CP-481,715, a Potent and Selective CCR1 Antagonist with Potential Therapeutic Implications for Inflammatory Diseases
Gladue, Ronald P., Tylaska, Laurie A., Brissette, William H., Lira, Paul D., Kath, John C., Poss, Christopher S., Brown, Matthew F., Paradis, Timothy J., Conklyn, Maryrose J., Ogborne, Kevin T., McGlynn, Molly A., Lillie, Brett M., DiRico, Amy P., Mairs, Erin N., McElroy, Eric B., Martin, William H., Stock, Ingrid A., Shepard, Richard M., Showell, Henry J., Neote, Kuldeep
Published in The Journal of biological chemistry (17.10.2003)
Published in The Journal of biological chemistry (17.10.2003)
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The discovery of structurally novel CCR1 antagonists derived from a hydroxyethylene peptide isostere template
KATH, John C, DIRICO, Amy P, GLADUE, Ronald P, MARTIN, William H, MCELROY, Eric B, STOCK, Ingrid A, TYLASKA, Laurie A, DEYE ZHENG
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Novel CCR1 antagonists with improved metabolic stability
BROWN, Matthew F, AVERY, Mike, LIRA, Paul D, LILLIE, Brett M, LUNDQUIST, Greg D, MAIRS, Erin N, MCELROY, Eric B, MCGLYNN, Molly A, PARADIS, Timothy J, POSS, Christopher S, ROSSULEK, Michelle I, SHEPARD, Richard M, BRISSETTE, William H, SIMS, Jeff, STRELEVITZ, Timothy J, TRUESDELL, Susan, TYLASKA, Laurie A, YOON, Kwansik, DEYE ZHENG, CHANG, J. H, COLIZZA, Kevin, CONKLYN, Maryrose, DIRICO, Amy P, GLADUE, Ronald P, KATH, John C, KRUEGER, Suzanne S
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Journal Article
Potent small molecule CCR1 antagonists
KATH, John C, BRISSETTE, William H, MARTIN, William H, MCELROY, Eric B, MCGLYNN, Molly A, PARADIS, Timothy J, POSS, Christopher S, STOCK, Ingrid A, TYLASKA, Laurie A, DEYE ZHENG, BROWN, Matthew F, CONKLYN, Maryrose, DIRICO, Amy P, DORFF, Peter, GLADUE, Ronald P, LILLIE, Brett M, LIRA, Paul D, MAIRS, Erin N
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Journal Article
The Discovery of Structurally Novel CCR1 Antagonists Derived from a Hydroxyethylene Peptide Isostere Template
Kath, John C., DiRico, Amy P., Gladue, Ronald P., Martin, William H., McElroy, Eric B., Stock, Ingrid A., Tylaska, Laurie A., Zheng, Deye
Published in ChemInform (31.08.2004)
Published in ChemInform (31.08.2004)
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