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Jiang, Yutong, Andrews, Steven W., Condroski, Kevin R., Buckman, Brad, Serebryany, Vlad, Wenglowsky, Steve, Kennedy, April L., Madduru, Machender R., Wang, Bin, Lyon, Michael, Doherty, George A., Woodard, Benjamin T., Lemieux, Christine, Do, Mary Geck, Zhang, Hailong, Ballard, Joshua, Vigers, Guy, Brandhuber, Barbra J., Stengel, Peter, Josey, John A., Beigelman, Leonid, Blatt, Lawrence, Seiwert, Scott D.
Published in Journal of medicinal chemistry (13.03.2014)
Published in Journal of medicinal chemistry (13.03.2014)
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SAR and characterization of non-substrate isoindoline urea inhibitors of nicotinamide phosphoribosyltransferase (NAMPT)
Curtin, Michael L., Heyman, H. Robin, Clark, Richard F., Sorensen, Bryan K., Doherty, George A., Hansen, T. Matthew, Frey, Robin R., Sarris, Kathy A., Aguirre, Ana L., Shrestha, Anurupa, Tu, Noah, Woller, Kevin, Pliushchev, Marina A., Sweis, Ramzi F., Cheng, Min, Wilsbacher, Julie L., Kovar, Peter J., Guo, Jun, Cheng, Dong, Longenecker, Kenton L., Raich, Diana, Korepanova, Alla V., Soni, Nirupama B., Algire, Mikkel A., Richardson, Paul L., Marin, Violeta L., Badagnani, Ilaria, Vasudevan, Anil, Buchanan, F. Greg, Maag, David, Chiang, Gary G., Tse, Chris, Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
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Discovery of A‑1331852, a First-in-Class, Potent, and Orally-Bioavailable BCL‑XL Inhibitor
Wang, Le, Doherty, George A, Judd, Andrew S, Tao, Zhi-Fu, Hansen, T. Matthew, Frey, Robin R, Song, Xiaohong, Bruncko, Milan, Kunzer, Aaron R, Wang, Xilu, Wendt, Michael D, Flygare, John A, Catron, Nathaniel D, Judge, Russell A, Park, Chang H, Shekhar, Shashank, Phillips, Darren C, Nimmer, Paul, Smith, Morey L, Tahir, Stephen K, Xiao, Yu, Xue, John, Zhang, Haichao, Le, Phuong N, Mitten, Michael J, Boghaert, Erwin R, Gao, Wenqing, Kovar, Peter, Choo, Edna F, Diaz, Dolores, Fairbrother, Wayne J, Elmore, Steven W, Sampath, Deepak, Leverson, Joel D, Souers, Andrew James
Published in ACS medicinal chemistry letters (08.10.2020)
Published in ACS medicinal chemistry letters (08.10.2020)
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Discovery of diphenyl lactam derivatives as N-type calcium channel blockers
Doherty, George A., Bhatia, Pramila, Vortherms, Timothy A., Marsh, Kennan C., Wetter, Jill M., Mack, Helmut, Scott, Victoria E., Jarvis, Michael F., Stewart, Andrew O.
