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Ultra-High-Throughput Acoustic Droplet Ejection-Open Port Interface-Mass Spectrometry for Parallel Medicinal Chemistry
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Early Clinical Development of Lufotrelvir as a Potential Therapy for COVID-19
Allais, Christophe, Bernhardson, David, Brown, Adam R., Chinigo, Gary M., Desrosiers, Jean-Nicolas, DiRico, Kenneth J., Hotham, Ian, Jones, Brian P., Kulkarni, Samir A., Lewis, Chad A., Lira, Ricardo, Loach, Richard P., Morse, Peter D., Mousseau, James J., Perry, Matthew A., Peng, Zhihui, Place, David W., Rane, Anil M., Samp, Lacey, Singer, Robert A., Wang, Zheng, Weisenburger, Gerald A., Yayla, Hatice G., Zanghi, Joseph M.
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Metabolism-Directed Design of Oxetane-Containing Arylsulfonamide Derivatives as γ-Secretase Inhibitors
Stepan, Antonia F, Karki, Kapil, McDonald, W. Scott, Dorff, Peter H, Dutra, Jason K, DiRico, Kenneth J, Won, Annie, Subramanyam, Chakrapani, Efremov, Ivan V, O’Donnell, Christopher J, Nolan, Charles E, Becker, Stacey L, Pustilnik, Leslie R, Sneed, Blossom, Sun, Hao, Lu, Yasong, Robshaw, Ashley E, Riddell, David, O'Sullivan, Theresa J, Sibley, Evelyn, Capetta, Steven, Atchison, Kevin, Hallgren, Andrew J, Miller, Emily, Wood, Anthony, Obach, R. Scott
Published in Journal of medicinal chemistry (24.11.2011)
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Freeman-Cook, Kevin D, Amor, Paul, Bader, Scott, Buzon, Leanne M, Coffey, Steven B, Corbett, Jeffrey W, Dirico, Kenneth J, Doran, Shawn D, Elliott, Richard L, Esler, William, Guzman-Perez, Angel, Henegar, Kevin E, Houser, Janet A, Jones, Christopher S, Limberakis, Chris, Loomis, Katherine, McPherson, Kirk, Murdande, Sharad, Nelson, Kendra L, Phillion, Dennis, Pierce, Betsy S, Song, Wei, Sugarman, Eliot, Tapley, Susan, Tu, Meihua, Zhao, Zhengrong
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Humphries, Paul S., Benbow, John W., Bonin, Paul D., Boyer, David, Doran, Shawn D., Frisbie, Richard K., Piotrowski, David W., Balan, Gayatri, Bechle, Bruce M., Conn, Edward L., Dirico, Kenneth J., Oliver, Robert M., Soeller, Walter C., Southers, James A., Yang, Xiaojing
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Corbett, Jeffrey W., Freeman-Cook, Kevin D., Elliott, Richard, Vajdos, Felix, Rajamohan, Francis, Kohls, Darcy, Marr, Eric, Zhang, Hailong, Tong, Liang, Tu, Meihua, Murdande, Sharad, Doran, Shawn D., Houser, Janet A., Song, Wei, Jones, Christopher J., Coffey, Steven B., Buzon, Leanne, Minich, Martha L., Dirico, Kenneth J., Tapley, Susan, Kirk McPherson, R., Sugarman, Eliot, James Harwood, H., Esler, William
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Discovery of triazolopyrimidine-based PDE8B inhibitors: Exceptionally ligand-efficient and lipophilic ligand-efficient compounds for the treatment of diabetes
DeNinno, Michael P., Wright, Stephen W., Etienne, John B., Olson, Thanh V., Rocke, Benjamin N., Corbett, Jeffrey W., Kung, Daniel W., DiRico, Kenneth J., Andrews, Kim M., Millham, Michele L., Parker, Janice C., Esler, William, van Volkenburg, Maria, Boyer, David D., Houseknecht, Karen L., Doran, Shawn D.
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Published in The Journal of biological chemistry (02.12.2011)
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DeNinno, Michael P, Masamune, Hiroko, Chenard, Lois K, DiRico, Kenneth J, Eller, Cynthia, Etienne, John B, Tickner, Jeanene E, Kennedy, Scott P, Knight, Delvin R, Kong, Jimmy, Oleynek, Joseph J, Tracey, W. Ross, Hill, Roger J
Published in Journal of medicinal chemistry (30.01.2003)
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DENINNO, Michael P, MASAMUNE, Hiroko, OLEYNEK, Joseph J, TRACEY, W. Ross, HILL, Roger J, CHENARD, Lois K, DIRICO, Kenneth J, ELLER, Cynthia, ETIENNE, John B, TICKNER, Jeanene E, KENNEDY, Scott P, KNIGHT, Delvin R, KONG, Jimmy
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Year of Publication 01.10.2019
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Photorearrangements of acyclic conjugated enynes: a photochemical analog of the Bergman rearrangement
Zheng, Manli, DiRico, Kenneth J, Kirchhoff, Mary M, Phillips, Kristine M, Cuff, Lisa M, Johnson, Richard P
Published in Journal of the American Chemical Society (01.12.1993)
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Published in Tetrahedron letters (06.05.2009)
Published in Tetrahedron letters (06.05.2009)
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Discovery Tactics To Mitigate Toxicity Risks Due to Reactive Metabolite Formation with 2-(2-Hydroxyaryl)-5-(trifluoromethyl)pyrido[4,3-d]pyrimidin-4(3H)-one Derivatives, Potent Calcium-Sensing Receptor Antagonists and Clinical Candidate(s) for the Treatment of Osteoporosis
Kalgutkar, Amit S, Griffith, David A, Ryder, Tim, Sun, Hao, Miao, Zhuang, Bauman, Jonathan N, Didiuk, Mary T, Frederick, Kosea S, Zhao, Sabrina X, Prakash, Chandra, Soglia, John R, Bagley, Scott W, Bechle, Bruce M, Kelley, Ryan M, Dirico, Kenneth, Zawistoski, Michael, Li, Jianke, Oliver, Robert, Guzman-Perez, Angel, Liu, Kevin K. C, Walker, Daniel P, Benbow, John W, Morris, Joel
Published in Chemical research in toxicology (21.06.2010)
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Synthesis of Unprotected Carboxy Indazoles via Pd-Catalyzed Carbonylation
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Published in Synthetic communications (01.07.2012)
Published in Synthetic communications (01.07.2012)
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