Search Results - "Drąg, Marcin" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery

Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery

by Kryštůfek, Robin, Šácha, Pavel, Starková, Jana, Brynda, Jiří, Hradilek, Martin, Tloušt’ová, Eva, Grzymska, Justyna, Rut, Wioletta, Boucher, Michael J, Drąg, Marcin, Majer, Pavel, Hájek, Miroslav, Řezáčová, Pavlína, Madhani, Hiten D, Craik, Charles S, Konvalinka, Jan
Published in Journal of medicinal chemistry (27.05.2021)

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SARS-CoV-2 Mpro inhibitors and activity-based probes for patient-sample imaging

SARS-CoV-2 Mpro inhibitors and activity-based probes for patient-sample imaging

by Rut, Wioletta, Groborz, Katarzyna, Zhang, Linlin, Sun, Xinyuanyuan, Zmudzinski, Mikolaj, Pawlik, Bartlomiej, Wang, Xinyu, Jochmans, Dirk, Neyts, Johan, Młynarski, Wojciech, Hilgenfeld, Rolf, Drag, Marcin
Published in Nature chemical biology (01.02.2021)

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α-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases

α-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases

by Drąg, Marcin, Grembecka, Jolanta, Pawełczak, Małgorzata, Kafarski, Paweł
Published in European journal of medicinal chemistry (01.08.2005)

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Synthesis of a HyCoSuL peptide substrate library to dissect protease substrate specificity

Synthesis of a HyCoSuL peptide substrate library to dissect protease substrate specificity

by Poreba, Marcin, Salvesen, Guy S, Drag, Marcin
Published in Nature protocols (01.10.2017)

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Caspase substrates and inhibitors

Caspase substrates and inhibitors

by Poreba, Marcin, Strózyk, Aleksandra, Salvesen, Guy S, Drag, Marcin
Published in Cold Spring Harbor perspectives in biology (01.08.2013)

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Imaging of proteases using activity-based probes

Imaging of proteases using activity-based probes

by Zmudzinski, Mikolaj, Malon, Oliwia, Poręba, Marcin, Drąg, Marcin
Published in Current opinion in chemical biology (01.06.2023)

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SUMO-mediated regulation of NLRP3 modulates inflammasome activity

SUMO-mediated regulation of NLRP3 modulates inflammasome activity

by Barry, Rachael, John, Sidonie Wicky, Liccardi, Gianmaria, Tenev, Tencho, Jaco, Isabel, Chen, Chih-Hong, Choi, Justin, Kasperkiewicz, Paulina, Fernandes-Alnemri, Teresa, Alnemri, Emad, Drag, Marcin, Chen, Yuan, Meier, Pascal
Published in Nature communications (01.08.2018)

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The Strategies to Support the COVID-19 Vaccination with Evidence-Based Communication and Tackling Misinformation

The Strategies to Support the COVID-19 Vaccination with Evidence-Based Communication and Tackling Misinformation

by Rzymski, Piotr, Borkowski, Leszek, Drąg, Marcin, Flisiak, Robert, Jemielity, Jacek, Krajewski, Jacek, Mastalerz-Migas, Agnieszka, Matyja, Andrzej, Pyrć, Krzysztof, Simon, Krzysztof, Sutkowski, Michał, Wysocki, Jacek, Zajkowska, Joanna, Fal, Andrzej
Published in Vaccines (Basel) (01.02.2021)

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Selective Substrates and Activity-Based Probes for Imaging of the Human Constitutive 20S Proteasome in Cells and Blood Samples

Selective Substrates and Activity-Based Probes for Imaging of the Human Constitutive 20S Proteasome in Cells and Blood Samples

by Rut, Wioletta, Poręba, Marcin, Kasperkiewicz, Paulina, Snipas, Scott J, Drąg, Marcin
Published in Journal of medicinal chemistry (28.06.2018)

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Fluorescent Activity-Based Probe To Image and Inhibit Factor XIa Activity in Human Plasma

Fluorescent Activity-Based Probe To Image and Inhibit Factor XIa Activity in Human Plasma

by Modrzycka, Sylwia, Kołt, Sonia, Adams, Ty E., Potoczek, Stanisław, Huntington, James A., Kasperkiewicz, Paulina, Drąg, Marcin
Published in Journal of medicinal chemistry (23.03.2023)

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Extended substrate specificity and first potent irreversible inhibitor/activity-based probe design for Zika virus NS2B-NS3 protease

