Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin‐Targeted Conjugate
Raposo Moreira Dias, André, Pina, Arianna, Dean, Amelia, Lerchen, Hans‐Georg, Caruso, Michele, Gasparri, Fabio, Fraietta, Ivan, Troiani, Sonia, Arosio, Daniela, Belvisi, Laura, Pignataro, Luca, Dal Corso, Alberto, Gennari, Cesare
Published in Chemistry : a European journal (01.02.2019)
Published in Chemistry : a European journal (01.02.2019)
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Journal Article
Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery
Borbély, Adina, Figueras, Eduard, Martins, Ana, Bodero, Lizeth, Raposo Moreira Dias, André, López Rivas, Paula, Pina, Arianna, Arosio, Daniela, Gallinari, Paola, Frese, Marcel, Steinkühler, Christian, Gennari, Cesare, Piarulli, Umberto, Sewald, Norbert
Published in ChemistryOpen (Weinheim) (01.06.2019)
Published in ChemistryOpen (Weinheim) (01.06.2019)
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Journal Article
Multivalency Increases the Binding Strength of RGD Peptidomimetic‐Paclitaxel Conjugates to Integrin αVβ3
Raposo Moreira Dias, André, Pina, Arianna, Dal Corso, Alberto, Arosio, Daniela, Belvisi, Laura, Pignataro, Luca, Caruso, Michele, Gennari, Cesare
Published in Chemistry : a European journal (17.10.2017)
Published in Chemistry : a European journal (17.10.2017)
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Journal Article
Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin αVβ3
Raposo Moreira Dias, André, Bodero, Lizeth, Martins, Ana, Arosio, Daniela, Gazzola, Silvia, Belvisi, Laura, Pignataro, Luca, Steinkühler, Christian, Dal Corso, Alberto, Gennari, Cesare, Piarulli, Umberto
Published in ChemMedChem (06.05.2019)
Published in ChemMedChem (06.05.2019)
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Journal Article
Conjugates of Cryptophycin and RGD or iso DGR Peptidomimetics for Targeted Drug Delivery
Borbély, Adina, Figueras, Eduard, Martins, Ana, Bodero, Lizeth, Raposo Moreira Dias, André, López Rivas, Paula, Pina, Arianna, Arosio, Daniela, Gallinari, Paola, Frese, Marcel, Steinkühler, Christian, Gennari, Cesare, Piarulli, Umberto, Sewald, Norbert
Published in ChemistryOpen (Weinheim) (01.06.2019)
Published in ChemistryOpen (Weinheim) (01.06.2019)
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Journal Article
Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and αVβ3‐Integrin Ligands for Tumor Targeting
López Rivas, Paula, Ranđelović, Ivan, Raposo Moreira Dias, André, Pina, Arianna, Arosio, Daniela, Tóvári, József, Mező, Gábor, Dal Corso, Alberto, Pignataro, Luca, Gennari, Cesare
Published in European journal of organic chemistry (22.06.2018)
Published in European journal of organic chemistry (22.06.2018)
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Journal Article
Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α V β 3
Raposo Moreira Dias, André, Pina, Arianna, Dal Corso, Alberto, Arosio, Daniela, Belvisi, Laura, Pignataro, Luca, Caruso, Michele, Gennari, Cesare
Published in Chemistry : a European journal (17.10.2017)
Published in Chemistry : a European journal (17.10.2017)
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Journal Article
Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin (V3)
Dias, Andre Raposo Moreira, Bodero, Lizeth, Martins, Ana, Arosio, Daniela, Gazzola, Silvia, Belvisi, Laura, Pignataro, Luca, Steinkuhler, Christian, Dal Corso, Alberto, Gennari, Cesare, Piarulli, Umberto
Published in ChemMedChem (06.05.2019)
Published in ChemMedChem (06.05.2019)
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Journal Article
Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and V3-Integrin Ligands for Tumor Targeting
Rivas, Paula Lopez, Randelovic, Ivan, Dias, Andre Raposo Moreira, Pina, Arianna, Arosio, Daniela, Tovari, Jozsef, Mezo, Gabor, Dal Corso, Alberto, Pignataro, Luca, Gennari, Cesare
Published in European journal of organic chemistry (22.06.2018)
Published in European journal of organic chemistry (22.06.2018)
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Benchmarking Strategies of Sustainable Process Chemistry Development: Human-Based, Machine Learning, and Quantum Mechanics
Almeida, A. Filipa, Branco, Sofia, Carvalho, Luisa C. R., Dias, Andre Raposo Moreira, Leitão, Emília P. T., Loureiro, Rui M. S., Lucas, Susana D., Mendonça, Ricardo F., Oliveira, Rudi, Rocha, Inês L. D., Sardinha, Joao, Silva, Saúl, Sobral, Luís M. S., Lourenço, Nuno M. T., Valente, Pedro C.
Published in Organic process research & development (19.07.2024)
Published in Organic process research & development (19.07.2024)
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Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin α V β 3
Raposo Moreira Dias, André, Bodero, Lizeth, Martins, Ana, Arosio, Daniela, Gazzola, Silvia, Belvisi, Laura, Pignataro, Luca, Steinkühler, Christian, Dal Corso, Alberto, Gennari, Cesare, Piarulli, Umberto
Published in ChemMedChem (06.05.2019)
Published in ChemMedChem (06.05.2019)
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Journal Article
Frontispiece: Multivalency Increases the Binding Strength of RGD Peptidomimetic‐Paclitaxel Conjugates to Integrin αVβ3
Raposo Moreira Dias, André, Pina, Arianna, Dal Corso, Alberto, Arosio, Daniela, Belvisi, Laura, Pignataro, Luca, Caruso, Michele, Gennari, Cesare
Published in Chemistry : a European journal (17.10.2017)
Published in Chemistry : a European journal (17.10.2017)
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Journal Article
Frontispiece: Multivalency Increases the Binding Strength of RGD Peptidomimetic‐Paclitaxel Conjugates to Integrin α V β 3
Raposo Moreira Dias, André, Pina, Arianna, Dal Corso, Alberto, Arosio, Daniela, Belvisi, Laura, Pignataro, Luca, Caruso, Michele, Gennari, Cesare
Published in Chemistry : a European journal (17.10.2017)
Published in Chemistry : a European journal (17.10.2017)
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Journal Article
Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and α V β 3 ‐Integrin Ligands for Tumor Targeting
López Rivas, Paula, Ranđelović, Ivan, Raposo Moreira Dias, André, Pina, Arianna, Arosio, Daniela, Tóvári, József, Mező, Gábor, Dal Corso, Alberto, Pignataro, Luca, Gennari, Cesare
Published in European journal of organic chemistry (22.06.2018)
Published in European journal of organic chemistry (22.06.2018)
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Journal Article
Synthesis and Biological Evaluation of RGD and iso DGR–Monomethyl Auristatin Conjugates Targeting Integrin α V β 3
Raposo Moreira Dias, André, Bodero, Lizeth, Martins, Ana, Arosio, Daniela, Gazzola, Silvia, Belvisi, Laura, Pignataro, Luca, Steinkühler, Christian, Dal Corso, Alberto, Gennari, Cesare, Piarulli, Umberto
Published in ChemMedChem (06.05.2019)
Published in ChemMedChem (06.05.2019)
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Journal Article