Biochemical and pharmacological characterization of AZD1981, an orally available selective DP2 antagonist in clinical development for asthma
Schmidt, JA, Bell, FM, Akam, E, Marshall, C, Dainty, IA, Heinemann, A, Dougall, IG, Bonnert, RV, Sargent, CA
Published in British journal of pharmacology (01.04.2013)
Published in British journal of pharmacology (01.04.2013)
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Biochemical and pharmacological characterization of AZD 1981, an orally available selective DP 2 antagonist in clinical development for asthma
Schmidt, JA, Bell, FM, Akam, E, Marshall, C, Dainty, IA, Heinemann, A, Dougall, IG, Bonnert, RV, Sargent, CA
Published in British journal of pharmacology (01.04.2013)
Published in British journal of pharmacology (01.04.2013)
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Journal Article
Lead Generation Using Pharmacophore Mapping and Three-Dimensional Database Searching: Application to Muscarinic M 3 Receptor Antagonists
Marriott, David P., Dougall, Iain G., Meghani, Premji, Liu, Yu-Jiang, Flower, Darren R.
Published in Journal of medicinal chemistry (26.08.1999)
Published in Journal of medicinal chemistry (26.08.1999)
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Further concerns over Cheng-Prusoff analysis
Leff, Paul, Dougall, Iain G.
Published in Trends in pharmacological sciences (Regular ed.) (01.04.1993)
Published in Trends in pharmacological sciences (Regular ed.) (01.04.1993)
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Dual D-2-receptor and beta(2)-adrenoceptor agonists for the treatment of airway diseases. 1. Discovery and biological evaluation of some 7-(2-aminoethyl)-4-hydroxybenzothiazol-2(3H)-one analogues
Bonnert, RV, Brown, RC, Chapman, D, Cheshire, DR, Dixon, J, Ince, F, Kinchin, EC, Lyons, AJ, Davis, AM, Hallam, C, Harper, ST, Unitt, JF, Dougall, IG, Jackson, DM, McKechnie, K, Young, A, Simpson, WT
Published in Journal of medicinal chemistry (03.12.1998)
Published in Journal of medicinal chemistry (03.12.1998)
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Estimation of the efficacy and affinity of the beta 2-adrenoceptor agonist salmeterol in guinea-pig trachea
Dougall, I G, Harper, D, Jackson, D M, Leff, P
Published in British journal of pharmacology (01.12.1991)
Published in British journal of pharmacology (01.12.1991)
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Adventures in the pharmacological analysis of P2 receptors
Fagura, Malbinder S., Jarvis, Gavin E., Dougall, Iain G., Leff, Paul
Published in Journal of the autonomic nervous system (03.07.2000)
Published in Journal of the autonomic nervous system (03.07.2000)
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