Extended substrate specificity and first potent irreversible inhibitor/activity-based probe design for Zika virus NS2B-NS3 protease

by Rut, Wioletta, Zhang, Linlin, Kasperkiewicz, Paulina, Poreba, Marcin, Hilgenfeld, Rolf, Drąg, Marcin
Published in Antiviral research (01.03.2017)

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Activity profiling and crystal structures of inhibitor-bound SARS-CoV-2 papain-like protease: A framework for anti-COVID-19 drug design

Activity profiling and crystal structures of inhibitor-bound SARS-CoV-2 papain-like protease: A framework for anti-COVID-19 drug design

by Rut, Wioletta, Lv, Zongyang, Zmudzinski, Mikolaj, Patchett, Stephanie, Nayak, Digant, Snipas, Scott J, El Oualid, Farid, Huang, Tony T, Bekes, Miklos, Drag, Marcin, Olsen, Shaun K
Published in Science advances (16.10.2020)

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Green-Emitting 4,5-Diaminonaphthalimides in Activity-Based Probes for the Detection of Thrombin

Green-Emitting 4,5-Diaminonaphthalimides in Activity-Based Probes for the Detection of Thrombin

by Krzeszewski, Maciej, Modrzycka, Sylwia, Bousquet, Manon H. E., Jacquemin, Denis, Drąg, Marcin, Gryko, Daniel T.
Published in Organic letters (05.08.2022)

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Diagnostic and therapeutic potential of protease inhibition

Diagnostic and therapeutic potential of protease inhibition

by Ćwilichowska, Natalia, Świderska, Karolina W, Dobrzyń, Agnieszka, Drąg, Marcin, Poręba, Marcin
Published in Molecular aspects of medicine (01.12.2022)

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Substrate specificity profiling of heat-sensitive serine protease from the fungus Onygena corvina

Substrate specificity profiling of heat-sensitive serine protease from the fungus Onygena corvina

by Kasperkiewicz, Paulina, Kołt, Sonia, Janiszewski, Tomasz, Skowron, Piotr M., Krefft, Daria, Brodzik, Robert, Koller, Klaus-Peter, Drąg, Marcin
Published in Biochimie (01.11.2024)

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Investigation of osteoclast cathepsin K activity in osteoclastogenesis and bone loss using a set of chemical reagents

Investigation of osteoclast cathepsin K activity in osteoclastogenesis and bone loss using a set of chemical reagents

by Janiszewski, Tomasz, Kołt, Sonia, Ciastoń, Izabela, Vizovisek, Matej, Poręba, Marcin, Turk, Boris, Drąg, Marcin, Kozieł, Joanna, Kasperkiewicz, Paulina
Published in Cell chemical biology (16.02.2023)

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Leveraging Peptide Substrate Libraries to Design Inhibitors of Bacterial Lon Protease

Leveraging Peptide Substrate Libraries to Design Inhibitors of Bacterial Lon Protease

by Babin, Brett M, Kasperkiewicz, Paulina, Janiszewski, Tomasz, Yoo, Euna, Dra̧g, Marcin, Bogyo, Matthew
Published in ACS chemical biology (15.11.2019)

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Exploring the prime site in caspases as a novel chemical strategy for understanding the mechanisms of cell death: a proof of concept study on necroptosis in cancer cells

Exploring the prime site in caspases as a novel chemical strategy for understanding the mechanisms of cell death: a proof of concept study on necroptosis in cancer cells

by Groborz, Katarzyna, Gonzalez Ramirez, Monica L., Snipas, Scott J., Salvesen, Guy S., Drąg, Marcin, Poręba, Marcin
Published in Cell death and differentiation (01.02.2020)

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Potent and selective caspase-2 inhibitor prevents MDM-2 cleavage in reversine-treated colon cancer cells

Potent and selective caspase-2 inhibitor prevents MDM-2 cleavage in reversine-treated colon cancer cells

by Poreba, Marcin, Rut, Wioletta, Groborz, Katarzyna, Snipas, Scott J., Salvesen, Guy S., Drag, Marcin
Published in Cell death and differentiation (01.12.2019)

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Noninvasive optical detection of granzyme B from natural killer cells with enzyme-activated fluorogenic probes

Noninvasive optical detection of granzyme B from natural killer cells with enzyme-activated fluorogenic probes

by Janiszewski, Tomasz, Kołt, Sonia, Kaiserman, Dion, Snipas, Scott J., Li, Shuang, Kulbacka, Julita, Saczko, Jolanta, Bovenschen, Niels, Salvesen, Guy, Drąg, Marcin, Bird, Phillip I., Kasperkiewicz, Paulina
Published in The Journal of biological chemistry (10.07.2020)

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