Aryl amination using ligand-free Ni(II) salts and photoredox catalysis
Corcoran, Emily B., Pirnot, Michael T., Lin, Shishi, Dreher, Spencer D., DiRocco, Daniel A., Davies, Ian W., Buchwald, Stephen L., MacMillan, David W. C.
Published in Science (American Association for the Advancement of Science) (15.07.2016)
Published in Science (American Association for the Advancement of Science) (15.07.2016)
Get full text
Journal Article
The importance of synthetic chemistry in the pharmaceutical industry
Campos, Kevin R, Coleman, Paul J, Alvarez, Juan C, Dreher, Spencer D, Garbaccio, Robert M, Terrett, Nicholas K, Tillyer, Richard D, Truppo, Matthew D, Parmee, Emma R
Published in Science (American Association for the Advancement of Science) (18.01.2019)
Published in Science (American Association for the Advancement of Science) (18.01.2019)
Get full text
Journal Article
Response to Comment on "Predicting reaction performance in C-N cross-coupling using machine learning"
Estrada, Jesús G, Ahneman, Derek T, Sheridan, Robert P, Dreher, Spencer D, Doyle, Abigail G
Published in Science (American Association for the Advancement of Science) (16.11.2018)
Published in Science (American Association for the Advancement of Science) (16.11.2018)
Get full text
Journal Article
Nanomole-scale high-throughput chemistry for the synthesis of complex molecules
Santanilla, Alexander Buitrago, Regalado, Erik L., Pereira, Tony, Shevlin, Michael, Bateman, Kevin, Campeau, Louis-Charles, Schneeweis, Jonathan, Berritt, Simon, Shi, Zhi-Cai, Nantermet, Philippe, Liu, Yong, Helmy, Roy, Welch, Christopher J., Vachal, Petr, Davies, Ian W., Cernak, Tim, Dreher, Spencer D.
Published in Science (American Association for the Advancement of Science) (02.01.2015)
Published in Science (American Association for the Advancement of Science) (02.01.2015)
Get full text
Journal Article
Palladium-Catalyzed C(sp3)–H Arylation of Diarylmethanes at Room Temperature: Synthesis of Triarylmethanes via Deprotonative-Cross-Coupling Processes
Zhang, Jiadi, Bellomo, Ana, Creamer, Andrea D, Dreher, Spencer D, Walsh, Patrick J
Published in Journal of the American Chemical Society (22.08.2012)
Published in Journal of the American Chemical Society (22.08.2012)
Get full text
Journal Article
Chemistry informer libraries: a chemoinformatics enabled approach to evaluate and advance synthetic methods
Kutchukian, Peter S., Dropinski, James F., Dykstra, Kevin D., Li, Bing, DiRocco, Daniel A., Streckfuss, Eric C., Campeau, Louis-Charles, Cernak, Tim, Vachal, Petr, Davies, Ian W., Krska, Shane W., Dreher, Spencer D.
Published in Chemical science (Cambridge) (01.01.2016)
Published in Chemical science (Cambridge) (01.01.2016)
Get full text
Journal Article
NiXantphos: A Deprotonatable Ligand for Room-Temperature Palladium-Catalyzed Cross-Couplings of Aryl Chlorides
Zhang, Jiadi, Bellomo, Ana, Trongsiriwat, Nisalak, Jia, Tiezheng, Carroll, Patrick J, Dreher, Spencer D, Tudge, Matthew T, Yin, Haolin, Robinson, Jerome R, Schelter, Eric J, Walsh, Patrick J
Published in Journal of the American Chemical Society (30.04.2014)
Published in Journal of the American Chemical Society (30.04.2014)
Get full text
Journal Article
Palladium-Catalyzed Enantioselective Arylation of Aryl Sulfenate Anions: A Combined Experimental and Computational Study
Jia, Tiezheng, Zhang, Mengnan, McCollom, Samuel P, Bellomo, Ana, Montel, Sonia, Mao, Jianyou, Dreher, Spencer D, Welch, Christopher J, Regalado, Erik L, Williamson, R. Thomas, Manor, Brian C, Tomson, Neil C, Walsh, Patrick J
Published in Journal of the American Chemical Society (21.06.2017)
Published in Journal of the American Chemical Society (21.06.2017)
Get full text
Journal Article
P2Et Phosphazene: A Mild, Functional Group Tolerant Base for Soluble, Room Temperature Pd-Catalyzed C–N, C–O, and C–C Cross-Coupling Reactions
Buitrago Santanilla, Alexander, Christensen, Melodie, Campeau, Louis-Charles, Davies, Ian W, Dreher, Spencer D
Published in Organic letters (02.07.2015)
Published in Organic letters (02.07.2015)
Get full text
Journal Article
Synthesis of Complex Druglike Molecules by the Use of Highly Functionalized Bench-Stable Organozinc Reagents
Greshock, Thomas J., Moore, Keith P., McClain, Ray T., Bellomo, Ana, Chung, Cheol K., Dreher, Spencer D., Kutchukian, Peter S., Peng, Zhengwei, Davies, Ian W., Vachal, Petr, Ellwart, Mario, Manolikakes, Sophia M., Knochel, Paul, Nantermet, Philippe G.
Published in Angewandte Chemie (International ed.) (24.10.2016)
Published in Angewandte Chemie (International ed.) (24.10.2016)
Get full text
Journal Article
Frequency and spatial distribution of cartilage thickness change in knee osteoarthritis and its relation to clinical and radiographic covariates – data from the osteoarthritis initiative
Buck, R.J, Wirth, W, Dreher, D, Nevitt, M, Eckstein, F
Published in Osteoarthritis and cartilage (01.01.2013)
Published in Osteoarthritis and cartilage (01.01.2013)
Get full text
Journal Article