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
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항-C-MET 항체 약물 접합체
BOGHAERT ERWIN R, PHILLIPS ANDREW C, JI CHENG, ANDERSON MARK, DOHERTY GEORGE A, REILLY REGINA M, BRUNCKO MILAN
Year of Publication 11.01.2024
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Year of Publication 11.01.2024
Patent
N-Tetrahydrofuroyl-( l)-phenylalanine derivatives as potent VLA-4 antagonists
Yang, Ginger X., Chang, Linda L., Truong, Quang, Doherty, George A., Magriotis, Plato A., de Laszlo, Stephen E., Li, Bing, MacCoss, Malcolm, Kidambi, Usha, Egger, Linda A., McCauley, Ermengilda, Van Riper, Gail, Mumford, Richard A., Schmidt, John A., Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (03.06.2002)
Published in Bioorganic & medicinal chemistry letters (03.06.2002)
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N-Isonicotinoyl-( l)-4-aminophenylalanine derivatives as tight binding VLA-4 antagonists
Doherty, George A., Yang, Ginger X., Borges, Edite, Tong, Sharon, McCauley, Ermengilda D., Treonz, Kelly M., Van Riper, Gail, Pacholok, Stephen, Si, Qian, Koo, Gloria C., Shah, Kashmira, Mumford, Richard A., Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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Substituted tetrahydrofuroyl-1-phenylalanine derivatives as potent and specific VLA-4 antagonists
Doherty, George A., Yang, Ginger X., Borges, Edite, Chang, Linda L., MacCoss, Malcolm, Tong, Sharon, Kidambi, Usha, Egger, Linda A., McCauley, Ermenegilda, Van Riper, Gail, Mumford, Richard A., Schmidt, John A., Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (03.06.2002)
Published in Bioorganic & medicinal chemistry letters (03.06.2002)
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Discovery of A-1331852, a First-in-Class, Potent, and Orally-Bioavailable BCL-X-L Inhibitor
Wang, Le, Doherty, George A., Judd, Andrew S., Tao, Zhi-Fu, Hansen, T. Matthew, Frey, Robin R., Song, Xiaohong, Bruncko, Milan, Kunzer, Aaron R., Wang, Xilu, Wendt, Michael D., Flygare, John A., Catron, Nathaniel D., Judge, Russell A., Park, Chang H., Shekhar, Shashank, Phillips, Darren C., Nimmer, Paul, Smith, Morey L., Tahir, Stephen K., Xiao, Yu, Xue, John, Zhang, Haichao, Le, Phuong N., Mitten, Michael J., Boghaert, Erwin R., Gao, Wenqing, Kovar, Peter, Choo, Edna F., Diaz, Dolores, Fairbrother, Wayne J., Elmore, Steven W., Sampath, Deepak, Leverson, Joel D., Souers, Andrew James
Published in ACS medicinal chemistry letters (08.10.2020)
Published in ACS medicinal chemistry letters (08.10.2020)
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Sulfonamide derivatives as Bcl-2-selective apoptosis-inducing agents for the treatment of cancer and immune diseases
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, WANG LE, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA, KUNZER AARON R
Year of Publication 18.01.2017
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Year of Publication 18.01.2017
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Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, WANG LE, DAI YUJIA, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA, KUNZER AARON R
Year of Publication 07.12.2016
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Year of Publication 07.12.2016
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6-SUBSTITUTED PHENOXYCHROMAN CARBOXYLIC ACID DERIVATIVES
KIM GANGHYEOK, CLARK CHRISTOPHER T, DOHERTY GEORGE A, ROMOFF TODD, BURGESS LAURENCE E, DELISLE ROBERT KIRK, CORRETTE CHRISTOPHER P, COOK ADAM, HUNT KEVIN W
Year of Publication 16.03.2011
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Year of Publication 16.03.2011
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APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, HANSEN TODD M, WANG LE, DAI YUJIA, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, KUNZER AARON, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA
Year of Publication 09.04.2013
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Year of Publication 09.04.2013
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SULFONAMIDE DERIVATIVES AS BCL-2-SELECTIVE APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE DISEASES
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, HANSEN TODD M, WANG LE, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, KUNZER AARON, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA
Year of Publication 12.12.2012
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Year of Publication 12.12.2012
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SULFONAMIDE DERIVATIVES AS BCL-2-SELECTIVE APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE DISEASES
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, WANG LE, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA, KUNZER AARON R
Year of Publication 20.09.2011
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Year of Publication 20.09.2011
Patent
APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES
MANTEI ROBERT A, WANG GARY T, PARK CHANG H, HASVOLD LISA, PARK, CHEOL MIN, WANG LE, DAI YUJIA, SONG XIAOHONG, ELMORE STEVEN W, BRUNCKO MILAN, SULLIVAN GERARD M, SOUERS ANDREW J, WANG XILU, MCCLELLAN WILLIAM J, TAO ZHI FU, PETROS ANDREW M, WENDT MICHAEL D, DOHERTY GEORGE A, DING HONG, HEXAMER LAURA, KUNZER AARON R
Year of Publication 05.09.2011
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Year of Publication 05.09.2011
Patent