A New DREADD Facilitates the Multiplexed Chemogenetic Interrogation of Behavior
Vardy, Eyal, Robinson, J. Elliott, Li, Chia, Olsen, Reid H.J., DiBerto, Jeffrey F., Giguere, Patrick M., Sassano, Flori M., Huang, Xi-Ping, Zhu, Hu, Urban, Daniel J., White, Kate L., Rittiner, Joseph E., Crowley, Nicole A., Pleil, Kristen E., Mazzone, Christopher M., Mosier, Philip D., Song, Juan, Kash, Thomas L., Malanga, C.J., Krashes, Michael J., Roth, Bryan L.
Published in Neuron (Cambridge, Mass.) (20.05.2015)
Published in Neuron (Cambridge, Mass.) (20.05.2015)
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Deschloroclozapine, a potent and selective chemogenetic actuator enables rapid neuronal and behavioral modulations in mice and monkeys
Nagai, Yuji, Miyakawa, Naohisa, Takuwa, Hiroyuki, Hori, Yukiko, Oyama, Kei, Ji, Bin, Takahashi, Manami, Huang, Xi-Ping, Slocum, Samuel T, DiBerto, Jeffrey F, Xiong, Yan, Urushihata, Takuya, Hirabayashi, Toshiyuki, Fujimoto, Atsushi, Mimura, Koki, English, Justin G, Liu, Jing, Inoue, Ken-Ichi, Kumata, Katsushi, Seki, Chie, Ono, Maiko, Shimojo, Masafumi, Zhang, Ming-Rong, Tomita, Yutaka, Nakahara, Jin, Suhara, Tetsuya, Takada, Masahiko, Higuchi, Makoto, Jin, Jian, Roth, Bryan L, Minamimoto, Takafumi
Published in Nature neuroscience (01.09.2020)
Published in Nature neuroscience (01.09.2020)
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Journal Article
TRUPATH, an open-source biosensor platform for interrogating the GPCR transducerome
Olsen, Reid H J, DiBerto, Jeffrey F, English, Justin G, Glaudin, Alexis M, Krumm, Brian E, Slocum, Samuel T, Che, Tao, Gavin, Ariana C, McCorvy, John D, Roth, Bryan L, Strachan, Ryan T
Published in Nature chemical biology (01.08.2020)
Published in Nature chemical biology (01.08.2020)
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Journal Article
Structure of a Hallucinogen-Activated Gq-Coupled 5-HT2A Serotonin Receptor
Kim, Kuglae, Che, Tao, Panova, Ouliana, DiBerto, Jeffrey F., Lyu, Jiankun, Krumm, Brian E., Wacker, Daniel, Robertson, Michael J., Seven, Alpay B., Nichols, David E., Shoichet, Brian K., Skiniotis, Georgios, Roth, Bryan L.
Published in Cell (17.09.2020)
Published in Cell (17.09.2020)
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Journal Article
Molecular insights into psychedelic drug action
Slocum, Samuel T., DiBerto, Jeffrey F., Roth, Bryan L.
