Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors
Brnardic, Edward J., Garbaccio, Robert M., Fraley, Mark E., Tasber, Edward S., Steen, Justin T., Arrington, Kenneth L., Dudkin, Vadim Y., Hartman, George D., Stirdivant, Steven M., Drakas, Bob A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Hardwick, James, Tao, Weikang, Beck, Stephen C., Mao, Xianzhi, Lobell, Robert B., Sepp-Lorenzino, Laura, Yan, Youwei, Ikuta, Mari, Munshi, Sanjeev K., Kuo, Lawrence C., Kreatsoulas, Constantine
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Journal Article
3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6
Fraley, Mark E., Steen, Justin T., Brnardic, Edward J., Arrington, Kenneth L., Spencer, Keith L., Hanney, Barbara A., Kim, Yuntae, Hartman, George D., Stirdivant, Steven M., Drakas, Bob A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Hardwick, James, Tao, Weikang, Beck, Stephen C., Mao, Xianzhi, Lobell, Robert B., Sepp-Lorenzino, Laura, Yan, Youwei, Ikuta, Mari, Munshi, Sanjeev K., Kuo, Lawrence C., Kreatsoulas, Constantine
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
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Journal Article
Optimization of a pyrazoloquinolinone class of Chkl kinase inhibitors
BRNARDIC, Edward J, GARBACCIO, Robert M, RICKERT, Keith, WALSH, Eileen S, HAMILTON, Kelly, BUSER, Carolyn A, HARDWICK, James, WEIKANG TAO, BECK, Stephen C, XIANZHI MAO, LOBELL, Robert B, SEPP-LORENZINO, Laura, FRALEY, Mark E, YOUWEI YAN, IKUTA, Mari, MUNSHI, Sanjeev K, KUO, Lawrence C, KREATSOULAS, Constantine, TASBER, Edward S, STEEN, Justin T, ARRINGTON, Kenneth L, DUDKIN, Vadim Y, HARTMAN, George D, STIRDIVANT, Steven M, DRAKAS, Bob A
Published in Bioorganic & medicinal chemistry letters (2007)
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Published in Bioorganic & medicinal chemistry letters (2007)
Journal Article