Structural and Atropisomeric Factors Governing the Selectivity of Pyrimido-benzodiazipinones as Inhibitors of Kinases and Bromodomains
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Published in ACS chemical biology (21.09.2018)
Published in ACS chemical biology (21.09.2018)
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ERK5 Inhibition Induces Autophagy-Mediated Cancer Cell Death by Activating ER Stress
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Published in Frontiers in cell and developmental biology (04.11.2021)
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Abstract 1234: The anticancer drug ABTL0812 induces cancer cell death by impairing Akt/mTORC1 axis and inducing ER stress-mediated cytotoxic autophagy
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Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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The anti-cancer drug ABTL0812 induces ER stress-mediated cytotoxic autophagy by increasing dihydroceramide levels in cancer cells
Muñoz-Guardiola, Pau, Casas, Josefina, Megías-Roda, Elisabet, Solé, Sònia, Perez-Montoyo, Héctor, Yeste-Velasco, Marc, Erazo, Tatiana, Diéguez-Martínez, Nora, Espinosa-Gil, Sergio, Muñoz-Pinedo, Cristina, Yoldi, Guillermo, Abad, Jose L, Segura, Miguel F, Moran, Teresa, Romeo, Margarita, Bosch-Barrera, Joaquim, Oaknin, Ana, Alfón, Jose, Domènech, Carles, Fabriàs, Gemma, Velasco, Guillermo, Lizcano, Jose M
Published in Autophagy (03.06.2021)
Published in Autophagy (03.06.2021)
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The ERK5/NF-κB signaling pathway targets endometrial cancer proliferation and survival
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Published in Cellular and molecular life sciences : CMLS (01.10.2022)
Published in Cellular and molecular life sciences : CMLS (01.10.2022)
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Discovery of a selective inhibitor of doublecortin like kinase 1
Ferguson, Fleur M., Nabet, Behnam, Raghavan, Srivatsan, Liu, Yan, Leggett, Alan L., Kuljanin, Miljan, Kalekar, Radha L., Yang, Annan, He, Shuning, Wang, Jinhua, Ng, Raymond W. S., Sulahian, Rita, Li, Lianbo, Poulin, Emily J., Huang, Ling, Koren, Jost, Dieguez-Martinez, Nora, Espinosa, Sergio, Zeng, Zhiyang, Corona, Cesear R., Vasta, James D., Ohi, Ryoma, Sim, Taebo, Kim, Nam Doo, Harshbarger, Wayne, Lizcano, Jose M., Robers, Matthew B., Muthaswamy, Senthil, Lin, Charles Y., Look, A. Thomas, Haigis, Kevin M., Mancias, Joseph D., Wolpin, Brian M., Aguirre, Andrew J., Hahn, William C., Westover, Kenneth D., Gray, Nathanael S.
Published in Nature chemical biology (01.06.2020)
Published in Nature chemical biology (01.06.2020)
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An ERK5-KLF2 signalling module regulates early embryonic gene expression and telomere rejuvenation in stem cells
Brown, Helen A, Williams, Charles A C, Zhou, Houjiang, Rios-Szwed, Diana, Fernandez-Alonso, Rosalia, Mansoor, Saria, McMulkin, Liam, Toth, Rachel, Gourlay, Robert, Peltier, Julien, Dieguez-Martinez, Nora, Trost, Matthias, Lizcano, Jose M, Stavridis, Marios P, Findlay, Greg M
Published in Biochemical journal (10.12.2021)
Published in Biochemical journal (10.12.2021)
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The ERK5/NF-κB signaling pathway targets endometrial cancer proliferation and survival
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Published in bioRxiv (31.05.2022)
Published in bioRxiv (31.05.2022)
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An ERK5-KLF2 signalling module regulates early embryonic gene expression dynamics and stem cell rejuvenation
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Published in bioRxiv (29.03.2021)
Published in bioRxiv (29.03.2021)
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