Published in Journal of neurochemistry (01.07.2022)
Published in Journal of neurochemistry (01.07.2022)
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Journal Article
Structure, function and pharmacology of human itch GPCRs
Cao, Can, Kang, Hye Jin, Singh, Isha, Chen, He, Zhang, Chengwei, Ye, Wenlei, Hayes, Byron W, Liu, Jing, Gumpper, Ryan H, Bender, Brian J, Slocum, Samuel T, Krumm, Brian E, Lansu, Katherine, McCorvy, John D, Kroeze, Wesley K, English, Justin G, DiBerto, Jeffrey F, Olsen, Reid H J, Huang, Xi-Ping, Zhang, Shicheng, Liu, Yongfeng, Kim, Kuglae, Karpiak, Joel, Jan, Lily Y, Abraham, Soman N, Jin, Jian, Shoichet, Brian K, Fay, Jonathan F, Roth, Bryan L
Published in Nature (London) (02.12.2021)
Published in Nature (London) (02.12.2021)
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Journal Article
Nanobody-enabled monitoring of kappa opioid receptor states
Che, Tao, English, Justin, Krumm, Brian E, Kim, Kuglae, Pardon, Els, Olsen, Reid H J, Wang, Sheng, Zhang, Shicheng, Diberto, Jeffrey F, Sciaky, Noah, Carroll, F Ivy, Steyaert, Jan, Wacker, Daniel, Roth, Bryan L
Published in Nature communications (02.03.2020)
Published in Nature communications (02.03.2020)
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Journal Article
Structures of the entire human opioid receptor family
Wang, Yue, Zhuang, Youwen, DiBerto, Jeffrey F., Zhou, X. Edward, Schmitz, Gavin P., Yuan, Qingning, Jain, Manish K., Liu, Weiyi, Melcher, Karsten, Jiang, Yi, Roth, Bryan L., Xu, H. Eric
Published in Cell (19.01.2023)
Published in Cell (19.01.2023)
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Journal Article
Insights into distinct signaling profiles of the µOR activated by diverse agonists
Qu, Qianhui, Huang, Weijiao, Aydin, Deniz, Paggi, Joseph M, Seven, Alpay B, Wang, Haoqing, Chakraborty, Soumen, Che, Tao, DiBerto, Jeffrey F, Robertson, Michael J, Inoue, Asuka, Suomivuori, Carl-Mikael, Roth, Bryan L, Majumdar, Susruta, Dror, Ron O, Kobilka, Brian K, Skiniotis, Georgios
Published in Nature chemical biology (01.04.2023)
Published in Nature chemical biology (01.04.2023)
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Journal Article
Serotonin engages an anxiety and fear-promoting circuit in the extended amygdala
Marcinkiewcz, Catherine A, Mazzone, Christopher M, D'Agostino, Giuseppe, Halladay, Lindsay R, Hardaway, J Andrew, DiBerto, Jeffrey F, Navarro, Montserrat, Burnham, Nathan, Cristiano, Claudia, Dorrier, Cayce E, Tipton, Gregory J, Ramakrishnan, Charu, Kozicz, Tamas, Deisseroth, Karl, Thiele, Todd E, McElligott, Zoe A, Holmes, Andrew, Heisler, Lora K, Kash, Thomas L
Published in Nature (London) (01.09.2016)
Published in Nature (London) (01.09.2016)
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Journal Article
Bespoke library docking for 5-HT2A receptor agonists with antidepressant activity
Kaplan, Anat Levit, Confair, Danielle N., Kim, Kuglae, Barros-Álvarez, Ximena, Rodriguiz, Ramona M., Yang, Ying, Kweon, Oh Sang, Che, Tao, McCorvy, John D., Kamber, David N., Phelan, James P., Martins, Luan Carvalho, Pogorelov, Vladimir M., DiBerto, Jeffrey F., Slocum, Samuel T., Huang, Xi-Ping, Kumar, Jain Manish, Robertson, Michael J., Panova, Ouliana, Seven, Alpay B., Wetsel, Autumn Q., Wetsel, William C., Irwin, John J., Skiniotis, Georgios, Shoichet, Brian K., Roth, Bryan L., Ellman, Jonathan A.
Published in Nature (London) (20.10.2022)
Published in Nature (London) (20.10.2022)
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Journal Article
Sex differences in the behavioral sequelae of chronic ethanol exposure
Jury, Nicholas J, DiBerto, Jeffrey F, Kash, Thomas L, Holmes, Andrew
Published in Alcohol (Fayetteville, N.Y.) (01.02.2017)
Published in Alcohol (Fayetteville, N.Y.) (01.02.2017)
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Journal Article
Chronic intermittent ethanol exposure dysregulates a GABAergic microcircuit in the bed nucleus of the stria terminalis
Pati, Dipanwita, Marcinkiewcz, Catherine A., DiBerto, Jeffrey F., Cogan, Elizabeth S., McElligott, Zoe A., Kash, Thomas L.
