Tolerability of fosaprepitant and bioequivalency to aprepitant in healthy subjects
Lasseter, Kenneth C, Gambale, Jay, Jin, Bo, Bergman, Art, Constanzer, Marvin, Dru, James, Han, Tae H, Majumdar, Anup, Evans, Judith K, Murphy, M Gail
Published in Journal of clinical pharmacology (01.07.2007)
Published in Journal of clinical pharmacology (01.07.2007)
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Assessment of the CYP3A-mediated drug interaction potential of anacetrapib, a potent cholesteryl ester transfer protein (CETP) inhibitor, in healthy volunteers
Krishna, Rajesh, Bergman, Arthur J, Jin, Bo, Garg, Amit, Roadcap, Brad, Chiou, Rita, Dru, James, Cote, Josee, Laethem, Tine, Wang, Regina W, Didolkar, Varsha, Vets, Eva, Gottesdiener, Keith, Wagner, John A
Published in Journal of clinical pharmacology (01.01.2009)
Published in Journal of clinical pharmacology (01.01.2009)
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Metabolism and Excretion of Anacetrapib, a Novel Inhibitor of the Cholesteryl Ester Transfer Protein, in Humans
KUMAR, Sanjeev, TAN, Eugene Y, KARANAM, Bindhu, DEAN, Dennis C, GENDRANO, Isaias Noel, GRAVES, Mark W, WAGNER, John A, KRISHNA, Rajesh, HARTMANN, Georgy, BIDDLE, Zachary, BERGMAN, Arthur J, DRU, James, HO, Jonathan Z, JONES, Allen N, STASKIEWICZ, Steve J, BRAUN, Matthew P
Published in Drug metabolism and disposition (01.03.2010)
Published in Drug metabolism and disposition (01.03.2010)
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Effects of aprepitant on cytochrome P450 3A4 activity using midazolam as a probe
Majumdar, Anup K, McCrea, Jacqueline B, Panebianco, Deborah L, Hesney, Michael, Dru, James, Constanzer, Marvin, Goldberg, Michael R, Murphy, Gail, Gottesdiener, Keith M, Lines, Christopher R, Petty, Kevin J, Blum, Robert A
Published in Clinical pharmacology and therapeutics (01.08.2003)
Published in Clinical pharmacology and therapeutics (01.08.2003)
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Lack of Effect of Aprepitant or Its Prodrug Fosaprepitant on QTc Intervals in Healthy Subjects
MARBURY, Thomas C, BO JIN, PANEBIANCO, Deborah, GAIL MURPHY, M, HONG SUN, EVANS, Judith K, HAN, Tae H, CONSTANZER, Marvin L, DRU, James, SHADLE, Craig R
Published in Anesthesia and analgesia (01.08.2009)
Published in Anesthesia and analgesia (01.08.2009)
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Effect of aprepitant on the pharmacokinetics of intravenous midazolam
Majumdar, Anup K, Yan, Kerri X, Selverian, Diana V, Barlas, Suna, Constanzer, Marvin, Dru, James, McCrea, Jacqueline B, Ahmed, Tuli, Frick, Glen S, Kraft, Walter K, Petty, Kevin J, Greenberg, Howard E
Published in Journal of clinical pharmacology (01.06.2007)
Published in Journal of clinical pharmacology (01.06.2007)
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