry (26.11.2014)
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Identification of novel EZH2 inhibitors through pharmacophore-based virtual screening and biological assays
Wu, Yunlong, Hu, Junchi, Ding, Hong, Chen, Limin, Zhang, Yuanyuan, Liu, Rongfeng, Xu, Pan, Du, Daohai, Lu, Wenchao, Liu, Jingqiu, Liu, Yan, Liu, Yu-Chih, Lu, Junyan, Zhang, Jin, Yao, Zhiyi, Luo, Cheng
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
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The discovery of a non-competitive GOT1 inhibitor, hydralazine hydrochloride, via a coupling reaction-based high-throughput screening assay
Wu, Qiqi, Sun, Zhongya, Chen, Zhifeng, Liu, Jingqiu, Ding, Hong, Luo, Cheng, Wang, Mingliang, Du, Daohai
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
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Structure-Based Design and Discovery of a Potent and Cell-Active LC3A/B Covalent Inhibitor
Zhou, Zhenfei, Huang, Siqi, Fan, Shijie, Li, Xueyuan, Wang, Chengyu, Yu, Wanlin, Du, Daohai, Zhang, Yuanyuan, Chen, Kaixian, Fu, Wei, Luo, Cheng
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Uncovering PROTAC Sensitivity and Efficacy by Multidimensional Proteome Profiling: A Case for STAT3
Suo, Yuying, Du, Daohai, Chen, Chao, Zhu, Hongwen, Wang, Xiongjun, Song, Nixue, Lu, Dayun, Yang, Yaxi, Li, Jiacheng, Wang, Jun, Luo, Zhongyuan, Zhou, Bing, Luo, Cheng, Zhou, Hu
Published in Journal of medicinal chemistry (28.03.2024)
Published in Journal of medicinal chemistry (28.03.2024)
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Author Correction: Structural basis of ketamine action on human NMDA receptors
Zhang, Youyi, Ye, Fei, Zhang, Tongtong, Lv, Shiyun, Zhou, Liping, Du, Daohai, Lin, He, Guo, Fei, Luo, Cheng, Zhu, Shujia
Published in Nature (London) (28.10.2021)
Published in Nature (London) (28.10.2021)
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Discovery of 2-substituted-N-(3-(3,4-dihydroisoquinolin-2(1H)-yl)-2-hydroxypropyl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide as potent and selective protein arginine methyltransferases 5 inhibitors: Design, synthesis and biological evaluation
Shao, Jingwei, Zhu, Kongkai, Du, Daohai, Zhang, Yuanyuan, Tao, Hongrui, Chen, Zhifeng, Jiang, Hualiang, Chen, Kaixian, Luo, Cheng, Duan, Wenhu
Published in European journal of medicinal chemistry (15.02.2019)
Published in European journal of medicinal chemistry (15.02.2019)
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Discovery and characterization of a novel glucose-6-phosphate dehydrogenase (G6PD) inhibitor via high-throughput screening
Luo, Zhongyuan, Du, Daohai, Liu, Yanjun, Lu, Tian, Liu, Liping, Jiang, Hualiang, Chen, Kaixian, Shan, Changliang, Luo, Cheng
Published in Bioorganic & medicinal chemistry letters (15.05.2021)
Published in Bioorganic & medicinal chemistry letters (15.05.2021)
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Computational and Structure-Based Development of High Potent Cell-Active Covalent Inhibitor Targeting the Peptidyl-Prolyl Isomerase NIMA-Interacting‑1 (Pin1)
Liu, Liping, Zhu, Rui, Li, Jiacheng, Pei, Yuan, Wang, Shuangshuang, Xu, Pan, Wang, Mingyu, Wen, Yu, Zhang, Hao, Du, Daohai, Ding, Hong, Jiang, Hualiang, Chen, Kaixian, Zhou, Bing, Yu, Lifang, Luo, Cheng
Published in Journal of medicinal chemistry (10.02.2022)
Published in Journal of medicinal chemistry (10.02.2022)
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Identification and assessments of novel and potent small-molecule inhibitors of EED-EZH2 interaction of polycomb repressive complex 2 by computational methods and biological evaluations
Zhu, Kongkai, Du, Daohai, Yang, Rui, Tao, Hongrui, Zhang, Hua
Published in Chemical and Pharmaceutical Bulletin (2019)
Published in Chemical and Pharmaceutical Bulletin (2019)
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Structure-Guided Development of Small-Molecule PRC2 Inhibitors Targeting EZH2–EED Interaction
Du, Daohai, Xu, Dandan, Zhu, Licheng, Stazi, Giulia, Zwergel, Clemens, Liu, Yanli, Luo, Zhongyuan, Li, Yuanqing, Zhang, Yuanyuan, Zhu, Kongkai, Ding, Yiluan, Liu, Jingqiu, Fan, Shijie, Zhao, Kaiyan, Zhang, Naixia, Kong, Xiangqian, Jiang, Hualiang, Chen, Kaixian, Zhao, Kehao, Valente, Sergio, Min, Jinrong, Duan, Wenhu, Luo, Cheng
Published in Journal of medicinal chemistry (24.06.2021)
Published in Journal of medicinal chemistry (24.06.2021)
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A RhoA structure with switch II flipped outward revealed the conformational dynamics of switch II region
Jiang, Hao, Zu, Shijia, Lu, Yu, Sun, Zhongya, Adeerjiang, Akejiang, Guo, Qiao, Zhang, Huimin, Dong, Chen, Wu, Qiqi, Ding, Hong, Du, Daohai, Wang, Mingliang, Liu, Chuanpeng, Tang, Yong, Liang, Zhongjie, Luo, Cheng
Published in Journal of structural biology (01.06.2023)
Published in Journal of structural biology (01.06.2023)
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Identification of novel inhibitors of histone acetyltransferase hMOF through high throughput screening
Zhang, Rukang, Wang, Jiang, Zhao, Liang, Liu, Shien, Du, Daohai, Ding, Hong, Chen, Shijie, Yue, Liyan, Liu, Yu-Chih, Zhang, Chenhua, Liu, Hong, Luo, Cheng
Published in European journal of medicinal chemistry (05.09.2018)
Published in European journal of medicinal chemistry (05.09.2018)
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(−)-Epigallocatechin Gallate is a Noncompetitive Inhibitor of NAD Kinase
Liu, Tonghai, Shi, Wenjia, Ding, Yiluan, Wu, Qiqi, Zhang, Bei, Zhang, Naixia, Wang, Mingliang, Du, Daohai, Zhang, Hao, Han, Bo, Guo, Dean, Zheng, Jie, Li, Qi, Luo, Cheng
Published in ACS medicinal chemistry letters (10.11.2022)
Published in ACS medicinal chemistry letters (10.11.2022)
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Expressed sequence tags analysis revealing the taxonomic position and fatty acid biosynthesis in an oleaginous green microalga, Myrmecia incisa Reisigl (Trebouxiophyceae, Chlorophyta)
Ouyang, LongLing, Du, DaoHai, Yu, ShuiYan, Li, ChunYang, Zhang, ChengWu, Gao, HongJian, Zhou, ZhiGang
Published in Chinese science bulletin (01.09.2012)
Published in Chinese science bulletin (01.09.2012)
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Removement of Ni²+ from Waste Water by Mentallothionein (MT) Transgenic Cyanobacterium
Ning Zou, Daohai Du, Shengchen Liu, Donghong Sun, Binggen Ru
Published in 2008 2nd International Conference on Bioinformatics and Biomedical Engineering (01.05.2008)
Published in 2008 2nd International Conference on Bioinformatics and Biomedical Engineering (01.05.2008)
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