Parallel Functional Activity Profiling Reveals Valvulopathogens Are Potent 5-Hydroxytryptamine2B Receptor Agonists: Implications for Drug Safety Assessment
Huang, Xi-Ping, Setola, Vincent, Yadav, Prem N., Allen, John A., Rogan, Sarah C., Hanson, Bonnie J., Revankar, Chetana, Robers, Matt, Doucette, Chris, Roth, Bryan L.
Published in Molecular pharmacology (01.10.2009)
Published in Molecular pharmacology (01.10.2009)
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Journal Article
A Homogeneous Fluorescent Live-Cell Assay for Measuring 7-Transmembrane Receptor Activity and Agonist Functional Selectivity Through Beta-Arrestin Recruitment
Hanson, Bonnie J., Wetter, Justin, Bercher, Mark R., Kopp, Leisha, Fuerstenau-Sharp, Maya, Vedvik, Kevin L., Zielinski, Thomas, Doucette, Chris, Whitney, Pamela J., Revankar, Chetana
Published in Journal of biomolecular screening (01.08.2009)
Published in Journal of biomolecular screening (01.08.2009)
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Journal Article
Parallel functional activity profiling reveals valvulopathogens are potent 5-hydroxytryptamine(2B) receptor agonists: implications for drug safety assessment
Huang, Xi-Ping, Setola, Vincent, Yadav, Prem N, Allen, John A, Rogan, Sarah C, Hanson, Bonnie J, Revankar, Chetana, Robers, Matt, Doucette, Chris, Roth, Bryan L
Published in Molecular pharmacology (01.10.2009)
Published in Molecular pharmacology (01.10.2009)
Get full text
Journal Article