Tryptophan 2,3-Dioxygenase (TDO) Inhibitors. 3-(2-(Pyridyl)ethenyl)indoles as Potential Anticancer Immunomodulators
Dolušić, Eduard, Larrieu, Pierre, Moineaux, Laurence, Stroobant, Vincent, Pilotte, Luc, Colau, Didier, Pochet, Lionel, Van den Eynde, Benoît, Masereel, Bernard, Wouters, Johan, Frédérick, Raphaël
Published in Journal of medicinal chemistry (11.08.2011)
Published in Journal of medicinal chemistry (11.08.2011)
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Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase
Pilotte, Luc, Larrieu, Pierre, Stroobant, Vincent, Colau, Didier, Dolušić, Eduard, Frédérick, Raphaël, De Plaen, Etienne, Uyttenhove, Catherine, Wouters, Johan, Masereel, Bernard, Van den Eynde, Benoît J
Published in Proceedings of the National Academy of Sciences - PNAS (14.02.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (14.02.2012)
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Journal Article
Synthesis, evaluation and structure-activity relationship of new 3-carboxamide coumarins as FXIIa inhibitors
Bouckaert, Charlotte, Serra, Silvia, Rondelet, Grégoire, Dolušić, Eduard, Wouters, Johan, Dogné, Jean-Michel, Frédérick, Raphaël, Pochet, Lionel
Published in European journal of medicinal chemistry (03.03.2016)
Published in European journal of medicinal chemistry (03.03.2016)
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Convenient one-pot formation of highly functionalized 5-bromo-2-aminothiazoles, potential endocannabinoid hydrolase MAGL inhibitors
Prevost, Julien R.C., Kozlova, Arina, Es Saadi, Bouazza, Yildiz, Esra, Modaffari, Sara, Lambert, Didier M., Pochet, Lionel, Wouters, Johan, Dolušić, Eduard, Frédérick, Raphaël
Published in Tetrahedron letters (05.12.2018)
Published in Tetrahedron letters (05.12.2018)
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Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors
Dolušić, Eduard, Larrieu, Pierre, Blanc, Sébastien, Sapunaric, Frédéric, Pouyez, Jenny, Moineaux, Laurence, Colette, Delphine, Stroobant, Vincent, Pilotte, Luc, Colau, Didier, Ferain, Thierry, Fraser, Graeme, Galleni, Moreno, Frère, Jean-Marie, Masereel, Bernard, Van den Eynde, Benoît, Wouters, Johan, Frédérick, Raphaël
Published in European journal of medicinal chemistry (01.07.2011)
Published in European journal of medicinal chemistry (01.07.2011)
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Gold Electrode Incorporating Corrole as an Ion-Channel Mimetic Sensor for Determination of Dopamine
Kurzatkowska, Katarzyna, Dolusic, Eduard, Dehaen, Wim, Sieroń-Stołtny, Karolina, Sieroń, Aleksander, Radecka, Hanna
Published in Analytical chemistry (Washington) (01.09.2009)
Published in Analytical chemistry (Washington) (01.09.2009)
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Efficient synthesis of aryldipyrromethanes in water and their application in the synthesis of corroles and dipyrromethenes
Rohand, Taoufik, Dolusic, Eduard, Ngo, Thien H., Maes, Wouter, Dehaen, Wim
Published in ARKIVOC (28.04.2007)
Published in ARKIVOC (28.04.2007)
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Indoleamine 2,3-dioxygenase inhibitory activity of derivatives of marine alkaloid tsitsikammamine A
Dolušić, Eduard, Larrieu, Pierre, Meinguet, Céline, Colette, Delphine, Rives, Arnaud, Blanc, Sébastien, Ferain, Thierry, Pilotte, Luc, Stroobant, Vincent, Wouters, Johan, Van den Eynde, Benoît, Masereel, Bernard, Delfourne, Evelyne, Frédérick, Raphaël
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
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Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors
Dolušić, Eduard, Larrieu, Pierre, Blanc, Sébastien, Sapunaric, Frédéric, Norberg, Bernadette, Moineaux, Laurence, Colette, Delphine, Stroobant, Vincent, Pilotte, Luc, Colau, Didier, Ferain, Thierry, Fraser, Graeme, Galeni, Moreno, Frère, Jean-Marie, Masereel, Bernard, Van den Eynde, Benoît, Wouters, Johan, Frédérick, Raphaël
Published in Bioorganic & medicinal chemistry (15.02.2011)
Published in Bioorganic & medicinal chemistry (15.02.2011)
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Synthesis, crystal structures and electronic properties of isomers of chloro-pyridinylvinyl-1H-indoles
Moineaux, Laurence, Laurent, Sophie, Reniers, Jérémy, Dolušić, Eduard, Galleni, Moreno, Frère, Jean-Marie, Masereel, Bernard, Frédérick, Raphaël, Wouters, Johan
Published in European journal of medicinal chemistry (01.08.2012)
Published in European journal of medicinal chemistry (01.08.2012)
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Corrigendum to “Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors” [Bioorg. Med. Chem. (2011) 1550–1561]
Dolušić, Eduard, Larrieu, Pierre, Blanc, Sébastien, Sapunaric, Frédéric, Norberg, Bernadette, Moineaux, Laurence, Colette, Delphine, Stroobant, Vincent, Pilotte, Luc, Colau, Didier, Ferain, Thierry, Fraser, Graeme, Galleni, Moreno, Frère, Jean-Marie, Masereel, Bernard, Eynde, Benoît Van den, Wouters, Johan, Frédérick, Raphaël
Published in Bioorganic & medicinal chemistry (01.05.2011)
Published in Bioorganic & medicinal chemistry (01.05.2011)
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Journal Article
Auxin activity and molecular structure of 2-alkylindole-3-acetic acids
ANTOLIC, Snjezana, DOLUSIC, Eduard, KOZIC, Erika K, KOJIC-PRODIC, Biserka, MAGNUS, Volker, RAMEK, Michael, TOMIC, Sanja
Published in Plant growth regulation (01.03.2003)
Published in Plant growth regulation (01.03.2003)
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Journal Article
Biotinylated Indoles as Probes for Indole-Binding Proteins
Dolušić, Eduard, Kowalczyk, Mariusz, Magnus, Volker, Sandberg, Göran, Normanly, Jennifer
Published in Bioconjugate chemistry (01.03.2001)
Published in Bioconjugate chemistry (01.03.2001)
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PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR MEDICAL TREATMENT
GAO LING-JIE, PFLEIDERER WOLFGANG, DOLUSIC EDUARD, HERDEWIJN PIET, DE JONGHE STEVEN
Year of Publication 22.10.2009
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Year of Publication 22.10.2009
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