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Indole and Tryptophan Metabolism: Endogenous and Dietary Routes to Ah Receptor Activation
Hubbard, Troy D., Murray, Iain A., Perdew, Gary H.
Published in Drug metabolism and disposition (01.10.2015)
Published in Drug metabolism and disposition (01.10.2015)
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Physiologically Based Pharmacokinetic (PBPK) Modeling and Simulation Approaches: A Systematic Review of Published Models, Applications, and Model Verification
Sager, Jennifer E., Yu, Jingjing, Ragueneau-Majlessi, Isabelle, Isoherranen, Nina
Published in Drug metabolism and disposition (01.11.2015)
Published in Drug metabolism and disposition (01.11.2015)
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Trimethylamine and Trimethylamine N-Oxide, a Flavin-Containing Monooxygenase 3 (FMO3)-Mediated Host-Microbiome Metabolic Axis Implicated in Health and Disease
Fennema, Diede, Phillips, Ian R, Shephard, Elizabeth A
Published in Drug metabolism and disposition (01.11.2016)
Published in Drug metabolism and disposition (01.11.2016)
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The Nonclinical Disposition and Pharmacokinetic/Pharmacodynamic Properties of N-Acetylgalactosamine–Conjugated Small Interfering RNA Are Highly Predictable and Build Confidence in Translation to Human
McDougall, Robin, Ramsden, Diane, Agarwal, Sagar, Agarwal, Saket, Aluri, Krishna, Arciprete, Michael, Brown, Christopher, Castellanos-Rizaldos, Elena, Charisse, Klaus, Chong, Saeho, Cichocki, Joseph, Fitzgerald, Kevin, Goel, Varun, Gu, Yongli, Guenther, Dale, Habtemariam, Bahru, Jadhav, Vasant, Janas, Maja, Jayaraman, Muthusamy, Kurz, Jeffrey, Li, Jing, Liu, Ju, Liu, Xiumin, Liou, Steven, Maclauchlin, Chris, Maier, Martin, Manoharan, Muthiah, Nair, Jayaprakash K., Robbie, Gabriel, Schmidt, Karyn, Smith, Peter, Theile, Christopher, Vaishnaw, Akshay, Waldron, Scott, Xu, Yuanxin, Zhang, Xuemei, Zlatev, Ivan, Wu, Jing-Tao
Published in Drug metabolism and disposition (01.06.2022)
Published in Drug metabolism and disposition (01.06.2022)
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Adverse Drug Reactions and Toxicity of the Food and Drug Administration–Approved Antisense Oligonucleotide Drugs
Alhamadani, Feryal, Zhang, Kristy, Parikh, Rajvi, Wu, Hangyu, Rasmussen, Theodore P., Bahal, Raman, Zhong, Xiao-bo, Manautou, José E.
Published in Drug metabolism and disposition (01.06.2022)
Published in Drug metabolism and disposition (01.06.2022)
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Disposition of Nirmatrelvir, an Orally Bioavailable Inhibitor of SARS-CoV-2 3C-Like Protease, across Animals and Humans
Eng, Heather, Dantonio, Alyssa L., Kadar, Eugene P., Obach, R. Scott, Di, Li, Lin, Jian, Patel, Nandini C., Boras, Britton, Walker, Gregory S., Novak, Jonathan J., Kimoto, Emi, Singh, Ravi Shankar P., Kalgutkar, Amit S.
Published in Drug metabolism and disposition (01.05.2022)
Published in Drug metabolism and disposition (01.05.2022)
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Inhibition of the Multidrug Resistance P-Glycoprotein: Time for a Change of Strategy?