Published in Neuropharmacology (15.05.2020)
Published in Neuropharmacology (15.05.2020)
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Journal Article
Structure-based design of bitopic ligands for the µ-opioid receptor
Faouzi, Abdelfattah, Wang, Haoqing, Zaidi, Saheem A, DiBerto, Jeffrey F, Che, Tao, Qu, Qianhui, Robertson, Michael J, Madasu, Manish K, El Daibani, Amal, Varga, Balazs R, Zhang, Tiffany, Ruiz, Claudia, Liu, Shan, Xu, Jin, Appourchaux, Kevin, Slocum, Samuel T, Eans, Shainnel O, Cameron, Michael D, Al-Hasani, Ream, Pan, Ying Xian, Roth, Bryan L, McLaughlin, Jay P, Skiniotis, Georgios, Katritch, Vsevolod, Kobilka, Brian K, Majumdar, Susruta
Published in Nature (London) (26.01.2023)
Published in Nature (London) (26.01.2023)
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Journal Article
The G protein-biased κ-opioid receptor agonist RB-64 is analgesic with a unique spectrum of activities in vivo
White, Kate L, Robinson, J Elliott, Zhu, Hu, DiBerto, Jeffrey F, Polepally, Prabhakar R, Zjawiony, Jordan K, Nichols, David E, Malanga, C J, Roth, Bryan L
Published in The Journal of pharmacology and experimental therapeutics (01.01.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2015)
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Journal Article
The paraventricular thalamus provides a polysynaptic brake on limbic CRF neurons to sex-dependently blunt binge alcohol drinking and avoidance behavior in mice
Levine, Olivia B, Skelly, Mary Jane, Miller, John D, Rivera-Irizarry, Jean K, Rowson, Sydney A, DiBerto, Jeffrey F, Rinker, Jennifer A, Thiele, Todd E, Kash, Thomas L, Pleil, Kristen E
Published in Nature communications (23.08.2021)
Published in Nature communications (23.08.2021)
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Journal Article
Structural insights into the human niacin receptor HCA2-Gi signalling complex
Yang, Yang, Kang, Hye Jin, Gao, Ruogu, Wang, Jingjing, Han, Gye Won, DiBerto, Jeffrey F, Wu, Lijie, Tong, Jiahui, Qu, Lu, Wu, Yiran, Pileski, Ryan, Li, Xuemei, Zhang, Xuejun Cai, Zhao, Suwen, Kenakin, Terry, Wang, Quan, Stevens, Raymond C, Peng, Wei, Roth, Bryan L, Rao, Zihe, Liu, Zhi-Jie
Published in Nature communications (27.03.2023)
Published in Nature communications (27.03.2023)
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Journal Article
Manipulations of Central Amygdala Neurotensin Neurons Alter the Consumption of Ethanol and Sweet Fluids in Mice
Torruella-Suárez, María Luisa, Vandenberg, Jessica R, Cogan, Elizabeth S, Tipton, Gregory J, Teklezghi, Adonay, Dange, Kedar, Patel, Gunjan K, McHenry, Jenna A, Hardaway, J Andrew, Kantak, Pranish A, Crowley, Nicole A, DiBerto, Jeffrey F, Faccidomo, Sara P, Hodge, Clyde W, Stuber, Garret D, McElligott, Zoé A
Published in The Journal of neuroscience (15.01.2020)
Published in The Journal of neuroscience (15.01.2020)
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Journal Article
A Novel Mitragynine Analog with Low-Efficacy Mu Opioid Receptor Agonism Displays Antinociception with Attenuated Adverse Effects
Chakraborty, Soumen, DiBerto, Jeffrey F, Faouzi, Abdelfattah, Bernhard, Sarah M, Gutridge, Anna M, Ramsey, Steven, Zhou, Yuchen, Provasi, Davide, Nuthikattu, Nitin, Jilakara, Rahul, Nelson, Melissa N. F, Asher, Wesley B, Eans, Shainnel O, Wilson, Lisa L, Chintala, Satyanarayana M, Filizola, Marta, van Rijn, Richard M, Margolis, Elyssa B, Roth, Bryan L, McLaughlin, Jay P, Che, Tao, Sames, Dalibor, Javitch, Jonathan A, Majumdar, Susruta
Published in Journal of medicinal chemistry (23.09.2021)
Published in Journal of medicinal chemistry (23.09.2021)
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