Pharmacological profile of GR117289 in vitro: a novel, potent and specific non‐peptide angiotensin AT1 receptor antagonist
Robertson, M.J., Barnes, J.C., Drew, G.M., Clark, K.L., Marshall, F.H., Michel, A., Middlemiss, D., Ross, B.C., Scopes, D., Dowle, M.D.
Published in British journal of pharmacology (01.12.1992)
Published in British journal of pharmacology (01.12.1992)
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Journal Article
Cardiovascular effects of GR117289, a novel angiotensin AT1 receptor antagonist
Hilditch, A., Hunt, A.A.E., Gardner, C.J., Twissell, D.J., Polley, J., Travers, A., Drew, G.M., Middlemiss, D., Ross, B.C., Robertson, M.J.
Published in British journal of pharmacology (01.01.1994)
Published in British journal of pharmacology (01.01.1994)
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Journal Article
α2‐Adrenoceptor blocking profile of SK&F 104078: further evidence for receptor subtypes
Akers, I., Coates, J., Drew, G.M., Sullivan, A.T.
Published in British journal of pharmacology (01.04.1991)
Published in British journal of pharmacology (01.04.1991)
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Journal Article
Bromobenzofurans : a new class of potent, non-peptide antagonists of angiotensin II
Middlemiss, D, Drew, G.M., Ross, B.C., Robertson, M.J., Scopes, D.I.C., Dowle, M.D., Akers, J, Cardwell, K, Clark, K.L., Coote, S, Eldred, C.D., Hamblett, J, Hilditch, A, Hirst, G.C., Jack, T, Montana, J, Panchal, T.A., Paton, J.M.S., Shah, P, Stuart, G, Travers, A
Published in Bioorganic & medicinal chemistry letters (1991)
Published in Bioorganic & medicinal chemistry letters (1991)
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Journal Article
Alpha 2-adrenoceptor blocking profile of SK&F 104078: further evidence for receptor subtypes
Akers, I, Coates, J, Drew, G M, Sullivan, A T
Published in British journal of pharmacology (01.04.1991)
Published in British journal of pharmacology (01.04.1991)
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Journal Article
Cardiovascular effects of GR117289, a novel angiotensin AT 1 receptor antagonist
Hilditch, A., Hunt, A.A.E., Gardner, C.J., Twissell, D.J., Polley, J., Travers, A., Drew, G.M., Middlemiss, D., Ross, B.C., Robertson, M.J.
Published in British journal of pharmacology (01.01.1994)
Published in British journal of pharmacology (01.01.1994)
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Journal Article
Pharmacological profile of GR117289 in vitro : a novel, potent and specific non‐peptide angiotensin AT 1 receptor antagonist
Robertson, M.J., Barnes, J.C., Drew, G.M., Clark, K.L., Marshall, F.H., Michel, A., Middlemiss, D., Ross, B.C., Scopes, D., Dowle, M.D.
Published in British journal of pharmacology (01.12.1992)
Published in British journal of pharmacology (01.12.1992)
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Journal Article
Benzofuran based angiotensin II antagonists related to GR117289: enhancement of potency in vitro and oral activity
Middlemiss, D., Watson, S.P., Ross, B.C., Dowle, M.D., Scopes, D.I.C., Montana, J.G., Shah, P., Hirst, G.C., Panchal, T.A., Paton, J.M.S., Pass, M., Hubbard, T., Hamblett, J., Cardwell, K.S., Jack, T.I., Stuart, G., Coote, S., Bradshaw, J., Drew, G.M., Hilditch, A., Clark, K.L., Robertson, M.J., Bayliss, M.K., Donnelly, M., Palmer, E., Manchee, G.R.M.
Published in Bioorganic & medicinal chemistry letters (1993)
Published in Bioorganic & medicinal chemistry letters (1993)
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Journal Article
Benzofuran based non-peptide antagonists of angiotensin II related to GR117289: part IV; imidazopyridinylbenzofurans
Judd, D.B., Cardwell, K.S., Panchal, T.A., Jack, T.I., Pass, M., Hubbard, T., Dean, A.W., Butt, A.U., Hobson, J.E., Heron, N.M., Watson, S.P., Currie, G.S., Middlemiss, D., Allen, D.G., Aston, N.M., Paton, J.M.S., Drew, G.M., Hilditch, A., Gallacher, D., Bayliss, M.K., Donnelly, M.C.
Published in Bioorganic & medicinal chemistry letters (10.03.1994)
Published in Bioorganic & medicinal chemistry letters (10.03.1994)
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Journal Article
α2-Adrenoceptors mediate clonicine-induced sedation in the rat
Drew, G.M., Gower, Alma J., Marriott, A.S.
Published in British journal of pharmacology (01.09.1979)
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Published in British journal of pharmacology (01.09.1979)
Journal Article
α2‐ADRENOCEPTORS MEDIATE CLONIDINE‐INDUCED SEDATION IN THE RAT
DREW, G.M., GOWER, ALMA J., MARRIOTT, A.S.
Published in British journal of pharmacology (01.09.1979)
Published in British journal of pharmacology (01.09.1979)
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Journal Article
C-linked pyrazole biaryl tetrazoles as antagonists of angiotensin II
Middlemiss, D., Ross, B.C., Eldred, C., Montana, J.G., Shah, P., Hirst, G.C., Watson, S.P., Panchal, T.A., Paton, J.M.S., Hubbard, T., Drew, G.M., Robertson, M.J., Hilditch, A., Clark, K.L.
Published in Bioorganic & medicinal chemistry letters (01.10.1992)
Published in Bioorganic & medicinal chemistry letters (01.10.1992)
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Journal Article
Benzofuran based angiotensin II antagonists related to GR117289: Part III; GR138950, a triflamide with high oral bioavailability
Dowle, M.D., Judd, D.B., Middlemiss, D., Scopes, D.I.C., Ross, B.C., Pass, M., Tranquillini, E., Jack, T.I., Hobson, J.E., Panchal, T.A., Stuart, P.G., Drew, G.M., Robertson, M.J., Hilditch, A., Clark, K.L., Travers, A., Hunt, A.A.E., Manchee, G.R., Walker, D.G., Eddershaw, P.J., Donnelly, M., Bayliss, M.K.
Published in Bioorganic & medicinal chemistry letters (1993)
Published in Bioorganic & medicinal chemistry letters (1993)
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Journal Article