Callaghan, Richard, Luk, Frederick, Bebawy, Mary
Published in Drug metabolism and disposition (01.04.2014)
Published in Drug metabolism and disposition (01.04.2014)
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Brain Exposure of Two Selective Dual CDK4 and CDK6 Inhibitors and the Antitumor Activity of CDK4 and CDK6 Inhibition in Combination with Temozolomide in an Intracranial Glioblastoma Xenograft
Raub, Thomas J., Wishart, Graham N., Kulanthaivel, Palaniappan, Staton, Brian A., Ajamie, Rose T., Sawada, Geri A., Gelbert, Lawrence M., Shannon, Harlan E., Sanchez-Martinez, Concepcion, De Dios, Alfonso
Published in Drug metabolism and disposition (01.09.2015)
Published in Drug metabolism and disposition (01.09.2015)
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Quantitative Proteomics of Clinically Relevant Drug-Metabolizing Enzymes and Drug Transporters and Their Intercorrelations in the Human Small Intestine
Couto, Narciso, Al-Majdoub, Zubida M., Gibson, Stephanie, Davies, Pamela J., Achour, Brahim, Harwood, Matthew D., Carlson, Gordon, Barber, Jill, Rostami-Hodjegan, Amin, Warhurst, Geoffrey
Published in Drug metabolism and disposition (01.04.2020)
Published in Drug metabolism and disposition (01.04.2020)
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Cytochrome P450–Catalyzed Metabolism of Cannabidiol to the Active Metabolite 7-Hydroxy-Cannabidiol
Beers, Jessica L., Fu, Dong, Jackson, Klarissa D.
Published in Drug metabolism and disposition (01.10.2021)
Published in Drug metabolism and disposition (01.10.2021)
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Transcriptional, Functional, and Mechanistic Comparisons of Stem Cell–Derived Hepatocytes, HepaRG Cells, and Three-Dimensional Human Hepatocyte Spheroids as Predictive In Vitro Systems for Drug-Induced Liver Injury
Bell, Catherine C., Lauschke, Volker M., Vorrink, Sabine U., Palmgren, Henrik, Duffin, Rodger, Andersson, Tommy B., Ingelman-Sundberg, Magnus
Published in Drug metabolism and disposition (01.04.2017)
Published in Drug metabolism and disposition (01.04.2017)
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Commensal Gut Bacteria Convert the Immunosuppressant Tacrolimus to Less Potent Metabolites
Guo, Yukuang, Crnkovic, Camila Manoel, Won, Kyoung-Jae, Yang, Xiaotong, Lee, John Richard, Orjala, Jimmy, Lee, Hyunwoo, Jeong, Hyunyoung
Published in Drug metabolism and disposition (01.03.2019)
Published in Drug metabolism and disposition (01.03.2019)
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Drug Concentration Asymmetry in Tissues and Plasma for Small Molecule-Related Therapeutic Modalities
Zhang, Donglu, Hop, Cornelis E C A, Patilea-Vrana, Gabriela, Gampa, Gautham, Seneviratne, Herana Kamal, Unadkat, Jashvant D, Kenny, Jane R, Nagapudi, Karthik, Di, Li, Zhou, Lian, Zak, Mark, Wright, Matthew R, Bumpus, Namandjé N, Zang, Richard, Liu, Xingrong, Lai, Yurong, Khojasteh, S Cyrus
Published in Drug metabolism and disposition (01.10.2019)
Published in Drug metabolism and disposition (01.10.2019)
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Industry Perspective on the Pharmacokinetic and Absorption, Distribution, Metabolism, and Excretion Characterization of Heterobifunctional Protein Degraders
Volak, Laurie P., Duevel, Heide Marika, Humphreys, Sara, Nettleton, David, Phipps, Colin, Pike, Andy, Rynn, Caroline, Scott-Stevens, Paul, Zhang, Donglu, Zientek, Michael
Published in Drug metabolism and disposition (01.07.2023)
Published in Drug metabolism and disposition (01.07.2023)
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Berberine Directly Affects the Gut Microbiota to Promote Intestinal Farnesoid X Receptor Activation
Tian, Yuan, Cai, Jingwei, Gui, Wei, Nichols, Robert G., Koo, Imhoi, Zhang, Jingtao, Anitha, Mallappa, Patterson, Andrew D.
Published in Drug metabolism and disposition (01.02.2019)
Published in Drug metabolism and disposition (01.02.2019)
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Predicting the Potential for Cannabinoids to Precipitate Pharmacokinetic Drug Interactions via Reversible Inhibition or Inactivation of Major Cytochromes P450
Bansal, Sumit, Maharao, Neha, Paine, Mary F., Unadkat, Jashvant D.
Published in Drug metabolism and disposition (01.10.2020)
Published in Drug metabolism and disposition (01.10.2020)
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