Synthesis and biological activity of 5-aryl-4-(4-(5-methyl-1H-imidazol-4-yl)piperidin-1-yl)pyrimidine analogs as potent, highly selective, and orally bioavailable NHE-1 inhibitors
Atwal, Karnail S., O’Neil, Steven V., Ahmad, Saleem, Doweyko, Lidia, Kirby, Mark, Dorso, Charles R., Chandrasena, Gamini, Chen, Bang-Chi, Zhao, Rulin, Zahler, Robert
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
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Arylcyclopropanecarboxyl Guanidines as Novel, Potent, and Selective Inhibitors of the Sodium Hydrogen Exchanger Isoform-1
Ahmad, Saleem, Doweyko, Lidia M, Dugar, Sundeep, Grazier, Nyeemah, Ngu, Khehyong, Wu, Shung C, Yost, Kenneth J, Chen, Bang-Chi, Gougoutas, Jack Z, DiMarco, John D, Lan, Shih-Jung, Gavin, Brian J, Chen, Alice Y, Dorso, Charles R, Serafino, Randy, Kirby, Mark, Atwal, Karnail S
Published in Journal of medicinal chemistry (27.09.2001)
Published in Journal of medicinal chemistry (27.09.2001)
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Aminoimidazoles as bioisosteres of acylguanidines: novel, potent, selective and orally bioavailable inhibitors of the sodium hydrogen exchanger isoform-1
Ahmad, Saleem, Ngu, Khehyong, Combs, Donald W, Wu, Shung C, Weinstein, David S, Liu, Wen, Chen, Bang-Chi, Chandrasena, Gamini, Dorso, Charles R, Kirby, Mark, Atwal, Karnail S
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
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Renal and depressor effects of SQ 29,072, a neutral endopeptidase inhibitor, in conscious hypertensive rats
Seymour, A A, Norman, J A, Asaad, M M, Fennell, S A, Swerdel, J N, Little, D K, Dorso, C R
Published in Journal of cardiovascular pharmacology (01.07.1990)
Published in Journal of cardiovascular pharmacology (01.07.1990)
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Proarrhythmic Effects of Pinacidil are Partially Mediated Through Enhancement of Catecholamine Release in Isolated Perfused Guinea-pig Hearts
D'Alonzo, Albert J., Zhu, Jia L., Darbenzio, Raymond B., Dorso, Charles R., Grover, Gary J.
Published in Journal of molecular and cellular cardiology (01.02.1998)
Published in Journal of molecular and cellular cardiology (01.02.1998)
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Renal abnormalities in mutant mice
Carpenter, Charles, Honkanen, Anita A, Mashimo, Hiroshi, Goss, Kendrick A, Huang, Paul, Fishman, Mark C, Asaad, Magdi, Dorso, Charles R, Cheung, Hong-son
Published in Nature (London) (28.03.1996)
Published in Nature (London) (28.03.1996)
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Renal and depressor activities of inhibitors of neutral endopeptidase and angiotensin converting enzyme in monkeys infused with angiotensin II
Seymour, A A, Asaad, M M, Abboa-Offei, B E, Smith, P L, Mathers, P D, Rogers, W L, Dorso, C R
Published in Journal of cardiovascular pharmacology (01.11.1996)
Published in Journal of cardiovascular pharmacology (01.11.1996)
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Determinants of in vivo activity of neutral endopeptidase 3.4.24.11 and angiotensin converting enzyme inhibitors
Seymour, A A, Asaad, M M, Abboa-Offei, B E, Smith, P L, Rogers, W L, Dorso, C R
Published in The Journal of pharmacology and experimental therapeutics (01.02.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.1996)
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Stability of plasma atrial natriuretic peptide after storage / Reply
Asaad, Magdi M, Dorso, Charles R, Rogers, W Lynn, Nelesen, Richard A
Published in Circulation (New York, N.Y.) (01.05.1994)
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Published in Circulation (New York, N.Y.) (01.05.1994)
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The effects of novel cathepsin E inhibitors on the big endothelin pressor response in conscious rats
Bird, J. Eileen, Waldron, Thomas L., Little, Deborah K., Asaad, Magdi M., Dorso, Charles R., DiDonato, Gerald, Norman, Jon A.
Published in Biochemical and biophysical research communications (15.01.1992)
Published in Biochemical and biophysical research communications (15.01.1992)
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