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Structural Alert/Reactive Metabolite Concept as Applied in Medicinal Chemistry to Mitigate the Risk of Idiosyncratic Drug Toxicity: A Perspective Based on the Critical Examination of Trends in the Top 200 Drugs Marketed in the United States
Stepan, Antonia F, Walker, Daniel P, Bauman, Jonathan, Price, David A, Baillie, Thomas A, Kalgutkar, Amit S, Aleo, Michael D
Published in Chemical research in toxicology (19.09.2011)
Published in Chemical research in toxicology (19.09.2011)
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Validation of a microdose probe drug cocktail for clinical drug interaction assessments for drug transporters and CYP3A
Prueksaritanont, T, Tatosian, D A, Chu, X, Railkar, R, Evers, R, Chavez-Eng, C, Lutz, R, Zeng, W, Yabut, J, Chan, G H, Cai, X, Latham, A H, Hehman, J, Stypinski, D, Brejda, J, Zhou, C, Thornton, B, Bateman, K P, Fraser, I, Stoch, S A
Published in Clinical pharmacology and therapeutics (01.04.2017)
Published in Clinical pharmacology and therapeutics (01.04.2017)
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Breast Cancer Resistance Protein (ABCG2) in Clinical Pharmacokinetics and Drug Interactions: Practical Recommendations for Clinical Victim and Perpetrator Drug-Drug Interaction Study Design
Lee, Caroline A, O’Connor, Meeghan A, Ritchie, Tasha K, Galetin, Aleksandra, Cook, Jack A, Ragueneau-Majlessi, Isabelle, Ellens, Harma, Feng, Bo, Taub, Mitchell E, Paine, Mary F, Polli, Joseph W, Ware, Joseph A, Zamek-Gliszczynski, Maciej J
Published in Drug metabolism and disposition (01.04.2015)
Published in Drug metabolism and disposition (01.04.2015)
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Serum retinyl esters are positively correlated with analyzed total liver vitamin A reserves collected from US adults at time of death
Olsen, Kiersten, Suri, Devika J, Davis, Christopher, Sheftel, Jesse, Nishimoto, Kohei, Yamaoka, Yusuke, Toya, Yutaka, Welham, Nathan V, Tanumihardjo, Sherry A
Published in The American journal of clinical nutrition (01.11.2018)
Published in The American journal of clinical nutrition (01.11.2018)
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Heme-nitrosylated hemoglobin and oxidative stress in women consuming combined contraceptives. Clinical application of the EPR spectroscopy
Lobysheva, Irina I., van Eeckhoudt, Sandrine, Dei Zotti, Flavia, Rifahi, Ahmad, Pothen, Lucie, Beauloye, Christophe, Balligand, Jean-Luc
Published in Free radical biology & medicine (01.07.2017)
Published in Free radical biology & medicine (01.07.2017)
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Assessment of Transporter Polymorphisms as a Factor in a BCRP Drug Interaction Study With Lanabecestat
Willis, Brian A, Andersen, Scott W, Ayan-Oshodi, Mosun, James, Douglas E, Liffick, Emily, Hillgren, Kathleen, Guo, Yingying, Monk, Scott A
Published in Journal of clinical pharmacology (01.01.2020)
Published in Journal of clinical pharmacology (01.01.2020)
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Drugs affecting renin-angiotensin-aldosterone system and the cancer risk: A meta-analysis of nested case-control studies
Dong-Mei, Liu, Wei, Zhang, Guang-Jun, Hao, Lu, James, Jian-Lun, Han, Jian, Zhang
Published in Pakistan journal of pharmaceutical sciences (01.01.2021)
Published in Pakistan journal of pharmaceutical sciences (01.01.2021)
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Best Practices for Metabolite Quantification in Drug Development: Updated Recommendation from The European Bioanalysis Forum
Timmerman, Philip, Blech, Stefan, White, Stephen, Green, Martha, Delatour, Claude, McDougall, Stuart, Mannens, Geert, Smeraglia, John, Williams, Stephen, Young, Graeme
Published in Bioanalysis (01.06.2016)
Published in Bioanalysis (01.06.2016)
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Safety and pharmacokinetics of the CIME combination of drugs and their metabolites after a single oral dosing in healthy volunteers
Lenuzza, Natacha, Duval, Xavier, Nicolas, Grégory, Thévenot, Etienne, Job, Sylvie, Videau, Orianne, Narjoz, Céline, Loriot, Marie-Anne, Beaune, Philippe, Becquemont, Laurent, Mentré, France, Funck-Brentano, Christian, Alavoine, Loubna, Arnaud, Philippe, Delaforge, Marcel, Bénech, Henri
Published in European journal of drug metabolism and pharmacokinetics (01.04.2016)
Published in European journal of drug metabolism and pharmacokinetics (01.04.2016)
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The prevention of adverse drug reactions in older subjects
Cherubini, Antonio, Ruggiero, Carmelinda, Gasperini, Beatrice, Dell'Aquila, Giuseppina, Cupido, Maria Grazia, Zampi, Elena, Zengarini, Elisa, Nguyen, Nguyen Hao, Serra, Rocco, Corsonello, Andrea, Lattanzio, Fabrizia
Published in Current drug metabolism (01.09.2011)
Published in Current drug metabolism (01.09.2011)
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Pharmacogenetics in geriatric medicine: challenges and opportunities for clinical practice
Pilotto, Alberto, Panza, Francesco, Seripa, Davide
Published in Current drug metabolism (01.09.2011)
Published in Current drug metabolism (01.09.2011)
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Controlled diuretic monotherapy in hypertensive patients: Efficiency and metabolic safety
Semenkin, A A, Zhivilova, L A, Nechaeva, G I, Chindareva, O I, Loginova, E N, Pritykina, T V
Published in Terapevtic̆eskii arhiv (01.01.2016)
Published in Terapevtic̆eskii arhiv (01.01.2016)
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