A bifunctional-biased mu-opioid agonist-neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects
Drieu la Rochelle, Armand, Guillemyn, Karel, Dumitrascuta, Maria, Martin, Charlotte, Utard, Valérie, Quillet, Raphaëlle, Schneider, Séverine, Daubeuf, François, Willemse, Tom, Mampuys, Pieter, Maes, Bert U W, Frossard, Nelly, Bihel, Frédéric, Spetea, Mariana, Simonin, Frédéric, Ballet, Steven
Published in Pain (Amsterdam) (01.09.2018)
Published in Pain (Amsterdam) (01.09.2018)
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The Neutrophil Dynamic Mass Redistribution Assay as a Medium throughput Primary Cell Screening Assay
Stott, Lisa A, la Rochelle, Armand Drieu, Brown, Susan, Osborne, Greg, Hutchings, Catherine J, Poulter, Simon, Bennett, Kirstie A, Barnes, Matt
Published in The Journal of pharmacology and experimental therapeutics (01.04.2024)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2024)
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Identification of an N-acylated-(D)Arg-Leu-NH2 Dipeptide as a Highly Selective Neuropeptide FF1 Receptor Antagonist That Potently Prevents Opioid-Induced Hyperalgesia
Quillet, Raphaelle, Schneider, Severine, Utard, Valerie, la Rochelle, Armand Drieu, Elhabazi, Khadija, Henningsen, Jo Beldring, Gizzi, Patrick, Schmitt, Martine, Kugler, Valerie, Simonneaux, Valerie, Ilien, Brigitte, Simonin, Frederic, Bihel, Frederic
Published in Journal of medicinal chemistry (10.06.2021)
Published in Journal of medicinal chemistry (10.06.2021)
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Identification of an N -acylated- D Arg-Leu-NH 2 Dipeptide as a Highly Selective Neuropeptide FF1 Receptor Antagonist That Potently Prevents Opioid-Induced Hyperalgesia
Quillet, Raphaëlle, Schneider, Séverine, Utard, Valérie, Drieu la Rochelle, Armand, Elhabazi, Khadija, Henningsen, Jo Beldring, Gizzi, Patrick, Schmitt, Martine, Kugler, Valérie, Simonneaux, Valérie, Ilien, Brigitte, Simonin, Frédéric, Bihel, Frédéric
Published in Journal of medicinal chemistry (10.06.2021)
Published in Journal of medicinal chemistry (10.06.2021)
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Journal Article
Identification of an N‑acylated‑DArg-Leu-NH2 Dipeptide as a Highly Selective Neuropeptide FF1 Receptor Antagonist That Potently Prevents Opioid-Induced Hyperalgesia
Quillet, Raphaëlle, Schneider, Séverine, Utard, Valérie, Drieu la Rochelle, Armand, Elhabazi, Khadija, Henningsen, Jo Beldring, Gizzi, Patrick, Schmitt, Martine, Kugler, Valérie, Simonneaux, Valérie, Ilien, Brigitte, Simonin, Frédéric, Bihel, Frédéric
Published in Journal of medicinal chemistry (10.06.2021)
Published in Journal of medicinal chemistry (10.06.2021)
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