Discovery of a benzimidazole-based dual FLT3/TrKA inhibitor targeting acute myeloid leukemia
Dokla, Eman M.E., Abdel-Aziz, Amal Kamal, Milik, Sandra N., McPhillie, Martin J., Minucci, Saverio, Abouzid, Khaled A.M.
Published in Bioorganic & medicinal chemistry (15.02.2022)
Published in Bioorganic & medicinal chemistry (15.02.2022)
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Journal Article
Development of benzimidazole-based derivatives as antimicrobial agents and their synergistic effect with colistin against gram-negative bacteria
Dokla, Eman M.E., Abutaleb, Nader S., Milik, Sandra N., Li, Daoyi, El-Baz, Karim, Shalaby, Menna-Allah W., Al-Karaki, Rawan, Nasr, Maha, Klein, Christian D., Abouzid, Khaled A.M., Seleem, Mohamed N.
Published in European journal of medicinal chemistry (15.01.2020)
Published in European journal of medicinal chemistry (15.01.2020)
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Journal Article
FLT3-PROTACs for combating AML resistance: Analytical overview on chimeric agents developed, challenges, and future perspectives
Hesham, Heba M., Dokla, Eman M.E., Elrazaz, Eman Z., Lasheen, Deena S., Abou El Ella, Dalal A.
Published in European journal of medicinal chemistry (05.11.2024)
Published in European journal of medicinal chemistry (05.11.2024)
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Journal Article
SAR investigation and optimization of benzimidazole-based derivatives as antimicrobial agents against Gram-negative bacteria
Dokla, Eman M.E., Abutaleb, Nader S., Milik, Sandra N., Kandil, Ezzat A.E.A., Qassem, Omar M., Elgammal, Yehia, Nasr, Maha, McPhillie, Martin J., Abouzid, Khaled A.M., Seleem, Mohamed N., Imming, Peter, Adel, Mai
Published in European journal of medicinal chemistry (05.02.2023)
Published in European journal of medicinal chemistry (05.02.2023)
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Journal Article
Novel sulfonamide-indolinone hybrids targeting mitochondrial respiration of breast cancer cells
Helmy, Sama W.A., Abdel-Aziz, Amal Kamal, Dokla, Eman M.E., Ahmed, Tarek E., Hatem, Yasmin, Abdel Rahman, Engy A., Sharaky, Marwa, Shahin, Mai I., Elrazaz, Eman Z., Serya, Rabah A.T., Henary, Maged, Ali, Sameh S., Abou El Ella, Dalal A.
Published in European journal of medicinal chemistry (15.03.2024)
Published in European journal of medicinal chemistry (15.03.2024)
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Journal Article
Nanoemulgel formulation of a benzimidazole derivative for wound healing
Dokla, Eman M.E., El-Gogary, Riham I., Abd-Elsaid, Nada M., Gad, Mariam, Abd-Elhalim, Reem K., Habib, Hana H., Eldeeb, Wesam, Eldahshan, Esraa R., Nassar, Salma H., Issa, Aya N., Rabeh, Neveen, Abd-Elkhalik, Samar, Nasr, Maha
Published in Journal of drug delivery science and technology (01.12.2023)
Published in Journal of drug delivery science and technology (01.12.2023)
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Journal Article
Indolin-2-one derivatives as selective Aurora B kinase inhibitors targeting breast cancer
Dokla, Eman M.E., Abdel-Aziz, Amal Kamal, Milik, Sandra N., Mahmoud, Amr H., Saadeldin, Mona Kamal, McPhillie, Martin J., Minucci, Saverio, Abouzid, Khaled A.M.
Published in Bioorganic chemistry (01.12.2021)
Published in Bioorganic chemistry (01.12.2021)
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Journal Article
Targeting YAP Degradation by a Novel 1,2,4-Oxadiazole Derivative via Restoration of the Function of the Hippo Pathway
Dokla, Eman M. E, Fang, Chun-Sheng, Chu, Po-Chen, Chang, Chih-Shiang, Abouzid, Khaled A. M, Chen, Ching S
Published in ACS medicinal chemistry letters (09.04.2020)
Published in ACS medicinal chemistry letters (09.04.2020)
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Journal Article
A 5′ AMP‐Activated Protein Kinase Enzyme Activator, Compound 59, Induces Autophagy and Apoptosis in Human Oral Squamous Cell Carcinoma
Weng, Jing‐Ru, Dokla, Eman M. E., Bai, Li‐Yuan, Chen, Ching‐Shih, Chiu, Shih‐Jiuan, Shieh, Tzong‐Ming
Published in Basic & clinical pharmacology & toxicology (01.07.2018)
Published in Basic & clinical pharmacology & toxicology (01.07.2018)
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Journal Article
Identification of novel pyrazole and benzimidazole based derivatives as PBP2a inhibitors: Design, synthesis, and biological evaluation
Shalaby, Menna-Allah, Dokla, Eman, Serya, Rabah, Abouzid, Khaled
Published in Archives of Pharmaceutical Sciences Ain Shams University (01.12.2019)
Published in Archives of Pharmaceutical Sciences Ain Shams University (01.12.2019)
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Journal Article
Development of Potent Adenosine Monophosphate Activated Protein Kinase (AMPK) Activators
Dokla, Eman M. E., Fang, Chun-Sheng, Lai, Po-Ting, Kulp, Samuel K., Serya, Rabah A. T., Ismail, Nasser S. M., Abouzid, Khaled A. M., Chen, Ching-Shih
Published in ChemMedChem (01.11.2015)
Published in ChemMedChem (01.11.2015)
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